General Information of the Compound
Compound ID
CP0467290
Compound Name
5-(2-(2-cyclopropoxy-5-(trifluoromethoxy)benzylamino)-1-phenyl-8-aza-bicyclo[3.2.1]octan-6-yl)-2H-1,2,4-triazol-3(4H)-one
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Structure
Formula
C26H28F3N5O3
Molecular Weight
515.536
Canonical SMILES
FC(F)(F)Oc1ccc(OC2CC2)c(CNC2CCC3NC2(CC3c2n[nH]c(=O)[nH]2)c2ccccc2)c1
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InChI
InChI=1S/C26H28F3N5O3/c27-26(28,29)37-18-8-10-21(36-17-6-7-17)15(12-18)14-30-22-11-9-20-19(23-31-24(35)34-33-23)13-25(22,32-20)16-4-2-1-3-5-16/h1-5,8,10,12,17,19-20,22,30,32H,6-7,9,11,13-14H2,(H2,31,33,34,35)
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InChIKey
QKMNCMIKEOYLQG-UHFFFAOYSA-N
Physicochemical Property
logP
3.831
Rotatable Bonds
8
Heavy Atom Count
37
Polar Areas
104.06
Hydrogen Bond Donor Count
4
Hydrogen Bond Acceptor Count
6
Complexity
37

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 136094778
ChEMBL ID
CHEMBL379010
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00897, Potassium voltage-gated channel subfamily H member 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 5800 nM
   TI
   LI
   LO
   TS
Protein ID: PT01410, Substance-P receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 0.61 nM
   TI
   LI
   LO
   TS