General Information of the Compound
Compound ID
CP0459717
Compound Name
6-[(3S,4S)-4-amino-3-methyl-2-oxa-8-azaspiro[4.5]decan-8-yl]-3-[3-chloro-2-(cyclobutylamino)pyridin-4-yl]-5-methyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
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Structure
Formula
C24H31ClN8O2
Molecular Weight
499.019
Canonical SMILES
C[C@@H]1OCC2(CCN(CC2)c2nc3[nH]nc(-c4ccnc(NC5CCC5)c4Cl)c3c(=O)n2C)[C@@H]1N
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InChI
InChI=1S/C24H31ClN8O2/c1-13-19(26)24(12-35-13)7-10-33(11-8-24)23-29-20-16(22(34)32(23)2)18(30-31-20)15-6-9-27-21(17(15)25)28-14-4-3-5-14/h6,9,13-14,19H,3-5,7-8,10-12,26H2,1-2H3,(H,27,28)(H,30,31)/t13-,19+/m0/s1
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InChIKey
JMFFJZHRARAACU-ORAYPTAESA-N
Physicochemical Property
logP
2.669
Rotatable Bonds
4
Heavy Atom Count
35
Polar Areas
126.98
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
9
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 124148125
ChEMBL ID
CHEMBL4450282
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01346, Tyrosine-protein phosphatase non-receptor type 11
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000269 KYSE-520 Homo sapiens (Human)  1
1
IC50 = 260 nM
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Cell Viability or Cytotoxicity Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000269 KYSE-520 Homo sapiens (Human)  1
1
IC50 = 380 nM
   TI
   LI
   LO
   TS