General Information of the Compound
Compound ID
CP0453189
Compound Name
4-{6-Methoxy-7-[2-(4-methyl-piperazin-1-yl)-ethoxy]-quinazolin-4-yl}-piperazine-1-carboxylic acid (4-cyano-phenyl)-amide
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Structure
Formula
C28H34N8O3
Molecular Weight
530.633
Canonical SMILES
COc1cc2c(ncnc2cc1OCCN1CCN(C)CC1)N1CCN(CC1)C(=O)Nc1ccc(cc1)C#N
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InChI
InChI=1S/C28H34N8O3/c1-33-7-9-34(10-8-33)15-16-39-26-18-24-23(17-25(26)38-2)27(31-20-30-24)35-11-13-36(14-12-35)28(37)32-22-5-3-21(19-29)4-6-22/h3-6,17-18,20H,7-16H2,1-2H3,(H,32,37)
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InChIKey
HYJFRKGSJGMOJJ-UHFFFAOYSA-N
Physicochemical Property
logP
2.49038
Rotatable Bonds
7
Heavy Atom Count
39
Polar Areas
110.09
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
9
Complexity
39

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 10918469
SID: 15968360
ChEMBL ID
CHEMBL125445
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00844, Platelet-derived growth factor receptor beta
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000197 MG-63 Homo sapiens (Human)  2
1
IC50 = 662 nM
   TI
   LI
   LO
   TS
2
IC50 = 750 nM
   TI
   LI
   LO
   TS