General Information of the Compound
Compound ID
CP0451480
Compound Name
5-(6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-4-yloxy)-N-[5-[1-(trifluoromethyl)cyclopropyl]-1,2-oxazol-3-yl]indole-1-carboxamide
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Structure
Formula
C22H17F3N6O3
Molecular Weight
470.411
Canonical SMILES
FC(F)(F)C1(CC1)c1cc(NC(=O)n2ccc3cc(Oc4ncnc5CNCc45)ccc23)no1
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InChI
InChI=1S/C22H17F3N6O3/c23-22(24,25)21(4-5-21)17-8-18(30-34-17)29-20(32)31-6-3-12-7-13(1-2-16(12)31)33-19-14-9-26-10-15(14)27-11-28-19/h1-3,6-8,11,26H,4-5,9-10H2,(H,29,30,32)
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InChIKey
NLPLUYRSIUXZHN-UHFFFAOYSA-N
Physicochemical Property
logP
4.4889
Rotatable Bonds
4
Heavy Atom Count
34
Polar Areas
107.1
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
8
Complexity
34

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 59394176
ChEMBL ID
CHEMBL4102438
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00864, Vascular endothelial growth factor receptor 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  1
1
IC50 = 5 nM
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