General Information of the Compound
Compound ID
CP0449451
Compound Name
3-[cyclopropylmethyl-[2-(5-fluoro-1H-indol-3-yl)ethyl]amino]-8-fluoro-3,4-dihydro-2H-chromene-5-carboxamide
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Structure
Formula
C24H25F2N3O2
Molecular Weight
425.479
Canonical SMILES
NC(=O)c1ccc(F)c2OCC(Cc12)N(CCc1c[nH]c2ccc(F)cc12)CC1CC1
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InChI
InChI=1S/C24H25F2N3O2/c25-16-3-6-22-19(9-16)15(11-28-22)7-8-29(12-14-1-2-14)17-10-20-18(24(27)30)4-5-21(26)23(20)31-13-17/h3-6,9,11,14,17,28H,1-2,7-8,10,12-13H2,(H2,27,30)
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InChIKey
TWAQVUKMYNLEQM-UHFFFAOYSA-N
Physicochemical Property
logP
3.8032
Rotatable Bonds
7
Heavy Atom Count
31
Polar Areas
71.35
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
3
Complexity
31

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 11418868
SID: 16515449
ChEMBL ID
CHEMBL379298
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00819, 5-hydroxytryptamine receptor 1A
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 97 nM
   TI
   LI
   LO
   TS
2
Ki = 7.3 nM
   TI
   LI
   LO
   TS
Protein ID: PT00871, Sodium-dependent serotonin transporter
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000232 JAR Homo sapiens (Human)  1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS