General Information of the Compound
Compound ID
CP0442377
Compound Name
4-[3-Cyano-6-methoxy-7-(3-piperidin-1-yl-propoxy)-quinolin-4-yl]-piperazine-1-carbothioic acid (6-phenyl-pyridin-3-ylmethyl)-amide
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Structure
Formula
C36H41N7O2S
Molecular Weight
635.838
Canonical SMILES
COc1cc2c(N3CCN(CC3)C(=S)NCc3ccc(nc3)-c3ccccc3)c(cnc2cc1OCCCN1CCCCC1)C#N
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InChI
InChI=1S/C36H41N7O2S/c1-44-33-21-30-32(22-34(33)45-20-8-15-41-13-6-3-7-14-41)39-26-29(23-37)35(30)42-16-18-43(19-17-42)36(46)40-25-27-11-12-31(38-24-27)28-9-4-2-5-10-28/h2,4-5,9-12,21-22,24,26H,3,6-8,13-20,25H2,1H3,(H,40,46)
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InChIKey
FJCGGUSGCZXDHJ-UHFFFAOYSA-N
Physicochemical Property
logP
5.62858
Rotatable Bonds
10
Heavy Atom Count
46
Polar Areas
89.78
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
8
Complexity
46

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 44394634
ChEMBL ID
CHEMBL184642
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00844, Platelet-derived growth factor receptor beta
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000197 MG-63 Homo sapiens (Human)  2
1
IC50 = 10 nM
   TI
   LI
   LO
   TS
2
IC50 = 100 nM
   TI
   LI
   LO
   TS