General Information of the Compound
Compound ID
CP0427983
Compound Name
ethyl 3-[[benzyl-[2-oxo-2-[[(2S)-1-oxo-1-(3-phenylprop-2-ynylamino)propan-2-yl]amino]ethyl]amino]methyl]-8-[(2,6-difluorophenyl)methyl]-2-[4-(ethylcarbamoylamino)phenyl]-5-oxoimidazo[1,2-a]pyrimidine-6-carboxylate
    Show/Hide
Structure
Formula
C47H46F2N8O6
Molecular Weight
856.931
Canonical SMILES
CCNC(=O)Nc1ccc(cc1)-c1nc2n(Cc3c(F)cccc3F)cc(C(=O)OCC)c(=O)n2c1CN(CC(=O)N[C@@H](C)C(=O)NCC#Cc1ccccc1)Cc1ccccc1
    Show/Hide
InChI
InChI=1S/C47H46F2N8O6/c1-4-50-46(62)53-35-23-21-34(22-24-35)42-40(57-44(60)37(45(61)63-5-2)28-56(47(57)54-42)27-36-38(48)19-12-20-39(36)49)29-55(26-33-16-10-7-11-17-33)30-41(58)52-31(3)43(59)51-25-13-18-32-14-8-6-9-15-32/h6-12,14-17,19-24,28,31H,4-5,25-27,29-30H2,1-3H3,(H,51,59)(H,52,58)(H2,50,53,62)/t31-/m0/s1
    Show/Hide
InChIKey
GKRNHZOOABIXOG-HKBQPEDESA-N
Physicochemical Property
logP
5.4824
Rotatable Bonds
16
Heavy Atom Count
63
Polar Areas
168.17
Hydrogen Bond Donor Count
4
Hydrogen Bond Acceptor Count
10
Complexity
63

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 44451397
ChEMBL ID
CHEMBL259220
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01836, Gonadotropin-releasing hormone receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
IC50 = 1100 nM
   TI
   LI
   LO
   TS
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 1600 nM
   TI
   LI
   LO
   TS