General Information of the Compound
Compound ID
CP0409412
Compound Name
2-Oxo-3-{1-[4-(1,1,3-trioxo-1,3-dihydro-1lambda*6*-benzo[d]isothiazol-2-yl)-butyl]-piperidin-4-yl}-2,3-dihydro-benzooxazole-6-carboxylic acid methyl ester
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Structure
Formula
C25H27N3O7S
Molecular Weight
513.572
Canonical SMILES
COC(=O)c1ccc2n(C3CCN(CCCCN4C(=O)c5ccccc5S4(=O)=O)CC3)c(=O)oc2c1
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InChI
InChI=1S/C25H27N3O7S/c1-34-24(30)17-8-9-20-21(16-17)35-25(31)28(20)18-10-14-26(15-11-18)12-4-5-13-27-23(29)19-6-2-3-7-22(19)36(27,32)33/h2-3,6-9,16,18H,4-5,10-15H2,1H3
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InChIKey
JWKSOUFQGFGEKE-UHFFFAOYSA-N
Physicochemical Property
logP
2.6429
Rotatable Bonds
7
Heavy Atom Count
36
Polar Areas
119.13
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
9
Complexity
36

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 19085921
ChEMBL ID
CHEMBL311290
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01089, Alpha-1A adrenergic receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 1033 nM
   TI
   LI
   LO
   TS
Protein ID: PT01007, Alpha-1B adrenergic receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000440 LM Homo sapiens (Human)  1
1
Ki = 1958 nM
   TI
   LI
   LO
   TS
Protein ID: PT01004, Alpha-1D adrenergic receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 3429 nM
   TI
   LI
   LO
   TS