General Information of the Compound
Compound ID
CP0392522
Compound Name
7-Chloro-4-[2-((R)-1-methyl-6-trifluoromethyl-piperidin-2-yl)-ethoxy]-2-oxo-3-((S)-3,4,5-trimethyl-phenyl)-1,2-dihydro-quinoline-6-carboxylic acid pyrimidin-4-ylamide
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Structure
Formula
C32H33ClF3N5O3
Molecular Weight
628.095
Canonical SMILES
CN1[C@H](CCOc2c(-c3cc(C)c(C)c(C)c3)c(=O)[nH]c3cc(Cl)c(cc23)C(=O)Nc2ccncn2)CCC[C@@H]1C(F)(F)F
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InChI
InChI=1S/C32H33ClF3N5O3/c1-17-12-20(13-18(2)19(17)3)28-29(44-11-9-21-6-5-7-26(41(21)4)32(34,35)36)23-14-22(24(33)15-25(23)39-31(28)43)30(42)40-27-8-10-37-16-38-27/h8,10,12-16,21,26H,5-7,9,11H2,1-4H3,(H,39,43)(H,37,38,40,42)/t21-,26+/m0/s1
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InChIKey
ZUTIZSMLCDYNNR-HFZDXXHNSA-N
Physicochemical Property
logP
7.00016
Rotatable Bonds
7
Heavy Atom Count
44
Polar Areas
100.21
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
6
Complexity
44

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 44395463
ChEMBL ID
CHEMBL365366
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01836, Gonadotropin-releasing hormone receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 2 nM
   TI
   LI
   LO
   TS
2
IC50 = 18 nM
   TI
   LI
   LO
   TS