General Information of the Compound
Compound ID
CP0385821
Compound Name
(2R,3S,5R)-2-(2,5-difluorophenyl)-5-[2-[3-(trifluoromethyl)phenyl]sulfonyl-4,6-dihydropyrrolo[3,4-c]pyrazol-5-yl]oxan-3-amine
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Structure
Formula
C23H21F5N4O3S
Molecular Weight
528.503
Canonical SMILES
N[C@H]1C[C@H](CO[C@@H]1c1cc(F)ccc1F)N1Cc2cn(nc2C1)S(=O)(=O)c1cccc(c1)C(F)(F)F
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InChI
InChI=1S/C23H21F5N4O3S/c24-15-4-5-19(25)18(7-15)22-20(29)8-16(12-35-22)31-9-13-10-32(30-21(13)11-31)36(33,34)17-3-1-2-14(6-17)23(26,27)28/h1-7,10,16,20,22H,8-9,11-12,29H2/t16-,20+,22-/m1/s1
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InChIKey
HECNNSAYFGDCAE-QGCDCVKKSA-N
Physicochemical Property
logP
3.5902
Rotatable Bonds
4
Heavy Atom Count
36
Polar Areas
90.45
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
7
Complexity
36

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 127035375
ChEMBL ID
CHEMBL3736067
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00989, Dipeptidyl peptidase 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000013 Sf9 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
Protein ID: PT00907, Dipeptidyl peptidase 4
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000013 Sf9 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 = 1.9 nM
   TI
   LI
   LO
   TS
Protein ID: PT00975, Dipeptidyl peptidase 8
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000053 COS-7 Chlorocebus aethiops (Green monkey)  1
1
IC50 = 27000 nM
   TI
   LI
   LO
   TS