General Information of the Compound
Compound ID
CP0384549
Compound Name
(1S,2S,6R,14R,15R,16R)-16-[(2R)-1-(2-bicyclo[2.2.1]heptanyl)-2-hydroxypropan-2-yl]-5-(cyclopropylmethyl)-15-methoxy-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-trien-11-ol
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Structure
Formula
C33H45NO4
Molecular Weight
519.726
Canonical SMILES
CO[C@]12CC[C@@]3(C[C@@H]1[C@](C)(O)CC1CC4CCC1C4)[C@H]1Cc4ccc(O)c5O[C@@H]2[C@]3(CCN1CC1CC1)c45
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InChI
InChI=1S/C33H45NO4/c1-30(36,16-23-14-20-5-6-21(23)13-20)25-17-31-9-10-33(25,37-2)29-32(31)11-12-34(18-19-3-4-19)26(31)15-22-7-8-24(35)28(38-29)27(22)32/h7-8,19-21,23,25-26,29,35-36H,3-6,9-18H2,1-2H3/t20?,21?,23?,25-,26-,29-,30-,31-,32+,33-/m1/s1
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InChIKey
KMMPJTLXSZEWDK-VAZJWBNESA-N
Physicochemical Property
logP
5.194
Rotatable Bonds
6
Heavy Atom Count
38
Polar Areas
62.16
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
5
Complexity
38

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 56658044
ChEMBL ID
CHEMBL1834413
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01200, Delta-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
EC50 = 49.3 nM
   TI
   LI
   LO
   TS
2
Ki = 7.13 nM
   TI
   LI
   LO
   TS
Protein ID: PT00983, Kappa-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
EC50 = 5.33 nM
   TI
   LI
   LO
   TS
2
Ki = 9.87 nM
   TI
   LI
   LO
   TS
Protein ID: PT01515, Mu-type opioid receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
EC50 = 6.1 nM
   TI
   LI
   LO
   TS
2
Ki = 11.4 nM
   TI
   LI
   LO
   TS
Protein ID: PT01360, Nociceptin receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
EC50 = 111 nM
   TI
   LI
   LO
   TS
2
Ki = 16 nM
   TI
   LI
   LO
   TS