General Information of the Compound
Compound ID
CP0368810
Compound Name
N-[3-[3-chloro-6-[2-methoxy-4-(4-methylpiperazin-1-yl)anilino]pyridin-2-yl]oxyphenyl]prop-2-enamide
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Structure
Formula
C26H28ClN5O3
Molecular Weight
493.995
Canonical SMILES
COc1cc(ccc1Nc1ccc(Cl)c(Oc2cccc(NC(=O)C=C)c2)n1)N1CCN(C)CC1
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InChI
InChI=1S/C26H28ClN5O3/c1-4-25(33)28-18-6-5-7-20(16-18)35-26-21(27)9-11-24(30-26)29-22-10-8-19(17-23(22)34-3)32-14-12-31(2)13-15-32/h4-11,16-17H,1,12-15H2,2-3H3,(H,28,33)(H,29,30)
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InChIKey
VMMYPYDOTNDREB-UHFFFAOYSA-N
Physicochemical Property
logP
5.1558
Rotatable Bonds
8
Heavy Atom Count
35
Polar Areas
78.96
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 152157601
ChEMBL ID
CHEMBL4515293
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02790, Dipeptidyl peptidase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000100 U-937 Homo sapiens (Human)  1
1
IC50 = 537 nM
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