General Information of the Compound
Compound ID
CP0342373
Compound Name
2,4-dimethyl-5-[4-methyl-5-[3-[1-[4-(trifluoromethyl)phenyl]-4-azabicyclo[5.1.0]octan-4-yl]propylsulfanyl]-1,2,4-triazol-3-yl]-1,3-thiazole
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Structure
Formula
C25H30F3N5S2
Molecular Weight
521.678
Canonical SMILES
Cc1nc(C)c(s1)-c1nnc(SCCCN2CCC3CC3(CC2)c2ccc(cc2)C(F)(F)F)n1C
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InChI
InChI=1S/C25H30F3N5S2/c1-16-21(35-17(2)29-16)22-30-31-23(32(22)3)34-14-4-11-33-12-9-20-15-24(20,10-13-33)18-5-7-19(8-6-18)25(26,27)28/h5-8,20H,4,9-15H2,1-3H3
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InChIKey
HIVHEOCGLZASLB-UHFFFAOYSA-N
Physicochemical Property
logP
6.11014
Rotatable Bonds
7
Heavy Atom Count
35
Polar Areas
46.84
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
7
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 52949300
ChEMBL ID
CHEMBL1257926
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01005, D(2) dopamine receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 199.53 nM
   TI
   LI
   LO
   TS
Protein ID: PT00943, D(3) dopamine receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 3.981 nM
   TI
   LI
   LO
   TS