General Information of the Compound
Compound ID
CP0294392
Compound Name
(S)-N-((S)-1-cyano-2-phenylethyl)-3-cyclopropyl-2-((S)-2,2,2-trifluoro-1-(4'-(methylsulfonyl)biphenyl-4-yl)ethylamino)propanamide
    Show/Hide
Structure
Formula
C30H30F3N3O3S
Molecular Weight
569.649
Canonical SMILES
CS(=O)(=O)c1ccc(cc1)-c1ccc(cc1)[C@H](N[C@@H](CC1CC1)C(=O)N[C@@H](Cc1ccccc1)C#N)C(F)(F)F
    Show/Hide
InChI
InChI=1S/C30H30F3N3O3S/c1-40(38,39)26-15-13-23(14-16-26)22-9-11-24(12-10-22)28(30(31,32)33)36-27(18-21-7-8-21)29(37)35-25(19-34)17-20-5-3-2-4-6-20/h2-6,9-16,21,25,27-28,36H,7-8,17-18H2,1H3,(H,35,37)/t25-,27-,28-/m0/s1
    Show/Hide
InChIKey
JNRFQDUMCHRUFL-MYKRZTLLSA-N
Physicochemical Property
logP
5.36988
Rotatable Bonds
11
Heavy Atom Count
40
Polar Areas
99.06
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
5
Complexity
40

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 42633150
SID: 81072152
ChEMBL ID
CHEMBL1289988
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00974, Cathepsin B
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000063 Hep-G2 Homo sapiens (Human)  1
1
IC50 = 231 nM
   TI
   LI
   LO
   TS
Protein ID: PT03764, Cathepsin F
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000972 HIG-82 Oryctolagus cuniculus (Rabbit)  1
1
IC50 = 147 nM
   TI
   LI
   LO
   TS