General Information of the Compound
Compound ID
CP0192479
Compound Name
(5-Chloro-benzo[1,2,5]thiadiazol-4-yl)-(4,5-dihydro-1H-imidazol-2-yl)-amine
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Synonyms
5-Chloro-4-(2-imidazolin-2-ylamino)-2,1,3-benzothiadiazole
5-chloro-4-(2-imidazolin-2-yl-amino)-2,1,3-benzothiadiazole
5-chloro-N-(4,5-dihydro-1H-imidazol-2-yl)-2,1,3-benzothiadiazol-4-amine
Sirdalud
Sirdalud (TN)
Ternelin
Tizanidina
Tizanidina [INN-Spanish]
Tizanidine
Tizanidine (INN)
Tizanidine [INN:BAN]
Tizanidinum
Tizanidinum [INN-Latin]
Zanaflex (TN)
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Structure
Formula
C9H8ClN5S
Molecular Weight
253.718
Canonical SMILES
Clc1ccc2nsnc2c1NC1=NCCN1
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InChI
InChI=1S/C9H8ClN5S/c10-5-1-2-6-8(15-16-14-6)7(5)13-9-11-3-4-12-9/h1-2H,3-4H2,(H2,11,12,13)
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InChIKey
XFYDIVBRZNQMJC-UHFFFAOYSA-N
CAS
51322-75-9
Physicochemical Property
logP
1.7158
Rotatable Bonds
1
Heavy Atom Count
16
Polar Areas
62.2
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
6
Complexity
16

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 5487
SID: 15196825
ChEMBL ID
CHEMBL1079
DrugBank ID
DB00697
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02060, Alpha-1A adrenergic receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 264 nM
   TI
   LI
   LO
   TS
Protein ID: PT00644, Alpha-1B adrenergic receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 322 nM
   TI
   LI
   LO
   TS
Protein ID: PT01650, Alpha-2A adrenergic receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000028 PC-12 Homo sapiens (Human)  1
1
EC50 = 86 nM
   TI
   LI
   LO
   TS
Protein ID: PT01598, Alpha-2C adrenergic receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000028 PC-12 Homo sapiens (Human)  1
1
EC50 = 1231 nM
   TI
   LI
   LO
   TS
Clinical Information about the Compound
Drug 1 ( Tizanidine )
Drug Name Tizanidine
Company Elan Pharmaceuticals
Indication
Spasm
Approved