General Information of the Compound
Compound ID
CP0176687
Compound Name
5-chloro-2-N-[4-(4-methylpiperazin-1-yl)phenyl]-4-N-[3-(trifluoromethyl)phenyl]pyrimidine-2,4-diamine
    Show/Hide
Formula
C22H22ClF3N6
Molecular Weight
462.907
Canonical SMILES
CN1CCN(CC1)c1ccc(Nc2ncc(Cl)c(Nc3cccc(c3)C(F)(F)F)n2)cc1
    Show/Hide
InChI
InChI=1S/C22H22ClF3N6/c1-31-9-11-32(12-10-31)18-7-5-16(6-8-18)29-21-27-14-19(23)20(30-21)28-17-4-2-3-15(13-17)22(24,25)26/h2-8,13-14H,9-12H2,1H3,(H2,27,28,29,30)
    Show/Hide
InChIKey
CJGXYTXDCLOCPM-UHFFFAOYSA-N
Physicochemical Property
logP
5.3878
Rotatable Bonds
5
Heavy Atom Count
32
Polar Areas
56.32
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
6
Complexity
32

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
ChEMBL ID
CHEMBL4862932
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02790, Dipeptidyl peptidase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000100 U-937 Homo sapiens (Human)  1
1
IC50 = 144 nM
   TI
   LI
   LO
   TS
CL000040 THP-1 Homo sapiens (Human)  1
1
IC50 = 1005 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 142 nM