General Information of the Compound
Compound ID
CP0154920
Compound Name
5-[(2S)-3-(5-chlorospiro[3H-1-benzofuran-2,4'-piperidine]-1'-yl)-2-hydroxypropoxy]-4H-1,4-benzoxazin-3-one
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Structure
Formula
C23H25ClN2O5
Molecular Weight
444.915
Canonical SMILES
O[C@H](COc1cccc2OCC(=O)Nc12)CN1CCC2(Cc3cc(Cl)ccc3O2)CC1
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InChI
InChI=1S/C23H25ClN2O5/c24-16-4-5-18-15(10-16)11-23(31-18)6-8-26(9-7-23)12-17(27)13-29-19-2-1-3-20-22(19)25-21(28)14-30-20/h1-5,10,17,27H,6-9,11-14H2,(H,25,28)/t17-/m0/s1
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InChIKey
LUXDNYIVTMMDTA-KRWDZBQOSA-N
Physicochemical Property
logP
2.8803
Rotatable Bonds
5
Heavy Atom Count
31
Polar Areas
80.26
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
6
Complexity
31

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 69435853
ChEMBL ID
CHEMBL3099951
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01070, C-C chemokine receptor type 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 7.1 nM
   TI
   LI
   LO
   TS
Protein ID: PT00897, Potassium voltage-gated channel subfamily H member 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 600 nM
   TI
   LI
   LO
   TS