General Information of the Compound
Compound ID
CP0153397
Compound Name
1-Cyclohexyl-2-[4-(di-pyridin-3-yl-methoxy)-2-fluoro-phenyl]-1H-benzoimidazole-5-carboxylic acid
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Structure
Formula
C31H27FN4O3
Molecular Weight
522.58
Canonical SMILES
OC(=O)c1ccc2n(C3CCCCC3)c(nc2c1)-c1ccc(OC(c2cccnc2)c2cccnc2)cc1F
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InChI
InChI=1S/C31H27FN4O3/c32-26-17-24(39-29(21-6-4-14-33-18-21)22-7-5-15-34-19-22)11-12-25(26)30-35-27-16-20(31(37)38)10-13-28(27)36(30)23-8-2-1-3-9-23/h4-7,10-19,23,29H,1-3,8-9H2,(H,37,38)
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InChIKey
GUDDSFDGSKXACG-UHFFFAOYSA-N
Physicochemical Property
logP
7.0042
Rotatable Bonds
7
Heavy Atom Count
39
Polar Areas
90.13
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
6
Complexity
39

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 15956785
ChEMBL ID
CHEMBL383304
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00013, RNA-directed RNA polymerase
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000540 Huh-5-2 Homo sapiens (Human)  1
1
EC50 = 2600 nM
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Biochemical Assays
1 IC50 = 1100 nM
2 IC50 = 2200 nM
Cell Viability or Cytotoxicity Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000540 Huh-5-2 Homo sapiens (Human)  1
1
CC50 > 50000 nM
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