General Information of the Compound
Compound ID
CP0059673
Compound Name
(3-amino-1-hydroxy-1-phosphonopropyl)phosphonic acid
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Synonyms
(3-AMINO-1-HYDROXY-1-PHOSPHONO-PROPYL)PHOSPHONIC ACID
(3-Amino-1-hydroxypropylidene)bisphosphonic acid
(3-Amino-1-hydroxypropylidene)diphosphonic acid
(3-amino-1-hydroxy-1-phosphonopropyl)phosphonic acid
(3-amino-1-hydroxypropane-1,1-diyl)bis(phosphonic acid)
(3-amino-1-hydroxypropylidene)-1,1-biphosphonate
(3-amino-1-hydroxypropylidene)-1,1-bisphosphonate
1-hydroxy-3-aminopropane-1,1-diphosphonic acid
3-Amino-1-hydroxypropylidene-1,1-diphosphonate
AHPrBP
Acide pamidronique
Acide pamidronique [INN-French]
Acido pamidronico
Acido pamidronico [INN-Spanish]
Acidum pamidronicum
Acidum pamidronicum [INN-Latin]
Amidronate
Amino-1-hydroxypropane-1,1-diphosphonate
Aminohydroxypropylidene diphosphonate
Aminomux
Aminopropanehydroxydiphosphonate
Aredia
Bisphosphonate 6
Novartis brand of pamidronate disodium salt
PAMIDRONATE DISODIUM
PAMIDRONIC ACID
Pamidronate
Pamidronate calcium
Pamidronate monosodium
Pamidronic acid (INN)
Pamidronic acid [INN:BAN]
Ribodroat
Ribodroat (TN)
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Structure
Formula
C3H11NO7P2
Molecular Weight
235.069
Canonical SMILES
NCCC(O)(P(O)(O)=O)P(O)(O)=O
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InChI
InChI=1S/C3H11NO7P2/c4-2-1-3(5,12(6,7)8)13(9,10)11/h5H,1-2,4H2,(H2,6,7,8)(H2,9,10,11)
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InChIKey
WRUUGTRCQOWXEG-UHFFFAOYSA-N
CAS
40391-99-9
Physicochemical Property
logP
-1.6633
Rotatable Bonds
4
Heavy Atom Count
13
Polar Areas
161.31
Hydrogen Bond Donor Count
6
Hydrogen Bond Acceptor Count
4
Complexity
13

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 4674
SID: 14798245
ChEMBL ID
CHEMBL834
DrugBank ID
DB00282
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT06109, Geminin
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000015 SW480 Homo sapiens (Human)  1
1
Potency ~ 13335.9 nM
   TI
   LI
   LO
   TS
Clinical Information about the Compound
Drug 1 ( Pamidronate )
Drug Name Pamidronate
Indication
Hypercalcaemia
Approved
Target(s)
Geranyltranstransferase (FDPS)
Inhibitor