General Information of the Compound
Compound ID
CP0031250
Compound Name
N-[5-[5-[2-(cyclopropylmethylamino)pyrimidin-4-yl]-2-(1-methylpiperidin-4-yl)-1,3-thiazol-4-yl]-2-fluorophenyl]methanesulfonamide
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Structure
Formula
C24H29FN6O2S2
Molecular Weight
516.668
Canonical SMILES
CN1CCC(CC1)c1nc(c(s1)-c1ccnc(NCC2CC2)n1)-c1ccc(F)c(NS(C)(=O)=O)c1
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InChI
InChI=1S/C24H29FN6O2S2/c1-31-11-8-16(9-12-31)23-29-21(17-5-6-18(25)20(13-17)30-35(2,32)33)22(34-23)19-7-10-26-24(28-19)27-14-15-3-4-15/h5-7,10,13,15-16,30H,3-4,8-9,11-12,14H2,1-2H3,(H,26,27,28)
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InChIKey
LIGMPEYLZKWWSR-UHFFFAOYSA-N
Physicochemical Property
logP
4.4088
Rotatable Bonds
8
Heavy Atom Count
35
Polar Areas
100.11
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
8
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 145991807
ChEMBL ID
CHEMBL4286841
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00897, Potassium voltage-gated channel subfamily H member 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 1340 nM
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