| Compound ID |
Compound Name |
Compound Formula |
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CP0313996
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[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[[(2S)-2-[[1-[[(2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylsulfanylbutanoyl]amino]cyclopentanecarbonyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
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C60H71F6N9O10S
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2
|
| 1 |
EC50 = 0.26 nM
|
|
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| 2 |
Ki = 5 nM
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CP0146998
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[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]hexanoylamino]-3-(1H-indol-3-yl)propanoate
Show/Hide
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C49H53F6N7O8
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2
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| 1 |
EC50 = 0.38 nM
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|
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| 2 |
Ki = 1.6 nM
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CP0053696
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[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
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C49H53F6N7O8
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2
|
| 1 |
EC50 = 1.1 nM
|
|
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| 2 |
Ki = 0.6 nM
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CP0404126
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[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylsulfanylbutanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C57H67F6N9O10S
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2
|
| 1 |
EC50 = 2.5 nM
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|
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| 2 |
Ki = 25 nM
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CP0045380
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(2S)-2-amino-N-[(1R)-1-[({[(1S)-1-{N'-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenylpropanoyl]hydrazinecarbonyl}-2-phenylethyl]carbamoyl}methyl)carbamoyl]ethyl]-3-(4-hydroxyphenyl)propanamide
Show/Hide
|
C46H56N10O10
|
2
|
| 1 |
EC50 = 2.6 nM
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|
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| 2 |
Ki = 2.6 nM
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CP0078358
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[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[[2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-(4-fluorophenyl)propanoyl]amino]acetyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C45H44F7N7O8
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2
|
| 1 |
EC50 = 3.4 nM
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|
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| 2 |
Ki = 4.5 nM
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CP0313995
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[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylsulfanylbutanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C48H51F6N7O8S
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2
|
| 1 |
EC50 = 4.8 nM
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| 2 |
Ki = 2.9 nM
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CP0419819
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[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylsulfanylbutanoyl]amino]-2-methylpropanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C58H69F6N9O10S
|
2
|
| 1 |
EC50 = 5.5 nM
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| 2 |
Ki = 3.1 nM
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CP0141881
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[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-(4-fluorophenyl)propanoate
Show/Hide
|
C32H31F7N4O6
|
2
|
| 1 |
EC50 = 6.7 nM
|
|
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| 2 |
Ki = 56 nM
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CP0440564
|
(2S)-2-{[(2S)-1-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenylpropanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-(benzylcarbamoyl)-2-(1H-indol-3-yl)ethyl]-4-methylpentanamide
Show/Hide
|
C52H63N9O8
|
1
|
| 1 |
EC50 = 10 nM
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CP0078359
|
[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]amino]propanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C34H34F6N4O5
|
2
|
| 1 |
EC50 = 12 nM
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| 2 |
Ki = 0.8 nM
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CP0385819
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(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]amino]propanoyl]amino]-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-3-(1H-indol-3-yl)propanamide
Show/Hide
|
C34H35F6N5O4
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2
|
| 1 |
EC50 = 24 nM
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| 2 |
Ki = 64 nM
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CP0385820
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[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[[2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-(4-chlorophenyl)propanoyl]amino]acetyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C45H44ClF6N7O8
|
2
|
| 1 |
EC50 = 25 nM
|
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| 2 |
Ki = 11 nM
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CP0294890
|
[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[[2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]acetyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C45H45F6N7O8
|
2
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| 1 |
EC50 = 27 nM
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| 2 |
Ki = 4.7 nM
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CP0382269
|
C-terminal modified bifunctional peptide, 2
Show/Hide
|
C52H62N8O9
|
1
|
| 1 |
EC50 = 31 nM
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CP0394035
|
(2S)-2-{[(2S)-1-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenylpropanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-({[3,5-bis(trifluoromethyl)phenyl]methyl}(methyl)carbamoyl)-2-(1H-indol-3-yl)ethyl]-4-methylpentanamide
Show/Hide
|
C55H63F6N9O8
|
1
|
| 1 |
EC50 = 31 nM
|
|
|
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CP0394033
|
C-terminal modified bifunctional peptide, 1
Show/Hide
|
C54H60F6N8O9
|
1
|
| 1 |
EC50 = 50 nM
|
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CP0043850
|
(2S)-2-{[(2S)-1-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenylpropanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-({[3,5-bis(trifluoromethyl)phenyl]methyl}carbamoyl)-2-(1H-indol-3-yl)ethyl]-4-methylpentanamide
Show/Hide
|
C54H61F6N9O8
|
1
|
| 1 |
EC50 = 72 nM
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CP0244494
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[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[[(2S)-1-[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]pyrrolidine-2-carbonyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C48H49F6N7O8
|
2
|
| 1 |
EC50 = 76 nM
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| 2 |
Ki = 5.7 nM
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CP0382268
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(2S)-2-{[(2S)-1-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenylpropanoyl]pyrrolidin-2-yl]formamido}-N-[(1S)-1-[benzyl(methyl)carbamoyl]-2-(1H-indol-3-yl)ethyl]-4-methylpentanamide
Show/Hide
|
C53H65N9O8
|
1
|
| 1 |
EC50 = 77 nM
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|
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CP0141882
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[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C32H30F6N4O5
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2
|
| 1 |
EC50 = 91 nM
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|
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| 2 |
Ki = 100 nM
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CP0066825
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[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C43H42F6N6O7
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2
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| 1 |
EC50 = 150 nM
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| 2 |
Ki = 35 nM
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CP0146784
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[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[3-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]propanoylamino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C46H47F6N7O8
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2
|
| 1 |
EC50 = 160 nM
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| 2 |
Ki = 58 nM
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CP0368138
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[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[[(2S)-2-[[(2R)-1-[(2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylsulfanylbutanoyl]pyrrolidine-2-carbonyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C59H69F6N9O10S
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2
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| 1 |
EC50 = 190 nM
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| 2 |
Ki = 13 nM
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CP0068481
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[3,5-bis(trifluoromethyl)phenyl]methyl (2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C34H33F6N5O6
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2
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| 1 |
EC50 = 280 nM
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| 2 |
Ki = 310 nM
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CP0402964
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(S)-2-amino-N-((R)-1-(2-((S)-3-(4-fluorophenyl)-1-oxo-1-(4-(N-phenylpropionamido)piperidin-1-yl)propan-2-ylamino)-2-oxoethylamino)-1-oxopropan-2-yl)-3-(4-hydroxy-2,6-dimethylphenyl)propanamide
Show/Hide
|
C39H49FN6O6
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2
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| 1 |
IC50 = 0.06457 nM
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| 2 |
Ki = 0.03 nM
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CP0379715
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(R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido)-N-(2-((S)-3-(4-chlorophenyl)-1-oxo-1-(4-(N-phenylpropionamido)piperidin-1-yl)propan-2-ylamino)-2-oxoethyl)hexanamide
Show/Hide
|
C42H55ClN6O6
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2
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| 1 |
IC50 = 0.1862 nM
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| 2 |
Ki = 0.08 nM
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CP0379720
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(R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-N-(2-((S)-3-(4-chlorophenyl)-1-oxo-1-(4-(N-phenylpropionamido)piperidin-1-yl)propan-2-ylamino)-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
Show/Hide
|
C46H53ClN6O6
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2
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| 1 |
IC50 = 0.257 nM
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| 2 |
Ki = 0.11 nM
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CP0379713
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(S)-2-amino-N-((R)-1-(2-((S)-3-(4-chlorophenyl)-1-oxo-1-(4-(N-phenylpropionamido)piperidin-1-yl)propan-2-ylamino)-2-oxoethylamino)-1-oxopropan-2-yl)-3-(4-hydroxy-2,6-dimethylphenyl)propanamide
Show/Hide
|
C39H49ClN6O6
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2
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| 1 |
IC50 = 0.302 nM
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| 2 |
Ki = 0.14 nM
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CP0372167
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(S)-1-((2S,5S,11R,14S)-14-amino-5-benzyl-2-butyl-15-(4-hydroxy-2,6-dimethylphenyl)-11-methyl-4,7,10,13-tetraoxo-3,6,9,12-tetraazapentadecane)-N-((S)-1-((S)-1-(3,4-dimethoxybenzylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-4-methyl-1-oxopentan-2-yl)pyrrolidine-2-carboxamide
Show/Hide
|
C62H82N10O11
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2
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| 1 |
IC50 = 0.3162 nM
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| 2 |
Ki = 0.15 nM
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CP0379711
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(R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido)-N-(2-oxo-2-((S)-1-oxo-3-phenyl-1-(4-(N-phenylpropionamido)piperidin-1-yl)propan-2-ylamino)ethyl)hexanamide
Show/Hide
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C42H56N6O6
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2
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| 1 |
IC50 = 0.3802 nM
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| 2 |
Ki = 0.18 nM
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CP0436682
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(S)-1-((2S,5S,11R,14S)-14-amino-5-benzyl-15-(4-hydroxy-2,6-dimethylphenyl)-11-methyl-2-(2-(methylthio)ethyl)-4,7,10,13-tetraoxo-3,6,9,12-tetraazapentadecane)-N-((S)-1-((S)-1-(3,5-bis(trifluoromethyl)benzylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-4-methyl-1-oxopentan-2-yl)pyrrolidine-2-carboxamide
Show/Hide
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C61H74F6N10O9S
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2
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| 1 |
IC50 = 0.3802 nM
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| 2 |
Ki = 0.18 nM
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CP0373037
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(3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazol-5-yl)methyl)-9-((1H-indol-3-yl)methyl)-30-amino-3-((S)-1-amino-1-oxo-3-phenylpropan-2-ylcarbamoyl)-21-benzyl-6-butyl-12-(3-guanidinopropyl)-31-(4-hydroxy-2,6-dimethylphenyl)-27-methyl-15-(naphthalen-2-ylmethyl)-5,8,11,14,17,20,23,26,29-nonaoxo-4,7,10,13,16,19,22,25,28-nonaazahentriacontan-1-oic acid
Show/Hide
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C80H98N18O14
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2
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| 1 |
IC50 = 0.3981 nM
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| 2 |
Ki = 0.21 nM
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CP0419476
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(3S)-4-[[(2S)-1-[[(1R)-2-[1-(1-adamantyloxycarbonyl)indol-3-yl]-1-carboxyethyl]amino]-1-oxohexan-2-yl]amino]-3-[[(2S)-2-[2-[(2S)-1-[[2-[[(2R)-1-[[(1S)-1-carboxy-2-(4-hydroxyphenyl)ethyl]amino]-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-1-oxo-3-phenylpropan-2-yl]hydrazinyl]-3-phenylpropanoyl]amino]-4-oxobutanoic acid
Show/Hide
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C64H77N9O15
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2
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| 1 |
IC50 = 0.4169 nM
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| 2 |
Ki = 0.23 nM
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CP0371819
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(3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]-3-phenylpropanamido]acetamido}-3-(1H-indol-3-yl)propanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C50H59N9O10
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2
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| 1 |
IC50 = 0.4266 nM
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| 2 |
Ki = 0.2 nM
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CP0199125
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(3S)-2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-[(2S)-1-oxo-3-phenyl-1-[4-(N-propanoylanilino)piperidin-1-yl]propan-2-yl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Show/Hide
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C44H51N5O5
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2
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| 1 |
IC50 = 0.4266 nM
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| 2 |
Ki = 0.2 nM
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CP0371833
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(3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-(1H-indol-3-yl)propanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C44H55N9O10
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2
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| 1 |
IC50 = 0.5248 nM
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| 2 |
Ki = 0.22 nM
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CP0078906
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(3S)-2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-[(2S)-3-(4-chlorophenyl)-1-oxo-1-[4-(N-propanoylanilino)piperidin-1-yl]propan-2-yl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Show/Hide
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C44H50ClN5O5
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2
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| 1 |
IC50 = 0.6761 nM
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| 2 |
Ki = 0.43 nM
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CP0534826
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(3R)-2-[(2S)-2-amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[2-[[(2S)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino]-2-oxoethyl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Show/Hide
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C46H51Cl2FN6O6
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2
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| 1 |
IC50 = 0.6918 nM
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| 2 |
Ki = 0.32 nM
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CP0890890
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(S)-2-amino-N-((R)-1-{[((S)-1-{(S)-1-benzyl-2-oxo-2-[4-(phenyl-propionyl-amino)-piperidin-1-yl]-ethylcarbamoyl}-2-phenyl-ethylcarbamoyl)-methyl]-carbamoyl}-ethyl)-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionamide
Show/Hide
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C48H59N7O7
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2
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| 1 |
IC50 = 0.7943 nM
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| 2 |
Ki = 0.36 nM
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CP0373195
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(2S)-1-[(2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylsulfanylbutanoyl]-N-[(2S)-1-[[(2S)-1-(benzylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamide
Show/Hide
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C57H72N10O9S
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2
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| 1 |
IC50 = 0.7943 nM
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| 2 |
Ki = 0.44 nM
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CP0379710
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(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-N-[(1R)-1-[({[(2S)-1-oxo-3-phenyl-1-[4-(N-phenylpropanamido)piperidin-1-yl]propan-2-yl]carbamoyl}methyl)carbamoyl]ethyl]propanamide
Show/Hide
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C39H50N6O6
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4
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| 1 |
IC50 = 0.7943 nM
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| 2 |
IC50 = 398.11 nM
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| 3 |
Ki = 0.36 nM
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| 4 |
Ki = 180 nM
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CP0379708
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(R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido)-N-(2-((S)-3-(4-fluorophenyl)-1-oxo-1-(4-(N-phenylpropionamido)piperidin-1-yl)propan-2-ylamino)-2-oxoethyl)hexanamide
Show/Hide
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C42H55FN6O6
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2
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| 1 |
IC50 = 0.8511 nM
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| 2 |
Ki = 0.4 nM
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CP0422116
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(S)-1-((2S,5S,11R,14S)-14-amino-5-benzyl-2-butyl-15-(4-hydroxy-2,6-dimethylphenyl)-11-methyl-4,7,10,13-tetraoxo-3,6,9,12-tetraazapentadecane)-N-((S)-1-((S)-1-((3,5-bis(trifluoromethyl)benzyl)(methyl)amino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-4-methyl-1-oxopentan-2-yl)pyrrolidine-2-carboxamide
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C63H78F6N10O9
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2
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| 1 |
IC50 = 0.9772 nM
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| 2 |
Ki = 0.46 nM
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CP0371862
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(3S)-3-[(2S)-2-[(2R)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]-3-phenylpropanamido]acetamido}-3-(1H-indol-3-yl)-N-methylpropanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C51H61N9O10
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2
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| 1 |
IC50 = 1 nM
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| 2 |
Ki = 0.42 nM
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CP0379719
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(R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-N-(2-((S)-3-(4-fluorophenyl)-1-oxo-1-(4-(N-phenylpropionamido)piperidin-1-yl)propan-2-ylamino)-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
Show/Hide
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C46H53FN6O6
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2
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| 1 |
IC50 = 1.072 nM
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| 2 |
Ki = 0.48 nM
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CP0403228
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(3S)-4-[[(2S)-1-[[(1S)-2-(1-acetylindol-3-yl)-1-carboxyethyl]amino]-1-oxohexan-2-yl]-[(2-chlorophenyl)carbamoyl]amino]-3-[[(2S)-2-[[[(2S)-1-[[2-[[(2R)-1-[[(1S)-1-carboxy-2-(4-hydroxyphenyl)ethyl]amino]-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-methylamino]-3-phenylpropanoyl]amino]-4-oxobutanoic acid
Show/Hide
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C63H71ClN10O15
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2
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| 1 |
IC50 = 1.122 nM
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| 2 |
Ki = 0.48 nM
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CP0546858
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(3R)-2-[(2S)-2-amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[2-[[(2S)-3-(4-chlorophenyl)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-1-oxopropan-2-yl]amino]-2-oxoethyl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Show/Hide
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C46H51Cl3N6O6
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2
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| 1 |
IC50 = 1.175 nM
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| 2 |
Ki = 0.54 nM
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CP0543992
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(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-N-[2-[[(2S)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino]-2-oxoethyl]hexanamide
Show/Hide
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C40H49Cl2FN6O6
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2
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| 1 |
IC50 = 1.23 nM
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| 2 |
Ki = 0.57 nM
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CP0495192
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(2R)-2-[[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]amino]-N-[2-[[(2S)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino]-2-oxoethyl]hexanamide
Show/Hide
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C42H53Cl2FN6O6
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2
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| 1 |
IC50 = 1.259 nM
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| 2 |
Ki = 0.58 nM
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CP0324102
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(3S)-4-[[(2S)-1-[[(2R)-1-[2-[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]hydrazinyl]-3-(1H-indol-2-yl)-1-oxopropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-[[(2S)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-3-phenylpropanoyl]amino]-4-oxobutanoic acid
Show/Hide
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C58H73N11O13
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2
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| 1 |
IC50 = 1.38 nM
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| 2 |
Ki = 0.63 nM
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CP0233352
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(2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylsulfanylbutanamide
Show/Hide
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C28H38N6O6S
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2
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| 1 |
IC50 = 1.38 nM
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| 2 |
Ki = 0.66 nM
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CP0043301
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(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]-N-methylacetamido}-N-(2-hydroxyethyl)-3-phenylpropanamide
Show/Hide
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C26H35N5O6
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2
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| 1 |
IC50 = 1.445 nM
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| 2 |
Ki = 0.66 nM
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CP0233356
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(S)-1-((2S,5S,11R,14S)-14-amino-5-benzyl-15-(4-hydroxyphenyl)-11-methyl-2-(2-(methylthio)ethyl)-4,7,10,13-tetraoxo-3,6,9,12-tetraazapentadecane)-N-((S)-1-((S)-1-(3,5-bis(trifluoromethyl)benzylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-4-methyl-1-oxopentan-2-yl)pyrrolidine-2-carboxamide
Show/Hide
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C59H70F6N10O9S
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3
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| 1 |
IC50 = 1.445 nM
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| 2 |
IC50 = 1.585 nM
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| 3 |
Ki = 0.66 nM
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CP0387532
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(S)-1-((2S,5S,11R,14S)-14-amino-5-benzyl-2-butyl-15-(4-hydroxyphenyl)-11-methyl-4,7,10,13-tetraoxo-3,6,9,12-tetraazapentadecane)-N-((S)-1-((S)-1-((S)-1-(3,5-bis(trifluoromethyl)benzylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-3-((2R,3R,4S,5S,6R)-6-ethyl-3,4,5-trihydroxytetrahydro-2H-pyran-2-yloxy)-1-oxopropan-2-ylamino)-4-methyl-1-oxopentan-2-yl)pyrrolidine-2-carboxamide
Show/Hide
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C70H89F6N11O15
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2
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| 1 |
IC50 = 1.479 nM
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| 2 |
Ki = 0.77 nM
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CP0108537
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(3R)-2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-[(2S)-1-oxo-3-phenyl-1-[4-(N-propanoylanilino)piperidin-1-yl]propan-2-yl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Show/Hide
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C44H51N5O5
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2
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| 1 |
IC50 = 1.585 nM
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| 2 |
Ki = 0.76 nM
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CP0543991
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(2S)-2-amino-N-[(2R)-1-[[2-[[(2S)-3-(4-chlorophenyl)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-1-oxopropan-2-yl]-3-(4-hydroxy-2,6-dimethylphenyl)propanamide
Show/Hide
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C39H47Cl3N6O6
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2
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| 1 |
IC50 = 1.585 nM
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| 2 |
Ki = 0.74 nM
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CP0342086
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(3R)-4-[[(2R)-1-[2-[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]hydrazinyl]-1-oxo-3-phenylpropan-2-yl]amino]-3-[[(2R)-2-[[(2S)-2-amino-3-(1H-indol-2-yl)propanoyl]amino]hexanoyl]amino]-4-oxobutanoic acid
Show/Hide
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C53H65N11O11
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2
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| 1 |
IC50 = 1.66 nM
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| 2 |
Ki = 0.8 nM
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CP0914986
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(S)-2-amino-N-((R)-1-{[((S)-1-{(S)-1-benzyl-2-oxo-2-[4-(phenyl-propionyl-amino)-piperidin-1-yl]-ethylcarbamoyl}-2-phenyl-ethylcarbamoyl)-methyl]-carbamoyl}-ethyl)-3-(4-hydroxy-phenyl)-propionamide
Show/Hide
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C46H55N7O7
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2
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| 1 |
IC50 = 1.778 nM
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| 2 |
Ki = 0.69 nM
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CP0403232
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(3S)-3-[[(2S)-2-[2-[(2S)-1-[[2-[[(2R)-1-[[(1S)-1-carboxy-2-(4-hydroxyphenyl)ethyl]amino]-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-1-oxo-3-phenylpropan-2-yl]hydrazinyl]-3-phenylpropanoyl]amino]-4-[[(2S)-1-[[(1R)-1-carboxy-2-[1-[(2-methylpropan-2-yl)oxycarbonyl]indol-3-yl]ethyl]amino]-1-oxohexan-2-yl]-methylamino]-4-oxobutanoic acid
Show/Hide
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C59H73N9O15
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2
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| 1 |
IC50 = 1.995 nM
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| 2 |
Ki = 0.82 nM
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CP0851949
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(3S,6R,9S,12S,15S,18S)-3-((1H-imidazol-5-yl)methyl)-12-((1H-indol-3-yl)methyl)-18-((S)-1-amino-1-oxo-3-phenylpropan-2-ylcarbamoyl)-1-(2-((R)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinolin-3-yl)-15-butyl-9-(3-guanidinopropyl)-6-(naphthalen-2-ylmethyl)-1,4,7,10,13,16-hexaoxo-2,5,8,11,14,17-hexaazaicosan-20-oic acid
Show/Hide
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C76H90N16O12
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2
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| 1 |
IC50 = 1.995 nM
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| 2 |
Ki = 0.91 nM
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CP0396946
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(S)-1-((2S,5S,11R,14S)-14-amino-5-benzyl-2-butyl-15-(4-hydroxyphenyl)-11-methyl-4,7,10,13-tetraoxo-3,6,9,12-tetraazapentadecane)-N-((S)-1-((S)-1-(3,5-bis(trifluoromethyl)benzylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-4-methyl-1-oxopentan-2-yl)pyrrolidine-2-carboxamide
Show/Hide
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C60H72F6N10O9
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2
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| 1 |
IC50 = 2.138 nM
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| 2 |
Ki = 1 nM
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CP0534824
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(2S)-2-amino-N-[(2R)-1-[[2-[[(2S)-3-(4-chlorophenyl)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-1-oxopropan-2-yl]-3-(4-hydroxyphenyl)propanamide
Show/Hide
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C37H43Cl3N6O6
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2
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| 1 |
IC50 = 2.344 nM
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| 2 |
Ki = 1.1 nM
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CP0379706
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(R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido)-N-((S)-1-oxo-3-phenyl-1-(4-(N-phenylpropionamido)piperidin-1-yl)propan-2-yl)hexanamide
Show/Hide
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C40H53N5O5
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2
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| 1 |
IC50 = 2.399 nM
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| 2 |
Ki = 1.1 nM
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CP0288626
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(3S)-4-[[(2S)-1-[[(2R)-1-[2-[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]hydrazinyl]-3-(1H-indol-2-yl)-1-oxopropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-[[(2S)-2-amino-3-phenylpropanoyl]amino]-4-oxobutanoic acid
Show/Hide
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C53H65N11O11
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2
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| 1 |
IC50 = 2.57 nM
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| 2 |
Ki = 1.1 nM
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CP0527959
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(3R)-2-[(2S)-2-amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(2S)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-3-(4-fluorophenyl)-1-oxopropan-2-yl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Show/Hide
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C44H48Cl2FN5O5
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2
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| 1 |
IC50 = 2.63 nM
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| 2 |
Ki = 1.2 nM
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CP0373267
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(3S,6S,12S,17R,20S)-12-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-6-benzyl-N-[(2S)-1-[[3,5-bis(trifluoromethyl)phenyl]methylamino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-3-butyl-2,5,8,11,19-pentaoxo-14,15-dithia-1,4,7,10,18-pentazabicyclo[18.3.0]tricosane-17-carboxamide
Show/Hide
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C57H64F6N10O9S2
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2
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| 1 |
IC50 = 2.692 nM
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| 2 |
Ki = 1.3 nM
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CP0403230
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(3S)-3-[[(2S)-2-[2-[(2S)-1-[[2-[[(2R)-1-[[(1S)-1-carboxy-2-(4-hydroxyphenyl)ethyl]amino]-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-1-oxo-3-phenylpropan-2-yl]hydrazinyl]-3-phenylpropanoyl]amino]-4-[[(2S)-1-[[(1R)-1-carboxy-2-(1H-indol-3-yl)ethyl]amino]-1-oxohexan-2-yl]amino]-4-oxobutanoic acid
Show/Hide
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C53H63N9O13
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2
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| 1 |
IC50 = 3.236 nM
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| 2 |
Ki = 1.4 nM
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CP0324104
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(3S)-3-[(2S)-2-[(2R)-2-amino-3-(1H-indol-2-yl)propanamido]hexanamido]-3-{[(2S)-1-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenylpropanehydrazido]-1-oxo-3-phenylpropan-2-yl]carbamoyl}propanoic acid
Show/Hide
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C53H65N11O11
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2
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| 1 |
IC50 = 3.236 nM
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| 2 |
Ki = 1.4 nM
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CP0402965
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(S)-2-amino-N-((R)-1-((S)-3-(4-chlorophenyl)-1-oxo-1-(4-(N-phenylpropionamido)piperidin-1-yl)propan-2-ylamino)-1-oxopropan-2-yl)-3-(4-hydroxy-2,6-dimethylphenyl)propanamide
Show/Hide
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C37H46ClN5O5
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2
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| 1 |
IC50 = 3.236 nM
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| 2 |
Ki = 1.6 nM
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CP0134169
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(3S)-3-[(2S)-2-[(2R)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-(1H-indol-3-yl)-N-methylpropanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C45H57N9O10
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2
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| 1 |
IC50 = 3.467 nM
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| 2 |
Ki = 1.5 nM
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CP0506050
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(S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-N-((R)-1-oxo-1-((S)-1-oxo-3-phenyl-1-(4-(N-phenylpropionamido)piperidin-1-yl)propan-2-ylamino)propan-2-yl)propanamide
Show/Hide
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C37H47N5O5
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2
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| 1 |
IC50 = 3.631 nM
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| 2 |
Ki = 1.7 nM
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CP0431982
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Bifunctional Peptide Ligand, 7 (TY018)
Show/Hide
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C60H71F6N9O10
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2
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| 1 |
IC50 = 3.802 nM
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| 2 |
Ki = 1.8 nM
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CP0534832
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(2S)-2-amino-N-[(2R)-1-[[2-[[(2S)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-1-oxo-3-phenylpropan-2-yl]amino]-2-oxoethyl]amino]-1-oxopropan-2-yl]-3-(4-hydroxyphenyl)propanamide
Show/Hide
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C37H44Cl2N6O6
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2
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| 1 |
IC50 = 4.571 nM
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| 2 |
Ki = 2.1 nM
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CP0371825
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(3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]hexanamido]acetamido}-3-(1H-indol-3-yl)-N-methylpropanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C48H63N9O10
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2
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| 1 |
IC50 = 4.677 nM
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| 2 |
Ki = 2 nM
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CP0288627
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(3R)-4-[[(2R)-1-[[(2S)-1-[2-[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]hydrazinyl]-3-(1H-indol-2-yl)-1-oxopropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-[[(2R)-2-amino-3-phenylpropanoyl]amino]-4-oxobutanoic acid
Show/Hide
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C53H65N11O11
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2
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| 1 |
IC50 = 5.129 nM
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| 2 |
Ki = 2.2 nM
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CP0371826
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(3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-(1H-indol-3-yl)-N-methylpropanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C45H57N9O10
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2
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| 1 |
IC50 = 5.248 nM
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| 2 |
Ki = 2.2 nM
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CP0383598
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Bifunctional Peptide Ligand, 5 (TY005)
Show/Hide
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C59H69F6N9O10S
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3
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| 1 |
IC50 = 6.026 nM
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| 2 |
IC50 = 6.31 nM
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| 3 |
Ki = 2.8 nM
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CP0371863
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(3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]hexanamido]acetamido}-3-(1H-indol-3-yl)propanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C47H61N9O10
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2
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| 1 |
IC50 = 6.026 nM
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| 2 |
Ki = 2.6 nM
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CP0400846
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(3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazol-5-yl)methyl)-9-((1H-indol-3-yl)methyl)-30-amino-3-((S)-1-amino-1-oxo-3-phenylpropan-2-ylcarbamoyl)-21-benzyl-6-butyl-12-(3-guanidinopropyl)-31-(4-hydroxyphenyl)-27-methyl-15-(naphthalen-2-ylmethyl)-5,8,11,14,17,20,23,26,29-nonaoxo-4,7,10,13,16,19,22,25,28-nonaazahentriacontan-1-oic acid
Show/Hide
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C78H94N18O14
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2
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| 1 |
IC50 = 6.31 nM
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| 2 |
Ki = 2.9 nM
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CP0454986
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(2S)-2-amino-3-(4-hydroxyphenyl)-N-[(1R)-1-[({[(2S)-1-oxo-1-{4-oxo-4-[4-(N-phenylpropanamido)piperidin-1-yl]butanehydrazido}-3-phenylpropan-2-yl]carbamoyl}methyl)carbamoyl]ethyl]propanamide
Show/Hide
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C41H52N8O8
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2
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| 1 |
IC50 = 6.607 nM
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| 2 |
Ki = 3.2 nM
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CP0439467
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3-{N'-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenylpropanoyl]hydrazinecarbonyl}-N-[1-(2-phenylethyl)piperidin-4-yl]propanamide
Show/Hide
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C40H52N8O7
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2
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| 1 |
IC50 = 7.586 nM
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| 2 |
Ki = 3.7 nM
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CP0403408
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(3S)-4-[[(2S)-1-[[(1R)-2-[1-(2-adamantyloxycarbonyl)indol-3-yl]-1-carboxyethyl]amino]-1-oxohexan-2-yl]amino]-3-[[(2S)-2-[2-[(2S)-1-[[2-[[(2R)-1-[[(1S)-1-carboxy-2-(4-hydroxyphenyl)ethyl]amino]-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-1-oxo-3-phenylpropan-2-yl]hydrazinyl]-3-phenylpropanoyl]amino]-4-oxobutanoic acid
Show/Hide
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C64H77N9O15
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2
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| 1 |
IC50 = 7.762 nM
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| 2 |
Ki = 3.4 nM
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CP0551809
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(3R)-2-[(2S)-2-amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(2S)-3-(4-chlorophenyl)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-1-oxopropan-2-yl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
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C44H48Cl3N5O5
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2
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| 1 |
IC50 = 7.762 nM
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| 2 |
Ki = 3.6 nM
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CP0375711
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(S)-1-((2S,5S,11R,14S)-14-amino-5-benzyl-2-butyl-15-(4-hydroxyphenyl)-11-methyl-4,7,10,13-tetraoxo-3,6,9,12-tetraazapentadecane)-N-((S)-1-((S)-1-(3,5-bis(trifluoromethyl)benzylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-1-oxo-3-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yloxy)propan-2-yl)pyrrolidine-2-carboxamide
Show/Hide
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C63H76F6N10O15
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2
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| 1 |
IC50 = 7.943 nM
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| 2 |
Ki = 3.7 nM
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CP0388012
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(2S,5R,11S,18S,21S)-2-amino-21-((S)-1-amino-1-oxo-3-phenylpropan-2-ylcarbamoyl)-18-((S)-2-((S)-2-((R)-2-((S)-2-amino-3-(1H-imidazol-5-yl)propanamido)-3-(4-chlorophenyl)propanamido)-5-guanidinopentanamido)-3-(1H-indol-3-yl)propanamido)-11-benzyl-1-(4-hydroxyphenyl)-5-methyl-3,6,9,12,19-pentaoxo-4,7,10,13,20-pentaazatricosan-23-oic acid
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C74H92ClN19O14
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2
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| 1 |
IC50 = 7.943 nM
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| 2 |
Ki = 3.5 nM
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CP0388014
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(6R,9S,12S,15R,18S,21S,24S,27S)-12-((1H-imidazol-5-yl)methyl)-21-((1H-indol-3-yl)methyl)-27-((S)-1-amino-1-oxo-3-phenylpropan-2-ylcarbamoyl)-9-benzyl-24-butyl-18-(3-guanidinopropyl)-1-(4-hydroxy-2,6-dimethylphenyl)-6-methyl-15-(naphthalen-2-ylmethyl)-4,7,10,13,16,19,22,25-octaoxo-3,5,8,11,14,17,20,23,26-nonaazanonacosan-29-oic acid
Show/Hide
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C78H95N17O13
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2
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| 1 |
IC50 = 7.943 nM
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| 2 |
Ki = 3.7 nM
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CP0372166
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(S)-N-((S)-1-((S)-3-(1H-indol-3-yl)-1-oxo-1-(3-(trifluoromethyl)benzylamino)propan-2-ylamino)-4-methyl-1-oxopentan-2-yl)-1-((2S,5S,11R,14S)-14-amino-5-benzyl-2-butyl-15-(4-hydroxy-2,6-dimethylphenyl)-11-methyl-4,7,10,13-tetraoxo-3,6,9,12-tetraazapentadecane)pyrrolidine-2-carboxamide
Show/Hide
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C61H77F3N10O9
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2
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| 1 |
IC50 = 8.511 nM
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| 2 |
Ki = 4.1 nM
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CP0324103
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(3R)-4-[[(2R)-1-[[(2S)-1-[2-[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]hydrazinyl]-3-(1H-indol-2-yl)-1-oxopropan-2-yl]amino]-1-oxohexan-2-yl]amino]-3-[[(2R)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-3-phenylpropanoyl]amino]-4-oxobutanoic acid
Show/Hide
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C58H73N11O13
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2
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| 1 |
IC50 = 9.12 nM
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| 2 |
Ki = 3.9 nM
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CP0419479
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(3S)-4-[[(2S)-1-[[(1S)-2-(1-acetylindol-3-yl)-1-carboxyethyl]amino]-1-oxohexan-2-yl]amino]-3-[[(2S)-2-[[[(2S)-1-[[2-[[(2R)-1-[[(1S)-1-carboxy-2-(4-hydroxyphenyl)ethyl]amino]-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-methylamino]-3-phenylpropanoyl]amino]-4-oxobutanoic acid
Show/Hide
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C56H67N9O14
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2
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| 1 |
IC50 = 10.72 nM
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| 2 |
Ki = 5.2 nM
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CP0394173
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Bifunctional Peptide Ligand, 4 (TY004)
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C60H71F6N9O10
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2
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| 1 |
IC50 = 10.72 nM
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| 2 |
Ki = 5 nM
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CP0176549
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(3R)-2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-[(2S)-3-(4-chlorophenyl)-1-oxo-1-[4-(N-propanoylanilino)piperidin-1-yl]propan-2-yl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Show/Hide
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C44H50ClN5O5
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2
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| 1 |
IC50 = 11.75 nM
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| 2 |
Ki = 5.5 nM
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CP0383594
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Bifunctional Peptide Ligand, 6 (TY023)
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C59H69F6N9O11S
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2
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| 1 |
IC50 = 12.02 nM
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| 2 |
Ki = 4.8 nM
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CP0373479
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(3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazol-5-yl)methyl)-9-((1H-indol-3-yl)methyl)-30-amino-3-((S)-1-amino-1-oxo-3-phenylpropan-2-ylcarbamoyl)-15,21-dibenzyl-6-butyl-12-(3-guanidinopropyl)-31-(4-hydroxyphenyl)-27-methyl-5,8,11,14,17,20,23,26,29-nonaoxo-4,7,10,13,16,19,22,25,28-nonaazahentriacontan-1-oic acid
Show/Hide
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C74H92N18O14
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2
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| 1 |
IC50 = 12.59 nM
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| 2 |
Ki = 6.2 nM
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CP0388015
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(S)-3-((4R,7S,10S,13R,16S,22S)-16-((1H-imidazol-5-yl)methyl)-7-((1H-indol-3-yl)methyl)-22-amino-20-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-10-(3-guanidinopropyl)-13-(naphthalen-2-ylmethyl)-6,9,12,15,18,21-hexaoxo-1,2-dithia-5,8,11,14,17,20-hexaazacyclotricosane-4-carboxamido)-4-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-4-oxobutanoic acid
Show/Hide
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C68H81N17O13S2
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2
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| 1 |
IC50 = 12.59 nM
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| 2 |
Ki = 5.6 nM
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CP0400843
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(3S,6R,9S,12S,15S,18S)-3-((1H-imidazol-5-yl)methyl)-12-((1H-indol-3-yl)methyl)-18-((S)-1-amino-1-oxo-3-phenylpropan-2-ylcarbamoyl)-1-((R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-1,2,3,4-tetrahydroisoquinolin-3-yl)-15-butyl-9-(3-guanidinopropyl)-6-(naphthalen-2-ylmethyl)-1,4,7,10,13,16-hexaoxo-2,5,8,11,14,17-hexaazaicosan-20-oic acid
Show/Hide
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C76H90N16O12
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2
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| 1 |
IC50 = 12.59 nM
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| 2 |
Ki = 6.2 nM
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CP0435191
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3-{N'-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenylpropanoyl]hydrazinecarbonyl}-N-phenyl-N-[1-(2-phenylethyl)piperidin-4-yl]propanamide
Show/Hide
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C46H56N8O7
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2
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| 1 |
IC50 = 13.18 nM
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| 2 |
Ki = 6.1 nM
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CP0373888
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(2S)-1-[(4S,7S,13S)-13-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-7-benzyl-6,9,12-trioxo-1,2-dithia-5,8,11-triazacyclotetradecane-4-carbonyl]-N-[(2S)-1-[[(2S)-1-[[3,5-bis(trifluoromethyl)phenyl]methylamino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamide
Show/Hide
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C57H64F6N10O9S2
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2
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| 1 |
IC50 = 15.49 nM
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| 2 |
Ki = 7.8 nM
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CP0342087
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(3R)-4-[[(2R)-1-[2-[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]hydrazinyl]-1-oxo-3-phenylpropan-2-yl]amino]-3-[[(2R)-2-[[(2S)-3-(1H-indol-2-yl)-2-[(2-methylpropan-2-yl)oxycarbonylamino]propanoyl]amino]hexanoyl]amino]-4-oxobutanoic acid
Show/Hide
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C58H73N11O13
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2
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| 1 |
IC50 = 16.22 nM
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| 2 |
Ki = 6.9 nM
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CP0386613
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(3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]-3-phenylpropanamido]acetamido}-3-(1H-indol-3-yl)-N-methylpropanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C51H61N9O10
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2
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| 1 |
IC50 = 18.62 nM
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| 2 |
Ki = 1 nM
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CP0388010
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(S)-3-((4R,7S,10S,13R,16S,22S)-16-((1H-imidazol-5-yl)methyl)-7-((1H-indol-3-yl)methyl)-22-amino-20-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)-13-benzyl-10-(3-guanidinopropyl)-6,9,12,15,18,21-hexaoxo-1,2-dithia-5,8,11,14,17,20-hexaazacyclotricosane-4-carboxamido)-4-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-4-oxobutanoic acid
Show/Hide
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C64H79N17O13S2
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2
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| 1 |
IC50 = 19.95 nM
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| 2 |
Ki = 9.1 nM
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CP0221759
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(3R)-2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-[(2S)-3-(4-fluorophenyl)-1-oxo-1-[4-(N-propanoylanilino)piperidin-1-yl]propan-2-yl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Show/Hide
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C44H50FN5O5
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2
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| 1 |
IC50 = 20.42 nM
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| 2 |
Ki = 9.3 nM
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CP0382815
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(2S)-1-[(4R,7S,13S)-13-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-7-benzyl-6,9,12-trioxo-1,2-dithia-5,8,11-triazacyclotetradecane-4-carbonyl]-N-[(2S)-1-[[(2S)-1-[[3,5-bis(trifluoromethyl)phenyl]methylamino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamide
Show/Hide
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C57H64F6N10O9S2
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2
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| 1 |
IC50 = 22.39 nM
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| 2 |
Ki = 5 nM
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CP0456322
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(S)-1-((2S,5S,11R,14S)-14-amino-5-benzyl-2-butyl-15-(4-hydroxy-2,6-dimethylphenyl)-11-methyl-4,7,10,13-tetraoxo-3,6,9,12-tetraazapentadecane)-N-((S)-1-((S)-1-(3,5-bis(trifluoromethyl)benzylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-4-methyl-1-oxopentan-2-yl)pyrrolidine-2-carboxamide
Show/Hide
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C62H76F6N10O9
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2
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| 1 |
IC50 = 23.99 nM
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| 2 |
Ki = 11 nM
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CP0435192
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(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenyl-N-[1-(2-phenylethyl)piperidin-4-yl]propanamide
Show/Hide
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C36H46N6O5
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2
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| 1 |
IC50 = 30.9 nM
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| 2 |
Ki = 14 nM
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CP0383437
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Bifunctional Peptide Ligand, 1 (TY003)
Show/Hide
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C63H69F6N9O10
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2
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| 1 |
IC50 = 31.62 nM
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| 2 |
Ki = 15 nM
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CP0379717
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(R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido)-N-((S)-3-(4-chlorophenyl)-1-oxo-1-(4-(N-phenylpropionamido)piperidin-1-yl)propan-2-yl)hexanamide
Show/Hide
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C40H52ClN5O5
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2
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| 1 |
IC50 = 39.81 nM
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| 2 |
Ki = 19 nM
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CP0439426
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(3S)-3-[(2S)-2-[(2R)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]hexanamido]acetamido}-3-(1H-indol-3-yl)propanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C47H61N9O10
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2
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| 1 |
IC50 = 47.86 nM
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| 2 |
Ki = 20 nM
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CP0432556
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(3S)-4-[[(2S)-1-[[(1S)-2-(1-acetylindol-3-yl)-1-carboxyethyl]amino]-1-oxohexan-2-yl]amino]-3-[[(2S)-2-[2-[(2S)-1-[[2-[[(2R)-1-[[(1S)-1-carboxy-2-(4-hydroxyphenyl)ethyl]amino]-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-1-oxo-3-phenylpropan-2-yl]hydrazinyl]-3-phenylpropanoyl]amino]-4-oxobutanoic acid
Show/Hide
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C55H65N9O14
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2
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| 1 |
IC50 = 53.7 nM
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| 2 |
Ki = 23 nM
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CP0372408
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(S)-2-((S)-2-(2-((R)-2-((S)-2-amino-3-(4-hydroxyphenyl)propanamido)propanamido)acetamido)-3-phenylpropanamido)-N-((S)-1-((S)-1-((S)-1-(3,5-bis(trifluoromethyl)benzylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-4-methyl-1-oxopentan-2-ylamino)-1-oxo-3-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yloxy)propan-2-yl)hexanamide
Show/Hide
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C64H80F6N10O15
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2
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| 1 |
IC50 = 75.86 nM
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| 2 |
Ki = 36 nM
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CP0431981
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Bifunctional Peptide Ligand, 3 (TY006)
Show/Hide
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C56H63F6N9O10
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2
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| 1 |
IC50 = 77.62 nM
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| 2 |
Ki = 36 nM
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CP0373038
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(3S,6S,9S,12S,15R,18S,21S,24R,27S)-18-((1H-imidazol-5-yl)methyl)-9-((1H-indol-3-yl)methyl)-27-amino-3-((S)-1-amino-1-oxo-3-phenylpropan-2-ylcarbamoyl)-21-benzyl-6-butyl-12-(3-guanidinopropyl)-28-(4-hydroxyphenyl)-24-methyl-15-(naphthalen-2-ylmethyl)-5,8,11,14,17,20,23,26-octaoxo-4,7,10,13,16,19,22,25-octaazaoctacosan-1-oic acid
Show/Hide
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C76H91N17O13
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2
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| 1 |
IC50 = 79.43 nM
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| 2 |
Ki = 42 nM
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CP0432554
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(3S)-3-[[(2S)-2-[2-[(2S)-1-[[2-[[(2R)-1-[[(1S)-1-carboxy-2-(4-hydroxyphenyl)ethyl]amino]-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-1-oxo-3-phenylpropan-2-yl]hydrazinyl]-3-phenylpropanoyl]amino]-4-[[(2S)-1-[[(1R)-1-carboxy-2-[1-[(2-methylpropan-2-yl)oxycarbonyl]indol-3-yl]ethyl]amino]-1-oxohexan-2-yl]amino]-4-oxobutanoic acid
Show/Hide
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C58H71N9O15
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2
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| 1 |
IC50 = 93.33 nM
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| 2 |
Ki = 45 nM
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CP0211343
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(3S)-3-{[(2S)-1-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenylpropanehydrazido]-1-oxo-3-phenylpropan-2-yl]carbamoyl}-3-[(2S)-2-[(2R)-2-{[(tert-butoxy)carbonyl]amino}-3-(1H-indol-2-yl)propanamido]hexanamido]propanoic acid
Show/Hide
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C58H73N11O13
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2
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| 1 |
IC50 = 93.33 nM
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| 2 |
Ki = 45 nM
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CP0373845
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(3S,6S,12S,17S,20S)-12-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-6-benzyl-N-[(2S)-1-[[3,5-bis(trifluoromethyl)phenyl]methylamino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-3-butyl-2,5,8,11,19-pentaoxo-14,15-dithia-1,4,7,10,18-pentazabicyclo[18.3.0]tricosane-17-carboxamide
Show/Hide
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C57H64F6N10O9S2
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2
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| 1 |
IC50 = 117.49 nM
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| 2 |
Ki = 54 nM
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CP0372407
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(S)-1-((2S,5S,11R,14S)-14-amino-5-benzyl-15-(4-hydroxyphenyl)-11-methyl-4,7,10,13-tetraoxo-2-(((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yloxy)methyl)-3,6,9,12-tetraazapentadecane)-N-((S)-1-((S)-1-(3,5-bis(trifluoromethyl)benzylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-4-methyl-1-oxopentan-2-yl)pyrrolidine-2-carboxamide
Show/Hide
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C63H76F6N10O15
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2
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| 1 |
IC50 = 123.03 nM
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| 2 |
Ki = 59 nM
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CP0403229
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(3S)-3-[[(2S)-2-[2-[(2S)-1-[[2-[[(2R)-1-[[(1S)-1-carboxy-2-(4-hydroxyphenyl)ethyl]amino]-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-1-oxo-3-phenylpropan-2-yl]hydrazinyl]-3-phenylpropanoyl]amino]-4-[[(2S)-1-[[(1S)-1-carboxy-2-[1-[(2-methylpropan-2-yl)oxycarbonyl]indol-3-yl]ethyl]amino]-1-oxohexan-2-yl]amino]-4-oxobutanoic acid
Show/Hide
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C58H71N9O15
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2
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| 1 |
IC50 = 138.04 nM
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| 2 |
Ki = 59 nM
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CP0394172
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Bifunctional Peptide Ligand, 8 (TY019)
Show/Hide
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C61H73F6N9O10
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2
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| 1 |
IC50 = 162.18 nM
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| 2 |
Ki = 77 nM
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CP0409706
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Bifunctional Peptide Ligand, 2 (TY007)
Show/Hide
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C63H69F6N9O10
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2
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| 1 |
IC50 = 199.53 nM
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| 2 |
Ki = 93 nM
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CP0099651
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(3S)-3-[(2S)-2-[(2S)-2-(2-{2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]acetamido}acetamido)-3-(1H-indol-3-yl)-N-methylpropanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C44H55N9O10
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2
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| 1 |
IC50 = 199.53 nM
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| 2 |
Ki = 85 nM
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CP0371822
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(3S)-3-[(2S)-2-[(2S)-2-(2-{[(2R)-1-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]pyrrolidin-2-yl]formamido}acetamido)-3-(1H-indol-3-yl)-N-methylpropanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C47H59N9O10
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2
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| 1 |
IC50 = 199.53 nM
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| 2 |
Ki = 85 nM
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CP0456236
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(3R)-2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-[(2R)-3-(4-chlorophenyl)-1-oxo-1-[4-(N-propanoylanilino)piperidin-1-yl]propan-2-yl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Show/Hide
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C44H50ClN5O5
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2
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| 1 |
IC50 = 275.42 nM
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| 2 |
Ki = 130 nM
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CP0451656
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(3S)-3-[(2S)-2-[(2R)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]-3-phenylpropanamido]acetamido}-3-(1H-indol-3-yl)propanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C50H59N9O10
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2
|
| 1 |
IC50 = 398.11 nM
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| 2 |
Ki = 170 nM
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CP0042886
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(3R)-2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-[(2R)-3-(4-chlorophenyl)-1-[4-cyclohexyl-4-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]-1-oxopropan-2-yl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Show/Hide
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C44H54ClN7O4
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2
|
| 1 |
IC50 = 524.81 nM
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| 2 |
Ki = 250 nM
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CP0371828
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(3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-[(3S)-3-amino-3-formamidopropanoic acid]-3-(4-hydroxyphenyl)propanamido]-3-phenylpropanamido]acetamido}-3-(1H-indol-3-yl)-N-methylpropanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C55H66N10O13
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2
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| 1 |
IC50 = 549.54 nM
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| 2 |
Ki = 250 nM
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CP0400844
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(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenylpropanamide
Show/Hide
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C23H29N5O5
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3
|
| 1 |
IC50 = 724.44 nM
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| 2 |
IC50 = 794.33 nM
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| 3 |
Ki = 300 nM
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CP0371834
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(3S)-3-[(2S)-2-[(2R)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]hexanamido]acetamido}-3-(1H-indol-3-yl)-N-methylpropanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C48H63N9O10
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2
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| 1 |
IC50 = 724.44 nM
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| 2 |
Ki = 310 nM
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CP0371865
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(3S)-3-[(2S)-2-[(2R)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-(1H-indol-3-yl)propanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C44H55N9O10
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2
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| 1 |
IC50 = 1995.26 nM
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| 2 |
Ki = 860 nM
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CP0388011
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(S)-3-((3S,6S,9S,12S,18R,26S)-12-((1H-imidazol-5-yl)methyl)-3-((1H-indol-2-yl)methyl)-18-((S)-2-amino-3-(4-hydroxyphenyl)propanamido)-9-(4-chlorobenzyl)-6-(3-guanidinopropyl)-2,5,8,11,14,17,20-heptaoxo-1,4,7,10,13,16,21-heptaazacyclohexacosane-26-carboxamido)-4-((R)-1-amino-1-oxo-3-phenylpropan-2-ylamino)-4-oxobutanoic acid
Show/Hide
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C66H81ClN18O14
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2
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| 1 |
IC50 = 2511.89 nM
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| 2 |
Ki = 1300 nM
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CP0442594
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(3S)-3-[(2S)-2-[(2S)-2-(2-{[(2S)-1-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]pyrrolidin-2-yl]formamido}acetamido)-3-(1H-indol-3-yl)-N-methylpropanamido]hexanamido]-3-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}propanoic acid
Show/Hide
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C47H59N9O10
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2
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| 1 |
IC50 = 3388.44 nM
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| 2 |
Ki = 1500 nM
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CP0388013
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(3S,6S,9S,12S,15R,18S)-18-((1H-imidazol-5-yl)methyl)-9-((1H-indol-3-yl)methyl)-3-((S)-1-amino-1-oxo-3-phenylpropan-2-ylcarbamoyl)-15-benzyl-6-butyl-12-(3-guanidinopropyl)-5,8,11,14,17,20,23-heptaoxo-23-((1-phenethylpiperidin-4-yl)(phenyl)amino)-4,7,10,13,16,19-hexaazatricosan-1-oic acid
Show/Hide
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C74H92N16O11
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2
|
| 1 |
IC50 = 5011.87 nM
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| 2 |
Ki = 2300 nM
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CP0198575
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N-[1-[[(5R)-5-amino-5,6,7,8-tetrahydronaphthalen-2-yl]methyl]piperidin-4-yl]-N-(4-chloro-3-methoxyphenyl)propanamide;2,2,2-trifluoroacetic acid
Show/Hide
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C28H35ClF3N3O4
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2
|
| 1 |
IC50 = 10000 nM
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| 2 |
Ki = 4500 nM
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CP0438224
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N-[1-[[(5R)-5-amino-5,6,7,8-tetrahydronaphthalen-2-yl]methyl]piperidin-4-yl]-N-(3,4-difluorophenyl)propanamide;2,2,2-trifluoroacetic acid
Show/Hide
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C27H32F5N3O3
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2
|
| 1 |
IC50 = 12302.69 nM
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| 2 |
Ki = 5700 nM
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CP0485809
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(2S)-2-amino-3-(4-hydroxyphenyl)-N-[(1R)-1-[({[(2S)-1-oxo-3-phenyl-1-[4-(N-phenylpropanamido)piperidin-1-yl]propan-2-yl]carbamoyl}methyl)carbamoyl]ethyl]propanamide
Show/Hide
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C37H46N6O6
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2
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| 1 |
IC50 = 13489.63 nM
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| 2 |
Ki = 7000 nM
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CP0120367
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N-[1-[[(5R)-5-amino-5,6,7,8-tetrahydronaphthalen-2-yl]methyl]piperidin-4-yl]-N-(3,4-dichlorophenyl)propanamide;2,2,2-trifluoroacetic acid
Show/Hide
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C27H32Cl2F3N3O3
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2
|
| 1 |
IC50 = 19498.45 nM
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| 2 |
Ki = 5200 nM
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CP0198574
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N-[[1-[[(5R)-5-amino-5,6,7,8-tetrahydronaphthalen-2-yl]methyl]piperidin-4-yl]methyl]-N-phenylpropanamide;2,2,2-trifluoroacetic acid
Show/Hide
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C28H36F3N3O3
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2
|
| 1 |
IC50 = 19498.45 nM
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| 2 |
Ki = 6000 nM
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CP0435259
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3-{phenyl[1-(2-phenylethyl)piperidin-4-yl]carbamoyl}propanoic acid
Show/Hide
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C23H28N2O3
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2
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| 1 |
IC50 = 19952.62 nM
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| 2 |
Ki = 9400 nM
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CP0357207
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N-[[1-[[(5S)-5-hydroxy-5,6,7,8-tetrahydronaphthalen-2-yl]methyl]piperidin-4-yl]methyl]-N-phenylpropanamide
Show/Hide
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C26H34N2O2
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2
|
| 1 |
IC50 = 25703.96 nM
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|
| 2 |
Ki = 7800 nM
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CP0190001
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(3S)-2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Show/Hide
|
C39H43N5O5
|
1
|
| 1 |
Ki = 0.12 nM
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|
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CP0369953
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(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-6-[[3-oxo-3-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)propyl]carbamoylamino]hexanoic acid
Show/Hide
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C75H100N16O12
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1
|
| 1 |
Ki = 0.26 nM
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|
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CP0369952
|
(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]-3-phenylpropanoyl]amino]-2-methylpropanoyl]amino]-3-methylbutanoyl]amino]-3-methylbutanoyl]amino]-N'-[2-oxo-2-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)ethyl]pentanediamide
Show/Hide
|
C61H83N11O10
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1
|
| 1 |
Ki = 0.28 nM
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|
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CP0087117
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(2S)-2-[[(2R)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-(4-chlorophenyl)propanoyl]amino]-4-methylpentanoyl]amino]-N-[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]-N'-[3-oxo-3-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)propyl]pentanediamide
Show/Hide
|
C64H88ClN11O10
|
1
|
| 1 |
Ki = 0.35 nM
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|
|
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CP0176551
|
(3S)-2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-[(2R)-3-(4-chlorophenyl)-1-oxo-1-[4-(N-propanoylanilino)piperidin-1-yl]propan-2-yl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Show/Hide
|
C44H50ClN5O5
|
1
|
| 1 |
Ki = 0.38 nM
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|
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CP0042126
|
(2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-(4-chlorophenyl)propanoyl]amino]-N-[(2S)-1-amino-1-oxo-3-(2,3,4,5,6-pentafluorophenyl)propan-2-yl]-N'-[6-oxo-6-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)hexyl]pentanediamide
Show/Hide
|
C62H72ClF5N10O9
|
1
|
| 1 |
Ki = 0.51 nM
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|
|
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CP0380169
|
(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-N-[(2S)-1-amino-1-oxo-3-(2,3,4,5,6-pentafluorophenyl)propan-2-yl]-N'-[6-oxo-6-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)hexyl]pentanediamide
Show/Hide
|
C74H96F5N15O11
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1
|
| 1 |
Ki = 0.63 nM
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|
|
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CP0100342
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(S)-2-amino-3-(4-hydroxy-phenyl)-N-((R)-1-{[((S)-1-{2-[(1-phenethyl-piperidin-4-yl)-phenyl-carbamoyl]-ethylcarbamoyl}-2-phenyl-ethylcarbamoyl)-methyl]-carbamoyl}-ethyl)-propionamide
Show/Hide
|
C45H55N7O6
|
1
|
| 1 |
Ki = 0.99 nM
|
|
|
|
CP0680488
|
(S)-2-amino-3-(4-hydroxyphenyl)-N-((R)-1-oxo-1-(2-oxo-2-((S)-1-oxo-1-(3-oxo-3-((1-phenethylpiperidin-4-yl)(phenyl)amino)propylamino)-3-phenylpropan-2-ylamino)ethylamino)propan-2-yl)propanamide hydrochloride
Show/Hide
|
C45H56ClN7O6
|
1
|
| 1 |
Ki = 1.1 nM
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|
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CP0337915
|
H-Dmt-Tic-NH2
Show/Hide
|
C21H25N3O3
|
1
|
| 1 |
Ki = 1.2 nM
|
|
|
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CP0061303
|
(2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenylpropanamido]-4-methylpentanoic acid
Show/Hide
|
C29H39N5O7
|
1
|
| 1 |
Ki = 1.3 nM
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|
|
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CP0377551
|
(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propionylamino]-5-guanidino-pentanoic acid [(S)-1-(2-carbamoyl-ethylcarbamoyl)-2-phenyl-ethyl]-amide
Show/Hide
|
C38H54N8O10
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
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CP0038418
|
13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7-benzyl-3,3,14,14-tetramethyl-6,9,12-trioxo-1,2-dithia-5,8,11-triaza-cyclotetradecane-4-carboxylic acid
Show/Hide
|
C30H39N5O7S2
|
1
|
| 1 |
Ki = 1.6 nM
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|
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CP0087118
|
(2S)-2-[[(2S)-2-[[(2S)-5-amino-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-(4-chlorophenyl)propanoyl]amino]-4-methylpentanoyl]amino]-5-carbamimidamidopentanoyl]amino]-5-carbamimidamidopentanoyl]amino]-5-oxopentanoyl]amino]-3-phenylpropanoyl]amino]-6-[[3-oxo-3-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)propyl]carbamoylamino]hexanoic acid
Show/Hide
|
C86H122ClN21O15
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1
|
| 1 |
Ki = 1.8 nM
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|
|
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CP0562220
|
(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenylpropanamido]-4-methylpentanamide
Show/Hide
|
C29H40N6O6
|
1
|
| 1 |
Ki = 2.4 nM
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|
|
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CP0266417
|
(2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]butanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methyl-N-[2-oxo-2-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)ethyl]pentanamide
Show/Hide
|
C51H66N8O7
|
1
|
| 1 |
Ki = 2.8 nM
|
|
|
|
CP0091844
|
BDBM50241435
Show/Hide
|
C75H126N24O15
|
1
|
| 1 |
Ki = 3.8 nM
|
|
|
|
CP0266403
|
(2S)-2-amino-3-(4-hydroxyphenyl)-N-[(2R)-1-oxo-1-[[2-oxo-2-[[(2S)-1-oxo-1-[[2-oxo-2-[[2-oxo-2-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)ethyl]amino]ethyl]amino]-3-phenylpropan-2-yl]amino]ethyl]amino]propan-2-yl]propanamide
Show/Hide
|
C46H56N8O7
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0336175
|
(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-5-carbamimidamidopentanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-phenylpropanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-N-[(2S)-1-amino-3-methyl-1-oxobutan-2-yl]-6-[[3-oxo-3-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)propyl]carbamoylamino]hexanamide
Show/Hide
|
C101H143N27O15
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1
|
| 1 |
Ki = 4.6 nM
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|
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CP0261470
|
(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-6-[[3-oxo-3-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)propyl]carbamoylamino]hexanoic acid
Show/Hide
|
C64H90N14O11
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1
|
| 1 |
Ki = 11 nM
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|
|
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CP0369954
|
(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methyl-N-[2-oxo-2-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)ethyl]pentanamide
Show/Hide
|
C49H62N8O7
|
1
|
| 1 |
Ki = 12 nM
|
|
|
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CP0087116
|
(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]-3-phenylpropanoyl]amino]-N-[(2S)-1-[[(2S)-1-[(2-amino-2-oxoethyl)amino]-3-methyl-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-N'-[2-oxo-2-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)ethyl]pentanediamide
Show/Hide
|
C59H79N11O10
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0100639
|
(2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methyl-N-[2-oxo-2-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)ethyl]pentanamide
Show/Hide
|
C50H64N8O7
|
1
|
| 1 |
Ki = 27 nM
|
|
|
|
CP0464563
|
(S)-N-(1-(2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl)piperidin-4-yl)-N-phenylpropionamide
Show/Hide
|
C25H33N3O3
|
1
|
| 1 |
Ki = 50 nM
|
|
|
|
CP0524728
|
(3R)-2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
Show/Hide
|
C21H25N3O3
|
1
|
| 1 |
Ki = 57 nM
|
|
|
|
CP0261448
|
(2S)-N-[(2S)-1-amino-3-(4-fluorophenyl)-1-oxopropan-2-yl]-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-(4-chlorophenyl)propanoyl]amino]-N'-[6-oxo-6-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)hexyl]pentanediamide
Show/Hide
|
C73H85ClFN11O9
|
1
|
| 1 |
Ki = 84 nM
|
|
|
|
CP0464564
|
N-[1-[(2S,3R)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)butanoyl]piperidin-4-yl]-N-phenylpropanamide
Show/Hide
|
C26H35N3O3
|
1
|
| 1 |
Ki = 260 nM
|
|
|
|
CP0042163
|
(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoyl]amino]-N'-[2-oxo-2-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)ethyl]pentanediamide
Show/Hide
|
C60H70N10O8
|
1
|
| 1 |
Ki = 590 nM
|
|
|
|
CP0112711
|
(2R)-1-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-N-[2-[[(2S)-1-[[(2S)-4-methyl-1-oxo-1-[[2-oxo-2-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)ethyl]amino]pentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-2-oxoethyl]pyrrolidine-2-carboxamide
Show/Hide
|
C52H66N8O7
|
1
|
| 1 |
Ki = 630 nM
|
|
|
|
CP0862673
|
(1S,4S,7R,10S)-11-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-4,7-dibenzyl-2,5,8,11-tetraazabicyclo[8.2.1]tridecane-3,6,9-trione 2,2,2-trifluoroacetate
Show/Hide
|
C34H36F3N5O7
|
1
|
| 1 |
Ki = 860 nM
|
|
|
|
CP0746439
|
(9H-fluoren-9-yl)methyl 2-oxo-2-((1-phenethylpiperidin-4-yl)(phenyl)amino)-ethylcarbamate hydrochloride
Show/Hide
|
C36H38ClN3O3
|
1
|
| 1 |
Ki = 1000 nM
|
|
|
|
CP0857344
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(1S,4R,7R,10S)-11-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-4,7-dibenzyl-2,5,8,11-tetraazabicyclo[8.2.1]tridecane-3,6,9-trione 2,2,2-trifluoroacetate
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C34H36F3N5O7
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1
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| 1 |
Ki = 1010 nM
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CP0445725
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N-[1-[(2S,3S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)butanoyl]piperidin-4-yl]-N-phenylpropanamide
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C26H35N3O3
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1
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| 1 |
Ki = 1700 nM
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CP0372417
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N-[1-[3-amino-3-(4-chlorophenyl)propanoyl]piperidin-4-yl]-N-phenylpropanamide
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C23H28ClN3O2
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1
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| 1 |
Ki = 2400 nM
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CP0526234
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N-[1-[3-amino-3-(4-methylphenyl)propanoyl]piperidin-4-yl]-N-phenylpropanamide
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C24H31N3O2
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1
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| 1 |
Ki = 2900 nM
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CP0372419
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(S)-N-(1-(2-amino-3-(naphthalen-2-yl)propanoyl)piperidin-4-yl)-N-phenylpropionamide
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C27H31N3O2
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1
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| 1 |
Ki = 3300 nM
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CP0304458
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N-[3-oxo-3-(N-[1-(2-phenylethyl)piperidin-4-yl]anilino)propyl]benzamide
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C29H33N3O2
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1
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| 1 |
Ki = 4600 nM
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CP0235395
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(S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrrolidine-2-carboxylic acid [(S)-1-((S)-1-carbamoyl-2-phenyl-ethylcarbamoyl)-2-(1H-indol-3-yl)-ethyl]-amide
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C34H38N6O5
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1
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| 1 |
Ki = 5100 nM
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CP0445726
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N-[1-[3-(3-chloro-4-methoxyphenyl)propanoyl]piperidin-4-yl]-N-phenylpropanamide
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C24H29ClN2O3
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1
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| 1 |
Ki = 6300 nM
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CP0434185
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(S)-N-(1-(2-amino-3,3-diphenylpropanoyl)piperidin-4-yl)-N-phenylpropionamide
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C29H33N3O2
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1
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| 1 |
Ki = 6500 nM
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CP0518076
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(S)-N-(1-(2-amino-3-phenylpropanoyl)piperidin-4-yl)-N-phenylpropionamide
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C23H29N3O2
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1
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| 1 |
Ki = 6900 nM
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CP0042160
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2-acetylamino-N-{2-[(1-phenethyl-piperidin-4-yl)-phenyl-carbamoyl]-ethyl}-3-phenyl-propionamide
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C33H40N4O3
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1
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| 1 |
Ki = 7600 nM
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CP0464598
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N-[1-[3-amino-3-(4-methoxyphenyl)propanoyl]piperidin-4-yl]-N-phenylpropanamide
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C24H31N3O3
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1
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| 1 |
Ki = 9000 nM
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CP0908289
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(R)-2-((R)-2-((2S,4S)-4-amino-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)pyrrolidine-2-carboxamido)-3-phenylpropanamido)-3-phenylpropanoic acid dihydrobromide
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C32H38BrN5O6
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1
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| 1 |
Ki > 10000 nM
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CP0120366
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N-[[1-[[(5R)-5-acetamido-5,6,7,8-tetrahydronaphthalen-2-yl]methyl]piperidin-4-yl]methyl]-N-phenylpropanamide
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C28H37N3O2
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1
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| 1 |
Ki > 10000 nM
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CP0158624
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N-[1-[[(5R)-5-amino-5,6,7,8-tetrahydronaphthalen-2-yl]methyl]piperidin-4-yl]-N-phenylpropanamide;2,2,2-trifluoroacetic acid
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C27H34F3N3O3
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1
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| 1 |
Ki > 10000 nM
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CP0210724
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N-[1-[2-[(5R)-5-amino-5,6,7,8-tetrahydronaphthalen-2-yl]ethyl]piperidin-4-yl]-N-phenylpropanamide;2,2,2-trifluoroacetic acid
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C28H36F3N3O3
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1
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| 1 |
Ki > 10000 nM
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CP0357206
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N-[1-[[(5S)-5-hydroxy-5,6,7,8-tetrahydronaphthalen-2-yl]methyl]piperidin-4-yl]-N-phenylpropanamide
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C25H32N2O2
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1
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| 1 |
Ki > 10000 nM
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CP0416785
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N-[1-[[(5R)-5-acetamido-5,6,7,8-tetrahydronaphthalen-2-yl]methyl]piperidin-4-yl]-N-phenylpropanamide
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C27H35N3O2
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1
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| 1 |
Ki > 10000 nM
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CP0445727
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N-[1-[3-(3-bromophenyl)propanoyl]piperidin-4-yl]-N-phenylpropanamide
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C23H27BrN2O2
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1
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| 1 |
Ki = 12000 nM
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CP0369951
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2-(1,3-dioxoisoindol-2-yl)-N-phenyl-N-[1-(2-phenylethyl)piperidin-4-yl]acetamide
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C29H30ClN3O3
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1
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| 1 |
Ki = 13000 nM
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CP0434186
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(S)-N-(1-(2-amino-3-(benzo[b]thiophen-3-yl)propanoyl)piperidin-4-yl)-N-phenylpropionamide
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C25H29N3O2S
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1
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| 1 |
Ki = 15000 nM
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CP0518075
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(S)-N-(1-(2-amino-2-(2,3-dihydro-1H-inden-2-yl)acetyl)piperidin-4-yl)-N-phenylpropionamide
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C25H31N3O2
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1
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| 1 |
Ki = 15000 nM
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CP0434183
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(S)-N-(1-(2-amino-3-(4-hydroxyphenyl)propanoyl)piperidin-4-yl)-N-phenylpropionamide
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C23H29N3O3
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1
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| 1 |
Ki = 16000 nM
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CP0672561
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2-(1,3-dioxoisoindolin-2-yl)-N-(1-phenethylpiperidin-4-yl)-N-phenylacetamide hydrochloride
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C29H30ClN3O3
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1
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| 1 |
Ki = 36000 nM
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CP0434187
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(S)-N-(1-(2-amino-3-(thiazol-4-yl)propanoyl)piperidin-4-yl)-N-phenylpropionamide
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C20H26N4O2S
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1
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| 1 |
Ki = 76000 nM
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