| Compound ID |
Compound Name |
Compound Formula |
|
CP0534826
|
(3R)-2-[(2S)-2-amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[2-[[(2S)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino]-2-oxoethyl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
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|
C46H51Cl2FN6O6
|
2
|
| 1 |
IC50 = 0.537 nM
|
|
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| 2 |
Ki = 0.13 nM
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CP0546858
|
(3R)-2-[(2S)-2-amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[2-[[(2S)-3-(4-chlorophenyl)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-1-oxopropan-2-yl]amino]-2-oxoethyl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
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|
C46H51Cl3N6O6
|
2
|
| 1 |
IC50 = 1.905 nM
|
|
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| 2 |
Ki = 0.53 nM
|
|
|
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CP0495192
|
(2R)-2-[[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]amino]-N-[2-[[(2S)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino]-2-oxoethyl]hexanamide
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|
C42H53Cl2FN6O6
|
2
|
| 1 |
IC50 = 6.026 nM
|
|
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| 2 |
Ki = 1.5 nM
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|
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CP0543991
|
(2S)-2-amino-N-[(2R)-1-[[2-[[(2S)-3-(4-chlorophenyl)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-1-oxopropan-2-yl]-3-(4-hydroxy-2,6-dimethylphenyl)propanamide
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|
C39H47Cl3N6O6
|
2
|
| 1 |
IC50 = 23.99 nM
|
|
|
| 2 |
Ki = 5.8 nM
|
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|
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CP0543992
|
(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-N-[2-[[(2S)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino]-2-oxoethyl]hexanamide
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|
C40H49Cl2FN6O6
|
2
|
| 1 |
IC50 = 83.18 nM
|
|
|
| 2 |
Ki = 20 nM
|
|
|
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CP0527959
|
(3R)-2-[(2S)-2-amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(2S)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-3-(4-fluorophenyl)-1-oxopropan-2-yl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
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|
C44H48Cl2FN5O5
|
2
|
| 1 |
IC50 = 97.72 nM
|
|
|
| 2 |
Ki = 28 nM
|
|
|
|
CP0551809
|
(3R)-2-[(2S)-2-amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(2S)-3-(4-chlorophenyl)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-1-oxopropan-2-yl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
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|
C44H48Cl3N5O5
|
2
|
| 1 |
IC50 = 123.03 nM
|
|
|
| 2 |
Ki = 34 nM
|
|
|
|
CP0534832
|
(2S)-2-amino-N-[(2R)-1-[[2-[[(2S)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-1-oxo-3-phenylpropan-2-yl]amino]-2-oxoethyl]amino]-1-oxopropan-2-yl]-3-(4-hydroxyphenyl)propanamide
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|
C37H44Cl2N6O6
|
2
|
| 1 |
IC50 = 181.97 nM
|
|
|
| 2 |
Ki = 44 nM
|
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|
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CP0534824
|
(2S)-2-amino-N-[(2R)-1-[[2-[[(2S)-3-(4-chlorophenyl)-1-[4-(3,4-dichloro-N-propanoylanilino)piperidin-1-yl]-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-1-oxopropan-2-yl]-3-(4-hydroxyphenyl)propanamide
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|
C37H43Cl3N6O6
|
2
|
| 1 |
IC50 = 190.55 nM
|
|
|
| 2 |
Ki = 47 nM
|
|
|
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CP0400844
|
(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamido]propanamido]acetamido}-3-phenylpropanamide
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|
C23H29N5O5
|
1
|
| 1 |
IC50 = 223.87 nM
|
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