| Compound ID |
Compound Name |
Compound Formula |
|
CP0206826
|
(2S)-2-[[5-[3-(2-amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)propyl]thiophene-3-carbonyl]amino]pentanedioic acid
Show/Hide
|
C19H21N5O6S
|
2
|
| 1 |
IC50 = 0.1 nM
|
|
|
| 2 |
IC50 = 654 nM
|
|
|
|
CP0055020
|
AGF94
Show/Hide
|
C19H21N5O6S
|
3
|
| 1 |
IC50 = 0.17 nM
|
|
|
| 2 |
IC50 = 126 nM
|
|
|
| 3 |
IC50 > 1000 nM
|
|
|
|
CP0374708
|
(2S)-2-[[4-[3-(2-amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)propyl]thiophene-2-carbonyl]amino]pentanedioic acid
Show/Hide
|
C19H21N5O6S
|
2
|
| 1 |
IC50 = 0.34 nM
|
|
|
| 2 |
IC50 = 557 nM
|
|
|
|
CP0386884
|
(2S)-2-[[5-[3-(2-amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)propyl]thiophene-2-carbonyl]amino]hexanedioic acid
Show/Hide
|
C20H23N5O6S
|
2
|
| 1 |
IC50 = 3.6 nM
|
|
|
| 2 |
IC50 > 1000 nM
|
|
|
|
CP0374709
|
(2S)-2-[[4-[3-(2,4-diaminofuro[2,3-d]pyrimidin-5-yl)propyl]thiophene-2-carbonyl]amino]pentanedioic acid
Show/Hide
|
C19H21N5O6S
|
2
|
| 1 |
IC50 = 17.5 nM
|
|
|
| 2 |
IC50 > 1000 nM
|
|
|
|
CP0041026
|
(2S)-2-[(5-{methyl[(2-methyl-4-oxo-1,4-dihydroquinazolin-6-yl)methyl]amino}thiophen-2-yl)formamido]pentanedioic acid
Show/Hide
|
C21H22N4O6S
|
2
|
| 1 |
IC50 = 22 nM
|
|
|
| 2 |
IC50 = 746 nM
|
|
|
|
CP0374710
|
(2S)-2-[[5-[3-(2,4-diaminofuro[2,3-d]pyrimidin-5-yl)propyl]thiophene-3-carbonyl]amino]pentanedioic acid
Show/Hide
|
C19H21N5O6S
|
2
|
| 1 |
IC50 = 54.3 nM
|
|
|
| 2 |
IC50 > 1000 nM
|
|
|
|
CP0036368
|
(2S)-2-{[4-(2-{2-amino-4-oxo-1H,4H,7H-pyrrolo[2,3-d]pyrimidin-5-yl}ethyl)phenyl]formamido}pentanedioic acid
Show/Hide
|
C20H21N5O6
|
2
|
| 1 |
IC50 = 60 nM
|
|
|
| 2 |
IC50 = 254 nM
|
|
|
|
CP0036197
|
2-[(4-{[(2,4-diaminopteridin-6-yl)methyl](methyl)amino}phenyl)formamido]pentanedioic acid
Show/Hide
|
C20H22N8O5
|
2
|
| 1 |
IC50 = 106 nM
|
|
|
| 2 |
IC50 = 211 nM
|
|
|
|
CP0419800
|
(2S)-2-[[5-[3-(2-amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)propyl]thiophene-2-carbonyl]amino]butanedioic acid
Show/Hide
|
C18H19N5O6S
|
2
|
| 1 |
IC50 = 347 nM
|
|
|
| 2 |
IC50 > 1000 nM
|
|
|
|
CP0379858
|
(2S)-2-[[5-[3-(2-amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)propyl]thiophene-2-carbonyl]amino]pentanoic acid
Show/Hide
|
C19H23N5O4S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0386883
|
4-[[5-[3-(2-amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)propyl]thiophene-2-carbonyl]amino]butanoic acid
Show/Hide
|
C18H21N5O4S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0411313
|
5-[3-(2-amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)propyl]thiophene-2-carboxylic acid
Show/Hide
|
C14H14N4O3S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
