| Compound ID |
Compound Name |
Compound Formula |
|
CP0503792
|
1-[(S)-2-Amino-3-(3-methyl-3H-imidazol-4-yl)-propionyl]-5-oxo-pyrrolidine-2-carboxylic acid {2-((S)-2-carbamoyl-pyrrolidin-1-yl)-1-[(S)-1-(1H-imidazol-4-yl)methyl]-2-oxo-ethyl}-amide
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|
C23H31N9O5
|
2
|
| 1 |
EC50 = 0.5 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0067202
|
1-[3-(1H-4-imidazolyl)-2-(5-oxotetrahydro-1H-2-pyrrolylcarboxamido)propanoyl]tetrahydro-1H-2-pyrrolecarboxamide
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|
C16H22N6O4
|
2
|
| 1 |
EC50 = 3 nM
|
|
|
| 2 |
Ki = 20 nM
|
|
|
|
CP0408102
|
1-[2-[5-oxo-(2S)-tetrahydro-1H-2-pyrrolylcarboxamido]-3-(2-propyl-1H-4-imidazolyl)-(2S)-propanoyl]-(2S)-tetrahydro-1H-2-pyrrolecarboxamide
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|
C19H28N6O4
|
2
|
| 1 |
EC50 = 290 nM
|
|
|
| 2 |
Ki = 320 nM
|
|
|
|
CP0381542
|
1-[3-[2-(tert-butyl)-1H-4-imidazolyl]-2-[5-oxo-(2S)-tetrahydro-1H-2-pyrrolylcarboxamido]-(2S)-propanoyl]-(2S)-tetrahydro-1H-2-pyrrolecarboxamide
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|
C20H30N6O4
|
2
|
| 1 |
EC50 > 100000 nM
|
|
|
| 2 |
Ki > 100000 nM
|
|
|
|
CP0391620
|
1-[3-{2-[1-(1-adamantyl)ethyl]-1H-4-imidazolyl}-2-[5-oxo-(2S)-tetrahydro-1H-2-pyrrolylcarboxamido]-(2S)-propanoyl]-(2S)-tetrahydro-1H-2-pyrrolecarboxamide
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|
C26H36N6O4
|
2
|
| 1 |
EC50 > 100000 nM
|
|
|
| 2 |
Ki > 100000 nM
|
|
|
|
CP0393980
|
1-[3-(2-cyclohexyl-1H-4-imidazolyl)-2-[5-oxo-(2S)-tetrahydro-1H-2-pyrrolylcarboxamido]-(2S)-propanoyl]-(2S)-tetrahydro-1H-2-pyrrolecarboxamide
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|
C22H32N6O4
|
2
|
| 1 |
EC50 > 100000 nM
|
|
|
| 2 |
Ki > 100000 nM
|
|
|
|
CP0431207
|
1-[3-(2-isopropyl-1H-4-imidazolyl)-2-[5-oxo-(2S)-tetrahydro-1H-2-pyrrolylcarboxamido]-(2S)-propanoyl]-(2S)-tetrahydro-1H-2-pyrrolecarboxamide
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|
C19H28N6O4
|
2
|
| 1 |
EC50 > 100000 nM
|
|
|
| 2 |
Ki > 100000 nM
|
|
|
|
CP0497471
|
1-[3-(2-cyclopropyl-1H-4-imidazolyl)-2-[5-oxo-(2S)-tetrahydro-1H-2-pyrrolylcarboxamido]-(2S)-propanoyl]-(2S)-tetrahydro-1H-2-pyrrolecarboxamide
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|
C19H26N6O4
|
2
|
| 1 |
EC50 > 100000 nM
|
|
|
| 2 |
Ki > 100000 nM
|
|
|
