Compound ID |
Compound Name |
Compound Formula |
CP0427334
|
N-[[(1R,3S)-3-(9-chloro-3-methyl-4-oxo-[1,2]oxazolo[4,3-c]quinolin-5-yl)cyclohexyl]methyl]benzamide
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|
C25H24ClN3O3
|
1
|
1 |
EC50 = 93 nM
|
|
|
CP0503983
|
N-[4-[6-hydroxy-3-[4-(2-piperidin-1-ylethoxy)benzoyl]-1-benzothiophen-2-yl]phenyl]-N-methylsulfonylmethanesulfonamide
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|
C30H32N2O7S3
|
1
|
1 |
IC50 = 800 nM
|
|
|
CP0393257
|
2-(3-(9-chloro-3-methyl-4-oxoisoxazolo[4,3-c]quinolin-5(4H)-yl)phenyl)-N-(3,4,5-trimethoxyphenyl)acetamide
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|
C28H24ClN3O6
|
1
|
1 |
IC50 = 1800 nM
|
|
|
CP0078757
|
(E)-3-((3-(2-(7-chloroquinolin-2-yl)vinyl)phenyl)(3-(dimethylamino)-3-oxopropylthio)methylthio)propanoic acid
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|
C26H27ClN2O3S2
|
2
|
1 |
IC50 = 3300 nM
|
|
|
2 |
Ki = 600 nM
|
|
|