| Compound ID |
Compound Name |
Compound Formula |
|
CP0008188
|
methyl 2-[(4-methylpiperazine-1-carbonyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
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|
C16H23N3O3S
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0466462
|
7-fluoro-4-hydroxy-12-methyl-2-oxo-N-(pyridin-3-ylmethyl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraene-3-carboxamide
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|
C20H18FN3O3
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0455856
|
N-[(6-aminopyridin-3-yl)methyl]-7-fluoro-4-hydroxy-12-methyl-2-oxo-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraene-3-carboxamide
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|
C20H19FN4O3
|
1
|
| 1 |
EC50 = 320 nM
|
|
|
|
CP0520072
|
ethyl 2-[(4-methylpiperazine-1-carbonyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
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|
C17H25N3O3S
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0542254
|
methyl 2-[(4-methylpiperazine-1-carbonyl)amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
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|
C15H21N3O3S
|
1
|
| 1 |
EC50 = 450 nM
|
|
|
|
CP0396963
|
ethyl 2-[(4-methylpiperazine-1-carbonyl)amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
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|
C16H23N3O3S
|
1
|
| 1 |
EC50 = 560 nM
|
|
|
|
CP0455857
|
7-fluoro-N-[(5-fluoropyridin-3-yl)methyl]-4-hydroxy-12-methyl-2-oxo-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraene-3-carboxamide
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|
C20H17F2N3O3
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0491821
|
methyl 2-[(4-methylpiperazine-1-carbonyl)amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
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|
C17H25N3O3S
|
1
|
| 1 |
EC50 = 1330 nM
|
|
|
|
CP0438170
|
7-fluoro-4-hydroxy-12-methyl-2-oxo-N-(2-pyridin-3-ylethyl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraene-3-carboxamide
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|
C21H20FN3O3
|
1
|
| 1 |
EC50 = 1350 nM
|
|
|
|
CP0575920
|
7-fluoro-4-hydroxy-12-methyl-N-[(4-methylpyridin-3-yl)methyl]-2-oxo-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraene-3-carboxamide
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|
C21H20FN3O3
|
1
|
| 1 |
EC50 = 1450 nM
|
|
|
|
CP0427046
|
N-(6,7-dihydro-5H-cyclopenta[b]pyridin-5-yl)-7-fluoro-4-hydroxy-12-methyl-2-oxo-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraene-3-carboxamide
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|
C22H20FN3O3
|
1
|
| 1 |
EC50 = 3000 nM
|
|
|
|
CP0578847
|
N-[[2-(dimethylamino)pyridin-3-yl]methyl]-7-fluoro-4-hydroxy-12-methyl-2-oxo-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraene-3-carboxamide
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|
C22H23FN4O3
|
1
|
| 1 |
EC50 = 3200 nM
|
|
|
|
CP0520071
|
ethyl 2-[(4-methylpiperazine-1-carbothioyl)amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
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|
C16H23N3O2S2
|
1
|
| 1 |
EC50 = 3460 nM
|
|
|
|
CP0550710
|
propan-2-yl 2-[(4-methylpiperazine-1-carbonyl)amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
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|
C17H25N3O3S
|
1
|
| 1 |
EC50 = 4590 nM
|
|
|
|
CP0484218
|
N-[(6-chloropyridin-3-yl)methyl]-7-fluoro-4-hydroxy-12-methyl-2-oxo-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraene-3-carboxamide
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|
C20H17ClFN3O3
|
1
|
| 1 |
EC50 = 5000 nM
|
|
|
|
CP0575417
|
ethyl 2-[(4-methylpiperazine-1-carbothioyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
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|
C17H25N3O2S2
|
1
|
| 1 |
EC50 = 6430 nM
|
|
|
|
CP0549723
|
propyl 2-[(4-methylpiperazine-1-carbonyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
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|
C18H27N3O3S
|
1
|
| 1 |
EC50 = 6630 nM
|
|
|
|
CP0561422
|
ethyl 2-[(4-ethylpiperazine-1-carbonyl)amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
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|
C17H25N3O3S
|
1
|
| 1 |
EC50 = 8550 nM
|
|
|
|
CP0542255
|
methyl 6-methyl-2-[(4-methylpiperazine-1-carbonyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
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|
C17H25N3O3S
|
1
|
| 1 |
EC50 = 11820 nM
|
|
|
|
CP0438557
|
propyl 2-[(4-methylpiperazine-1-carbonyl)amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
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|
C17H25N3O3S
|
1
|
| 1 |
EC50 = 14160 nM
|
|
|
|
CP0553253
|
propan-2-yl 2-[(4-methylpiperazine-1-carbothioyl)amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
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|
C17H25N3O2S2
|
1
|
| 1 |
EC50 = 16380 nM
|
|
|
|
CP0541649
|
propan-2-yl 2-[(4-methylpiperazine-1-carbothioyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
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|
C18H27N3O2S2
|
1
|
| 1 |
EC50 = 45240 nM
|
|
|
