| Compound ID |
Compound Name |
Compound Formula |
|
CP0168549
|
2-[4-[4,7-difluoro-5-(1-propylsulfonyl-3,6-dihydro-2H-pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]piperidin-1-yl]-5-propylpyrimidine
Show/Hide
|
C28H36F2N4O3S
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0486422
|
N-ethyl-4-[3-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]triazolo[4,5-c]pyridin-6-yl]-2,5-difluorobenzamide
Show/Hide
|
C25H26F2N8O
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0445889
|
1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-5-(2-fluoro-4-methylsulfonylphenyl)pyrazolo[3,4-c]pyridine
Show/Hide
|
C24H25FN6O2S
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0401513
|
2-[4-[4-fluoro-5-(1-propylsulfonyl-3,6-dihydro-2H-pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]piperidin-1-yl]-5-propylpyrimidine
Show/Hide
|
C28H37FN4O3S
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0570280
|
3-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-6-(2-fluoro-4-methylsulfonylphenyl)triazolo[4,5-c]pyridine
Show/Hide
|
C23H24FN7O2S
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0469670
|
propan-2-yl 2-[3-[4-(cyclopropylcarbamoyl)-3-fluorophenoxy]propyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C25H35FN2O4
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0474892
|
3-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-6-(3-fluoro-4-methylsulfonylphenyl)triazolo[4,5-c]pyridine
Show/Hide
|
C23H24FN7O2S
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0516007
|
tert-butyl 2-[3-(3-fluoro-4-methylsulfonylphenoxy)propyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C23H34FNO5S
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0474920
|
propan-2-yl 4-[5-[4-(ethylcarbamoyl)-2,5-difluorophenyl]pyrazolo[3,4-c]pyridin-1-yl]piperidine-1-carboxylate
Show/Hide
|
C24H27F2N5O3
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0520713
|
(1,1-difluoro-2-methylpropan-2-yl) 4-[5-(2-fluoro-4-methylsulfonylphenyl)pyrazolo[3,4-c]pyridin-1-yl]piperidine-1-carboxylate
Show/Hide
|
C23H25F3N4O4S
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0563272
|
N-ethyl-4-[3-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]triazolo[4,5-c]pyridin-6-yl]-2,3-difluorobenzamide
Show/Hide
|
C25H26F2N8O
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0459805
|
2-methylpropyl 4-[5-(4-methylsulfonylphenyl)pyrazolo[3,4-c]pyridin-1-yl]piperidine-1-carboxylate
Show/Hide
|
C23H28N4O4S
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
|
CP0443222
|
1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-5-(4-methylsulfonylphenyl)pyrazolo[3,4-c]pyridine
Show/Hide
|
C24H26N6O2S
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0474925
|
3-chloro-N-ethyl-4-[3-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]triazolo[4,5-c]pyridin-6-yl]benzamide
Show/Hide
|
C25H27ClN8O
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0444422
|
(1-methylcyclopropyl) 2-[3-(3-fluoro-4-methylsulfonylphenoxy)propyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C23H32FNO5S
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0495194
|
2-[4-[5-(1-propylsulfonyl-3,6-dihydro-2H-pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]piperidin-1-yl]-5-(trifluoromethyl)pyrimidine
Show/Hide
|
C26H31F3N4O3S
|
1
|
| 1 |
EC50 = 14 nM
|
|
|
|
CP0420553
|
propan-2-yl 4-[5-[2,5-difluoro-4-(propylcarbamoyl)phenyl]pyrazolo[3,4-c]pyridin-1-yl]piperidine-1-carboxylate
Show/Hide
|
C25H29F2N5O3
|
1
|
| 1 |
EC50 = 14 nM
|
|
|
|
CP0474939
|
1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-5-(4-methylsulfonylphenyl)indazole
Show/Hide
|
C25H27N5O2S
|
1
|
| 1 |
EC50 = 14 nM
|
|
|
|
CP0519926
|
tert-butyl 2-[3-(4-methylsulfonylphenoxy)propyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C23H35NO5S
|
1
|
| 1 |
EC50 = 14 nM
|
|
|
|
CP0530951
|
4-[1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]pyrazolo[3,4-c]pyridin-5-yl]-2,5-difluoro-N-(2-hydroxyethyl)benzamide
Show/Hide
|
C26H27F2N7O2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0483079
|
N-ethyl-4-[3-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]triazolo[4,5-c]pyridin-6-yl]-3-fluorobenzamide
Show/Hide
|
C25H27FN8O
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0550680
|
3-[[4-[4,7-difluoro-2-[1-(5-propylpyrimidin-2-yl)piperidin-4-yl]-2,3-dihydro-1-benzofuran-5-yl]-3,6-dihydro-2H-pyridin-1-yl]sulfonyl]propan-1-ol
Show/Hide
|
C28H36F2N4O4S
|
1
|
| 1 |
EC50 = 16 nM
|
|
|
|
CP0483080
|
N-ethyl-4-[3-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]triazolo[4,5-c]pyridin-6-yl]-2-methylbenzamide
Show/Hide
|
C26H30N8O
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0554708
|
2-chloro-N-ethyl-4-[3-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]triazolo[4,5-c]pyridin-6-yl]benzamide
Show/Hide
|
C25H27ClN8O
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0444423
|
propan-2-yl 2-[3-(3-fluoro-4-methylsulfonylphenoxy)propyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C22H32FNO5S
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
|
CP0512810
|
N-ethyl-4-[3-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]triazolo[4,5-c]pyridin-6-yl]-3-methylbenzamide
Show/Hide
|
C26H30N8O
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
|
CP0420558
|
tert-butyl 4-[5-(4-methylsulfonylphenyl)pyrazolo[3,4-c]pyridin-1-yl]piperidine-1-carboxylate
Show/Hide
|
C23H28N4O4S
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0573986
|
3-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-6-(4-methylsulfonylphenyl)triazolo[4,5-c]pyridine
Show/Hide
|
C23H25N7O2S
|
1
|
| 1 |
EC50 = 21 nM
|
|
|
|
CP0512809
|
(1,1-difluoro-2-methylpropan-2-yl) 4-[5-(4-methylsulfonylphenyl)pyrazolo[3,4-c]pyridin-1-yl]piperidine-1-carboxylate
Show/Hide
|
C23H26F2N4O4S
|
1
|
| 1 |
EC50 = 23 nM
|
|
|
|
CP0518058
|
cyclopentyl 2-[3-(3-fluoro-4-methylsulfonylphenoxy)propyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C24H34FNO5S
|
1
|
| 1 |
EC50 = 23 nM
|
|
|
|
CP0514932
|
tert-butyl 2-[3-(2-fluoro-4-methylsulfonylphenoxy)propyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C23H34FNO5S
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0420696
|
propan-2-yl 4-[5-(2-fluoro-4-methylsulfonylphenyl)pyrazolo[3,4-c]pyridin-1-yl]piperidine-1-carboxylate
Show/Hide
|
C22H25FN4O4S
|
1
|
| 1 |
EC50 = 27 nM
|
|
|
|
CP0558781
|
N-ethyl-4-[3-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]triazolo[4,5-c]pyridin-6-yl]-2,6-dimethylbenzamide
Show/Hide
|
C27H32N8O
|
1
|
| 1 |
EC50 = 27 nM
|
|
|
|
CP0495196
|
4-[[4-[2-methyl-2-[1-(5-propylpyrimidin-2-yl)piperidin-4-yl]-3H-1-benzofuran-5-yl]-3,6-dihydro-2H-pyridin-1-yl]sulfonyl]butan-1-ol
Show/Hide
|
C30H42N4O4S
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0575014
|
propan-2-yl 2-[3-[3-fluoro-4-(pyrrolidine-1-carbonyl)phenoxy]propyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C26H37FN2O4
|
1
|
| 1 |
EC50 = 29 nM
|
|
|
|
CP0455218
|
1-[1-(5-methylpyridin-2-yl)piperidin-4-yl]-5-(4-methylsulfonylphenyl)pyrazolo[3,4-c]pyridine
Show/Hide
|
C24H25N5O2S
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0420556
|
tert-butyl 4-[5-(4-methylsulfonylphenyl)indazol-1-yl]piperidine-1-carboxylate
Show/Hide
|
C24H29N3O4S
|
1
|
| 1 |
EC50 = 31 nM
|
|
|
|
CP0554709
|
1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-5-(4-methylsulfonylphenyl)benzotriazole
Show/Hide
|
C24H26N6O2S
|
1
|
| 1 |
EC50 = 31 nM
|
|
|
|
CP0550428
|
7-(5-ethylpyrimidin-2-yl)-2-[3-(4-methylsulfonylphenoxy)propyl]-7-azaspiro[3.5]nonane
Show/Hide
|
C24H33N3O3S
|
1
|
| 1 |
EC50 = 31 nM
|
|
|
|
CP0574976
|
2,2-dimethylpropyl 2-[3-(3-fluoro-4-methylsulfonylphenoxy)propyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C24H36FNO5S
|
1
|
| 1 |
EC50 = 31 nM
|
|
|
|
CP0495570
|
propan-2-yl 4-[6-[2,5-difluoro-4-(propan-2-ylcarbamoyl)phenyl]triazolo[4,5-c]pyridin-3-yl]piperidine-1-carboxylate
Show/Hide
|
C24H28F2N6O3
|
1
|
| 1 |
EC50 = 33 nM
|
|
|
|
CP0495195
|
2-[4-[5-(1-propylsulfonyl-3,6-dihydro-2H-pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]piperidin-1-yl]-5-(trifluoromethyl)pyridine
Show/Hide
|
C27H32F3N3O3S
|
1
|
| 1 |
EC50 = 34 nM
|
|
|
|
CP0559919
|
propan-2-yl 2-[3-[4-(azetidine-1-carbonyl)-3-fluorophenoxy]propyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C25H35FN2O4
|
1
|
| 1 |
EC50 = 34 nM
|
|
|
|
CP0489788
|
5-[2-[3-(4-methylsulfonylphenoxy)propyl]-7-azaspiro[3.5]nonan-7-yl]-3-propan-2-yl-1,2,4-oxadiazole
Show/Hide
|
C23H33N3O4S
|
1
|
| 1 |
EC50 = 35 nM
|
|
|
|
CP0573985
|
propan-2-yl 4-[6-[4-(ethylcarbamoyl)-2,5-difluorophenyl]triazolo[4,5-c]pyridin-3-yl]piperidine-1-carboxylate
Show/Hide
|
C23H26F2N6O3
|
1
|
| 1 |
EC50 = 37 nM
|
|
|
|
CP0474891
|
N-ethyl-4-[3-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]triazolo[4,5-c]pyridin-6-yl]-2-(trifluoromethyl)benzamide
Show/Hide
|
C26H27F3N8O
|
1
|
| 1 |
EC50 = 39 nM
|
|
|
|
CP0575015
|
propan-2-yl 2-[3-[3-fluoro-4-(3-hydroxyazetidine-1-carbonyl)phenoxy]propyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C25H35FN2O5
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0420559
|
propan-2-yl 4-[5-(4-methylsulfonylphenyl)pyrazolo[3,4-c]pyridin-1-yl]piperidine-1-carboxylate
Show/Hide
|
C22H26N4O4S
|
1
|
| 1 |
EC50 = 42 nM
|
|
|
|
CP0420677
|
propan-2-yl 4-[5-[4-(dimethylcarbamoyl)-2,5-difluorophenyl]pyrazolo[3,4-c]pyridin-1-yl]piperidine-1-carboxylate
Show/Hide
|
C24H27F2N5O3
|
1
|
| 1 |
EC50 = 46 nM
|
|
|
|
CP0521665
|
propan-2-yl 2-[3-[6-(cyclopropylcarbamoyl)pyridin-3-yl]oxypropyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C24H35N3O4
|
1
|
| 1 |
EC50 = 47 nM
|
|
|
|
CP0518063
|
propan-2-yl 2-[3-[4-[(2-amino-2-oxoethyl)carbamoyl]-3-fluorophenoxy]propyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C24H34FN3O5
|
1
|
| 1 |
EC50 = 48 nM
|
|
|
|
CP0495193
|
cyclohexyl 4-[5-(1-propylsulfonyl-3,6-dihydro-2H-pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]piperidine-1-carboxylate
Show/Hide
|
C28H40N2O5S
|
1
|
| 1 |
EC50 = 51 nM
|
|
|
|
CP0474152
|
propan-2-yl 4-[5-(4-carbamoyl-2,5-difluorophenyl)pyrazolo[3,4-c]pyridin-1-yl]piperidine-1-carboxylate
Show/Hide
|
C22H23F2N5O3
|
1
|
| 1 |
EC50 = 52 nM
|
|
|
|
CP0518062
|
propan-2-yl 2-[3-(4-carbamoyl-3-fluorophenoxy)propyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C22H31FN2O4
|
1
|
| 1 |
EC50 = 52 nM
|
|
|
|
CP0516006
|
tert-butyl 9-[2-(4-methylsulfonylphenoxy)ethyl]-3-azaspiro[5.5]undecane-3-carboxylate
Show/Hide
|
C24H37NO5S
|
1
|
| 1 |
EC50 = 55 nM
|
|
|
|
CP0550682
|
4-[[4-[7-fluoro-2-[1-(5-propylpyrimidin-2-yl)piperidin-4-yl]-2,3-dihydro-1-benzofuran-5-yl]-3,6-dihydro-2H-pyridin-1-yl]sulfonyl]butan-1-ol
Show/Hide
|
C29H39FN4O4S
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0512811
|
N-ethyl-4-[3-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]triazolo[4,5-c]pyridin-6-yl]-3-(trifluoromethyl)benzamide
Show/Hide
|
C26H27F3N8O
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0512808
|
propan-2-yl 4-[6-[4-(azetidine-1-carbonyl)-2,5-difluorophenyl]triazolo[4,5-c]pyridin-3-yl]piperidine-1-carboxylate
Show/Hide
|
C24H26F2N6O3
|
1
|
| 1 |
EC50 = 61 nM
|
|
|
|
CP0434958
|
2-[4-[7-fluoro-5-(1-propylsulfonyl-3,6-dihydro-2H-pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]piperidin-1-yl]-5-propylpyrimidine
Show/Hide
|
C28H37FN4O3S
|
1
|
| 1 |
EC50 = 62 nM
|
|
|
|
CP0445892
|
tert-butyl 4-[5-(4-methylsulfonylphenyl)benzotriazol-1-yl]piperidine-1-carboxylate
Show/Hide
|
C23H28N4O4S
|
1
|
| 1 |
EC50 = 63 nM
|
|
|
|
CP0387129
|
propan-2-yl 2-[3-[5-(cyclopropylcarbamoyl)pyridin-2-yl]oxypropyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C24H35N3O4
|
1
|
| 1 |
EC50 = 63 nM
|
|
|
|
CP0558780
|
propan-2-yl 4-[6-[2,5-difluoro-4-(pyrrolidine-1-carbonyl)phenyl]triazolo[4,5-c]pyridin-3-yl]piperidine-1-carboxylate
Show/Hide
|
C25H28F2N6O3
|
1
|
| 1 |
EC50 = 65 nM
|
|
|
|
CP0440296
|
5-cyclopropyl-2-[4-[5-(1-propylsulfonyl-3,6-dihydro-2H-pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]piperidin-1-yl]pyrimidine
Show/Hide
|
C28H36N4O3S
|
1
|
| 1 |
EC50 = 67 nM
|
|
|
|
CP0387128
|
propan-2-yl 2-[3-[4-[cyclopropyl(methyl)carbamoyl]-3-fluorophenoxy]propyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C26H37FN2O4
|
1
|
| 1 |
EC50 = 67 nM
|
|
|
|
CP0435110
|
2-[4-[2-methyl-5-(1-propylsulfonyl-3,6-dihydro-2H-pyridin-4-yl)-3H-1-benzofuran-2-yl]piperidin-1-yl]-5-propylpyrimidine
Show/Hide
|
C29H40N4O3S
|
1
|
| 1 |
EC50 = 70 nM
|
|
|
|
CP0512813
|
1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-6-methyl-5-(4-methylsulfonylphenyl)indazole
Show/Hide
|
C26H29N5O2S
|
1
|
| 1 |
EC50 = 70 nM
|
|
|
|
CP0440294
|
5-chloro-2-[4-[5-(1-propylsulfonyl-3,6-dihydro-2H-pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]piperidin-1-yl]pyrimidine
Show/Hide
|
C25H31ClN4O3S
|
1
|
| 1 |
EC50 = 78 nM
|
|
|
|
CP0571207
|
3-[[4-[2-methyl-2-[1-(5-propylpyrimidin-2-yl)piperidin-4-yl]-3H-1-benzofuran-5-yl]-3,6-dihydro-2H-pyridin-1-yl]sulfonyl]propan-1-ol
Show/Hide
|
C29H40N4O4S
|
1
|
| 1 |
EC50 = 78 nM
|
|
|
|
CP0514931
|
propan-2-yl 2-[3-(4-methylsulfonylphenoxy)propyl]-7-azaspiro[3.5]nonane-7-carboxylate
Show/Hide
|
C22H33NO5S
|
1
|
| 1 |
EC50 = 78 nM
|
|
|
|
CP0410112
|
5-propyl-2-[4-[5-(1-propylsulfonyl-3,6-dihydro-2H-pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]piperidin-1-yl]pyrimidine
Show/Hide
|
C28H38N4O3S
|
1
|
| 1 |
EC50 = 82 nM
|
|
|
|
CP0512812
|
N-ethyl-4-[3-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]triazolo[4,5-c]pyridin-6-yl]-3,5-dimethylbenzamide
Show/Hide
|
C27H32N8O
|
1
|
| 1 |
EC50 = 83 nM
|
|
|
|
CP0447769
|
propan-2-yl 4-[5-[2,5-difluoro-4-(2-hydroxyethylcarbamoyl)phenyl]pyrazolo[3,4-c]pyridin-1-yl]piperidine-1-carboxylate
Show/Hide
|
C24H27F2N5O4
|
1
|
| 1 |
EC50 = 92 nM
|
|
|
|
CP0570904
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propan-2-yl 4-[5-(4-carbamoyl-2-fluorophenyl)pyrazolo[3,4-c]pyridin-1-yl]piperidine-1-carboxylate
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C22H24FN5O3
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1
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| 1 |
EC50 = 97 nM
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CP0410113
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4-[[4-[4,7-difluoro-2-[1-(5-propylpyrimidin-2-yl)piperidin-4-yl]-2,3-dihydro-1-benzofuran-5-yl]-3,6-dihydro-2H-pyridin-1-yl]sulfonyl]-2-methylbutan-2-ol
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C30H40F2N4O4S
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1
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| 1 |
EC50 = 101 nM
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CP0401514
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propan-2-yl 4-[5-(1-propylsulfonyl-3,6-dihydro-2H-pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]piperidine-1-carboxylate
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C25H36N2O5S
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1
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| 1 |
EC50 = 103 nM
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CP0547021
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3-[[4-[7-fluoro-2-[1-(5-propylpyrimidin-2-yl)piperidin-4-yl]-2,3-dihydro-1-benzofuran-5-yl]-3,6-dihydro-2H-pyridin-1-yl]sulfonyl]propan-1-ol
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C28H37FN4O4S
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1
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| 1 |
EC50 = 122 nM
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CP0387127
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7-(5-ethylpyrimidin-2-yl)-2-[3-(3-fluoro-4-methylsulfonylphenoxy)propyl]-7-azaspiro[3.5]nonane
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C24H32FN3O3S
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1
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| 1 |
EC50 = 123 nM
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CP0518059
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tert-butyl 2-[4-(4-methylsulfonylphenoxy)butyl]-7-azaspiro[3.5]nonane-7-carboxylate
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C24H37NO5S
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1
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| 1 |
EC50 = 154 nM
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CP0443223
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propan-2-yl 4-[5-(4-methylsulfonylphenoxy)pyrazolo[3,4-c]pyridin-1-yl]piperidine-1-carboxylate
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C22H26N4O5S
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1
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| 1 |
EC50 = 177 nM
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CP0540591
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tert-butyl 2-[2-(4-methylsulfonylphenoxy)ethyl]-7-azaspiro[3.5]nonane-7-carboxylate
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C22H33NO5S
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1
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| 1 |
EC50 = 183 nM
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CP0420554
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propan-2-yl 4-[5-(6-methylsulfonylpyridin-3-yl)pyrazolo[3,4-c]pyridin-1-yl]piperidine-1-carboxylate
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C21H25N5O4S
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1
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| 1 |
EC50 = 197 nM
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CP0542451
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1-[1-(3-methylbutyl)piperidin-4-yl]-5-(4-methylsulfonylphenyl)pyrazolo[3,4-c]pyridine
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C23H30N4O2S
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1
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| 1 |
EC50 = 220 nM
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CP0540594
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7-(5-ethylpyrimidin-2-yl)-2-[3-(2-fluoro-4-methylsulfonylphenoxy)propyl]-7-azaspiro[3.5]nonane
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C24H32FN3O3S
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1
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| 1 |
EC50 = 225 nM
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CP0420555
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propan-2-yl 4-[5-(3-methylsulfonylphenoxy)pyrazolo[3,4-c]pyridin-1-yl]piperidine-1-carboxylate
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C22H26N4O5S
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1
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| 1 |
EC50 = 266 nM
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CP0469669
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7-(5-methylpyridin-2-yl)-2-[3-(4-methylsulfonylphenoxy)propyl]-7-azaspiro[3.5]nonane
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C24H32N2O3S
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1
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| 1 |
EC50 = 348 nM
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CP0435109
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5-propyl-2-[4-[5-(1-propylsulfonylpiperidin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]piperidin-1-yl]pyrimidine
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C28H40N4O3S
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1
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| 1 |
EC50 = 386 nM
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CP0550681
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4-[2-(1-benzylpiperidin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]-1-propylsulfonyl-3,6-dihydro-2H-pyridine
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C28H36N2O3S
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1
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| 1 |
EC50 = 521 nM
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CP0382256
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2-[4-[5-(2-fluoro-4-methylsulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]piperidin-1-yl]-5-propylpyrimidine
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C27H30FN3O3S
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1
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| 1 |
EC50 = 541 nM
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CP0440295
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5-propyl-2-[4-[5-(4-propylsulfonylpiperazin-1-yl)-2,3-dihydro-1-benzofuran-2-yl]piperidin-1-yl]pyrimidine
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C27H39N5O3S
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1
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| 1 |
EC50 = 544 nM
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CP0519925
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tert-butyl 2-[3-(4-methylsulfonylphenoxy)propyl]-6-azaspiro[2.5]octane-6-carboxylate
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C22H33NO5S
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1
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| 1 |
EC50 = 830 nM
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CP0511940
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1-propylsulfonyl-4-[2-(1-propylsulfonylpiperidin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]-3,6-dihydro-2H-pyridine
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C24H36N2O5S2
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1
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| 1 |
EC50 = 1003 nM
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CP0540592
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tert-butyl 2-[2-(4-methylsulfonylphenoxy)ethyl]-6-azaspiro[2.5]octane-6-carboxylate
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C21H31NO5S
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1
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| 1 |
EC50 = 2388 nM
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CP0519927
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tert-butyl 9-[3-(4-methylsulfonylphenoxy)propyl]-3-azaspiro[5.5]undecane-3-carboxylate
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C25H39NO5S
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1
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| 1 |
EC50 = 2590 nM
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CP0474893
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1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-4-methyl-5-(4-methylsulfonylphenyl)indazole
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C26H29N5O2S
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1
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| 1 |
EC50 = 3423 nM
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