Brief Information of the Compound and Protein
Compound Name
1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-6-methyl-5-(4-methylsulfonylphenyl)indazole
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PubChem ID
CID: 68021862
Canonical SMILES
CCc1cnc(nc1)N1CCC(CC1)n1ncc2cc(c(C)cc12)-c1ccc(cc1)S(C)(=O)=O
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Compound Formula C26H29N5O2S
Compound Structure
Protein Name
Glucose-dependent insulinotropic receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
Uniprot ID
Q8TDV5
Gene Name
GPR119
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000460 Flp-In-T-REx-293 Homo sapiens (Human)  1
1
EC50 = 70 nM
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