Brief Information of the Cell Line and Protein
Cell Line ID: CL000386 , Flp-In-CHO
Synonyms
Flp-In CHO
CHO Flp-In
CHO-Flp-In
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_U424
Protein ID: PT02590 , N-formyl peptide receptor 2
Gene Name FPR2
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P25090
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000386  Protein ID: PT02590
 
Compound ID Compound Name Compound Formula
CP0259831
1-(4-chlorophenyl)-3-[1-methyl-3-oxo-2-phenyl-5-(propan-2-yl)-2,3-dihydro-1H-pyrazol-4-yl]urea
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C20H21ClN4O2
 2
1
EC50 = 40.74 nM
   TI
   LI
   LO
   TS
2
EC50 = 95.5 nM
   TI
   LI
   LO
   TS
CP0391359
N-(4-chlorophenyl)-2-[5-[(2-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]hexanamide
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C25H28ClN3O3
 2
1
EC50 = 51.29 nM
   TI
   LI
   LO
   TS
2
EC50 = 70.79 nM
   TI
   LI
   LO
   TS
CP0423004
N-(4-chlorophenyl)-2-[5-[(2,3-dimethoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]hexanamide
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C26H30ClN3O4
 2
1
EC50 = 52.48 nM
   TI
   LI
   LO
   TS
2
EC50 = 61.66 nM
   TI
   LI
   LO
   TS
CP0476610
N-(4-chlorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]propanamide
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C22H22ClN3O3
 2
1
EC50 = 9549.93 nM
   TI
   LI
   LO
   TS
2
EC50 > 100000 nM
   TI
   LI
   LO
   TS