Brief Information of the Cell Line and Protein
Cell Line ID: CL000386 , Flp-In-CHO
Synonyms
Flp-In CHO
CHO Flp-In
CHO-Flp-In
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_U424
Protein ID: PT02415 , Sodium/glucose cotransporter 2
Gene Name SLC5A2
Organism Homo sapiens, Human
Protein Classification Transporter
Uniprot ID P31639
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000386  Protein ID: PT02415
 
Compound ID Compound Name Compound Formula
CP0538916
US8980829, 23
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C25H30ClFO7
 1
1
IC50 = 1.1 nM
   TI
   LI
   LO
   TS
CP0406152
US8980829, 22
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C25H31ClO7
 1
1
IC50 = 1.7 nM
   TI
   LI
   LO
   TS
CP0462833
US8980829, 8
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C24H29ClO7
 1
1
IC50 = 1.7 nM
   TI
   LI
   LO
   TS
CP0198642
(2S,3R,4R,5S,6R)-2-{4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl}-6-(hydroxymethyl)oxane-3,4,5-triol
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C21H25ClO6
 1
1
IC50 = 3 nM
   TI
   LI
   LO
   TS
CP0165584
BI-10773
   Show/Hide
C23H27ClO7
 1
1
IC50 = 3.1 nM
   TI
   LI
   LO
   TS
CP0468162
US8980829, 1
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C23H27ClO7
 1
1
IC50 = 5.6 nM
   TI
   LI
   LO
   TS
CP0388926
US8980829, 17
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C25H30ClNO7
 1
1
IC50 = 6.4 nM
   TI
   LI
   LO
   TS
CP0409846
US8980829, 12
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C23H26ClFO7
 1
1
IC50 = 6.5 nM
   TI
   LI
   LO
   TS
CP0472621
US8980829, 11
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C24H29ClO7S
 1
1
IC50 = 6.8 nM
   TI
   LI
   LO
   TS
CP0521104
US8980829, 10
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C24H29ClO6S
 1
1
IC50 = 7.4 nM
   TI
   LI
   LO
   TS
CP0406211
US8980829, 9
   Show/Hide
C24H28ClFO7
 1
1
IC50 = 7.5 nM
   TI
   LI
   LO
   TS
CP0538689
US8980829, 16
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C23H26ClFO6
 1
1
IC50 = 8.1 nM
   TI
   LI
   LO
   TS
CP0525161
US8980829, 5
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C24H29ClO7
 1
1
IC50 = 8.3 nM
   TI
   LI
   LO
   TS
CP0417364
US8980829, 14
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C23H28ClNO6
 1
1
IC50 = 8.4 nM
   TI
   LI
   LO
   TS
CP0385568
US8980829, 7
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C24H29ClO6
 1
1
IC50 = 8.5 nM
   TI
   LI
   LO
   TS
CP0407674
US8980829, 6
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C23H27ClO6
 1
1
IC50 = 9.6 nM
   TI
   LI
   LO
   TS
CP0516671
US8980829, 24
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C25H30ClFO8
 1
1
IC50 = 12 nM
   TI
   LI
   LO
   TS
CP0403413
US8980829, 25
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C27H34ClFO8
 1
1
IC50 = 12.3 nM
   TI
   LI
   LO
   TS
CP0472413
US8980829, 18
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C26H32ClNO7
 1
1
IC50 = 22 nM
   TI
   LI
   LO
   TS
CP0400915
US8980829, 15
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C24H30ClNO6
 1
1
IC50 = 23.6 nM
   TI
   LI
   LO
   TS
CP0409862
US8980829, 13
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C28H36ClNO8
 1
1
IC50 = 28.7 nM
   TI
   LI
   LO
   TS
CP0420229
US8980829, 26
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C25H32ClNO7
 1
1
IC50 = 69.4 nM
   TI
   LI
   LO
   TS
CP0472417
US8980829, 19
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C29H31ClFNO6
 1
1
IC50 = 97.2 nM
   TI
   LI
   LO
   TS