General Information of the Compound
Compound ID
CP0165584
Compound Name
BI-10773
    Show/Hide
Synonyms
(1S)-1,5-anhydro-1-(4-chloro-3-{4-[(3S)-tetrahydrofuran-3-yloxy]benzyl}phenyl)-D-glucitol
(2S,3R,4R,5S,6R)-2-(4-chloro-3-(4-(((S)-tetrahydrofuran-3-yl)oxy)benzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
1-chloro-4-(glucopyranos-1-yl)-2-(4-(tetrahydrofuran-3-yloxy)benzyl)benzene
864070-44-0
AK160980
BI 10773
BI-10773
BI10773
CHEBI:82720
Empagliflozin
Empagliflozin (BI 10773)
HDC1R2M35U
JARDIANCE
UNII-HDC1R2M35U
    Show/Hide
Structure
Formula
C23H27ClO7
Molecular Weight
450.915
Canonical SMILES
OC[C@H]1O[C@H]([C@H](O)[C@@H](O)[C@@H]1O)c1ccc(Cl)c(Cc2ccc(O[C@H]3CCOC3)cc2)c1
    Show/Hide
InChI
InChI=1S/C23H27ClO7/c24-18-6-3-14(23-22(28)21(27)20(26)19(11-25)31-23)10-15(18)9-13-1-4-16(5-2-13)30-17-7-8-29-12-17/h1-6,10,17,19-23,25-28H,7-9,11-12H2/t17-,19+,20+,21-,22+,23-/m0/s1
    Show/Hide
InChIKey
OBWASQILIWPZMG-QZMOQZSNSA-N
CAS
864070-44-0
Physicochemical Property
logP
1.6134
Rotatable Bonds
6
Heavy Atom Count
31
Polar Areas
108.61
Hydrogen Bond Donor Count
4
Hydrogen Bond Acceptor Count
7
Complexity
31

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 11949646
SID: 136350032
ChEMBL ID
CHEMBL2107830
DrugBank ID
DB09038
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT03804, Sodium/glucose cotransporter 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000386 Flp-In-CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 3235 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 8300 nM
Protein ID: PT02415, Sodium/glucose cotransporter 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000386 Flp-In-CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 3.1 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 3 nM
2 IC50 = 3.1 nM
Clinical Information about the Compound
Drug 1 ( Empagliflozin )
Drug Name Empagliflozin
Company Boehringer Ingelheim Pharmaceuticals; Eli Lilly
Indication
Type-1 diabetes
Approved
Target(s)
Sodium/glucose cotransporter 2 (SGLT2)
Modulator