Brief Information of the Cell Line and Protein
Cell Line ID: CL000386 , Flp-In-CHO
 Cell Line Info 
Synonyms
Flp-In CHO
CHO Flp-In
CHO-Flp-In
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_U424
Protein ID: PT01717 , Adenosine receptor A1
 Protein Info 
Gene Name ADORA1
Organism Rattus norvegicus, Rat
Protein Classification Membrane receptor
Uniprot ID P25099
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000386
 Cell Line Info 
 Protein ID: PT01717
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0543934
 Compound Info 
5-[5-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]pentanoylamino]-N-[3-[2-[[2-[4-(2,6-dioxo-1,3-dipropyl-7H-purin-8-yl)phenoxy]acetyl]amino]ethylamino]-3-oxopropyl]pentanamide
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C57H66BF2N11O9S
  1
1
Kd = 35.48 nM
 Bioactivity Info 
   TI
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CP0855184
 Compound Info 
3-(4-(2-(6-(4-(9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxytetrahydrofuran-2-yl)-9H-purin-6-ylamino)butylamino)-6-oxohexylamino)-2-oxoethoxy)styryl)-5,5-difluoro-7-(thiophen-2-yl)-5H-dipyrrolo[1,2-c:1',2'-f][1,3,2]diazaborinin-4-ium-5-uide
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C45H51BF2N10O7S
  1
1
Kd = 891.25 nM
 Bioactivity Info 
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CP0868745
 Compound Info 
3-(4-(2-(6-(4-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl)-9H-purin-6-ylamino)butylamino)-6-oxohexylamino)-2-oxoethoxy)styryl)-5,5-difluoro-7-(thiophen-2-yl)-5H-dipyrrolo[1,2-c:1',2'-f][1,3,2]diazaborinin-4-ium-5-uide
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C43H48BF2N9O7S
  1
1
Kd = 891.25 nM
 Bioactivity Info 
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CP0575002
 Compound Info 
(2S,3S,4R,5R)-5-[6-[4-[[2-[[(2R)-2-[[(2R)-2-[6-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]hexanoylamino]propanoyl]amino]propanoyl]amino]acetyl]amino]butylamino]purin-9-yl]-N-ethyl-3,4-dihydroxyoxolane-2-carboxamide
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C53H64BF2N13O10S
  1
1
Kd = 1778.28 nM
 Bioactivity Info 
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