Brief Information of the Cell Line and Protein
Cell Line ID: CL000330 , CHO Pro-4 MtxRII OuaR-2-4
Synonyms
Pro-4 MtxRII OuaR 2-4
MTXRIIOuaR2-4
R2
Category Transformed cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_C5SG
Protein ID: PT05723 , Reduced folate transporter
Gene Name SLC19A1
Organism Homo sapiens, Human
Protein Classification Transporter
Uniprot ID P41440
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000330  Protein ID: PT05723
 
Compound ID Compound Name Compound Formula
CP0035062
(S)-2-(4-(4-(2-amino-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-6-yl)butyl)benzamido)pentanedioic acid
   Show/Hide
C22H24N4O6S
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0882698
(5-(4-(2-amino-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-6-yl)butyl)thiophene-3-carbonyl)-L-glutamic acid
   Show/Hide
C20H22N4O6S2
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0915862
(5-(4-(2-amino-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-6-yl)butyl)thiophene-2-carbonyl)-L-glutamic acid
   Show/Hide
C20H22N4O6S2
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0915863
(5-(3-(2-amino-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-6-yl)propyl)thiophene-2-carbonyl)-L-glutamic acid
   Show/Hide
C19H20N4O6S2
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0915864
(4-(4-(2-amino-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-6-yl)butyl)thiophene-2-carbonyl)-L-glutamic acid
   Show/Hide
C20H22N4O6S2
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0915865
(5-(3-(2-amino-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-6-yl)propyl)thiophene-3-carbonyl)-L-glutamic acid
   Show/Hide
C19H20N4O6S2
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0915866
(5-(4-(2-amino-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-6-yl)butyl)furan-2-carbonyl)-L-glutamic acid
   Show/Hide
C20H22N4O7S
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0958003
(4-(3-(2-amino-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-6-yl)propyl)thiophene-2-carbonyl)-L-glutamic acid
   Show/Hide
C19H20N4O6S2
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS