| Compound ID |
Compound Name |
Compound Formula |
|
CP0913220
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-4-yl)-N-methyl-N-quinolin-8-yl-benzamide
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|
C25H21N3O3
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0505121
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-cyclohexanecarboxylic acid quinolin-8-ylamide
Show/Hide
|
C25H25N3O3
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
|
CP0919907
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-(7-methyl-quinolin-8-yl)-benzamide
Show/Hide
|
C26H21N3O3
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0469660
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-cyclohexanecarboxylic acid(7-methyl-quinolin-8-yl)-amide
Show/Hide
|
C26H27N3O3
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0497531
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-cyclohexanecarboxylic acid(4-methyl-quinolin-8-yl)-amide
Show/Hide
|
C26H27N3O3
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0860629
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-(2-methoxy-phenyl)-benzamide
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|
C23H20N2O4
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0870422
|
2-Chloro-4-((1R,2S,6R,7S)-3,5-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-quinolin-8-yl-benzamide
Show/Hide
|
C25H18ClN3O3
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0916216
|
N-(4-Bromo-phenyl)-4-((1R,2S,6R,7S)-3,5-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
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|
C22H17BrN2O3
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0870423
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-2-methyl-N-quinolin-8-yl-benzamide
Show/Hide
|
C26H21N3O3
|
1
|
| 1 |
EC50 = 2000 nM
|
|
|
|
CP0919908
|
trans-4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-(2-methoxy-cyclohexyl)-benzamide
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|
C23H26N2O4
|
1
|
| 1 |
EC50 = 2000 nM
|
|
|
|
CP0870419
|
N-(4-Chloro-phenyl)-4-((1R,2S,6R,7S)-3,5-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H17ClN2O3
|
1
|
| 1 |
EC50 = 3000 nM
|
|
|
|
CP0908469
|
N-(3,4-Difluoro-phenyl)-4-((1R,2S,6R,7S)-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H16F2N2O3
|
1
|
| 1 |
EC50 = 3000 nM
|
|
|
|
CP0908467
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-(4-fluoro-phenyl)-benzamide
Show/Hide
|
C22H17FN2O3
|
1
|
| 1 |
EC50 = 4000 nM
|
|
|
|
CP0669064
|
4-((1S,2S,6R,7R)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-quinolin-8-yl-benzamide
Show/Hide
|
C25H19N3O3
|
1
|
| 1 |
EC50 = 5000 nM
|
|
|
|
CP0915775
|
N-(3,4-Dichloro-phenyl)-4-((1R,2S,6R,7S)-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H16Cl2N2O3
|
1
|
| 1 |
EC50 = 5000 nM
|
|
|
|
CP0870420
|
N-(2,4-Difluoro-phenyl)-4-((1R,2S,6R,7S)-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H16F2N2O3
|
1
|
| 1 |
EC50 = 9000 nM
|
|
|
|
CP0902092
|
N-(3-Bromo-phenyl)-4-((1R,2S,6R,7S)-3,5-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H17BrN2O3
|
1
|
| 1 |
EC50 = 9000 nM
|
|
|
|
CP0439533
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-piperidine-1-carboxylic acid quinolin-8-ylamide
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|
C24H24N4O3
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
|
CP0501391
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-ylmethyl)-cyclohexanecarboxylic acid(7-methyl-quinolin-8-yl)-amide
Show/Hide
|
C27H29N3O3
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
|
CP0858259
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-(5,6,7,8-tetrahydro-quinolin-8-yl)-benzamide
Show/Hide
|
C25H23N3O3
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
|
CP0858261
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-pyridin-4-ylmethyl-benzamide
Show/Hide
|
C22H19N3O3
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
|
CP0879924
|
N-(3,4-Dibromo-phenyl)-4-((1R,2S,6R,7S)-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H16Br2N2O3
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
|
CP0916541
|
N-(2,4-Dichloro-phenyl)-4-((1R,2S,6R,7S)-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H16Cl2N2O3
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
|
CP0857598
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-(3-trifluoromethyl-phenyl)-benzamide
Show/Hide
|
C23H17F3N2O3
|
1
|
| 1 |
EC50 = 20000 nM
|
|
|
|
CP0891007
|
N-Benzyl-4-((1R,2S,6R,7S)-3,5-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C23H20N2O3
|
1
|
| 1 |
EC50 = 20000 nM
|
|
|
|
CP0481673
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-ylmethyl)-cyclohexanecarboxylic acid(4-methyl-quinolin-8-yl)-amide
Show/Hide
|
C27H29N3O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0505122
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-ylmethyl)-cyclohexanecarboxylic acid quinolin-8-ylamide
Show/Hide
|
C26H27N3O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0858260
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-(2-trifluoromethyl-phenyl)-benzamide
Show/Hide
|
C23H17F3N2O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0860630
|
N-(2-Chloro-phenyl)-4-((1R,2S,6R,7S)-3,5-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H17ClN2O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0860631
|
N-(2,5-Difluoro-phenyl)-4-((1R,2S,6R,7S)-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H16F2N2O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0860632
|
1-[4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-phenyl]-3-quinolin-8-yl-urea
Show/Hide
|
C25H20N4O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0870421
|
N-Cyclohexyl-4-((1R,2S,6R,7S)-3,5-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H24N2O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0879921
|
4-((1R,2S,6R,7R)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-phenyl-benzamide
Show/Hide
|
C22H18N2O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0879923
|
N-(2,6-Difluoro-phenyl)-4-((1R,2S,6R,7S)-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H16F2N2O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0879925
|
3-Chloro-4-((1R,2S,6R,7S)-3,5-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-quinolin-8-yl-benzamide
Show/Hide
|
C25H18ClN3O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0879926
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-2-methoxy-N-quinolin-8-yl-benzamide
Show/Hide
|
C26H21N3O4
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0891005
|
N-(3-Chloro-phenyl)-4-((1R,2S,6R,7S)-3,5-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H17ClN2O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0891006
|
N-(3,5-Difluoro-phenyl)-4-((1R,2S,6R,7S)-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H16F2N2O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0902062
|
N-(2-Bromo-phenyl)-4-((1R,2S,6R,7S)-3,5-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H17BrN2O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0902063
|
trans-4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-((2-hydroxy-cyclohexyl)-benzamide
Show/Hide
|
C22H24N2O4
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0908465
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-(2-fluoro-phenyl)-benzamide
Show/Hide
|
C22H17FN2O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0908470
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-methyl-N-quinolin-8-yl-benzamide
Show/Hide
|
C26H21N3O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0908499
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-(3-fluoro-phenyl)-benzamide
Show/Hide
|
C22H17FN2O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0916217
|
N-(2,4-Dibromo-phenyl)-4-((1R,2S,6R,7S)-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H16Br2N2O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0916218
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-pyridin-2-ylmethyl-benzamide
Show/Hide
|
C22H19N3O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0916540
|
N-(2,3-Difluoro-phenyl)-4-((1R,2S,6R,7S)-dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-benzamide
Show/Hide
|
C22H16F2N2O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0916542
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-(4-trifluoromethyl-phenyl)-benzamide
Show/Hide
|
C23H17F3N2O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0916543
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-N-pyridin-3-ylmethyl-benzamide
Show/Hide
|
C22H19N3O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0919909
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-3-methoxy-N-quinolin-8-yl-benzamide
Show/Hide
|
C26H21N3O4
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0935534
|
4-((1R,2S,6R,7S)-3,5-Dioxo-4-aza-tricyclo[5.2.1.0*2,6*]dec-8-en-4-yl)-3-methyl-N-quinolin-8-yl-benzamide
Show/Hide
|
C26H21N3O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
