Compound ID |
Compound Name |
Compound Formula |
CP0086566
|
(2S)-2-[[2-(azepan-1-yl)acetyl]amino]-4-methyl-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxo-3-phenylpropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pentanamide
Show/Hide
|
C35H48N4O5
|
1
|
1 |
IC50 = 159 nM
|
|
|
CP0098995
|
(2S)-2-[[2-(azepan-1-yl)acetyl]amino]-4-methyl-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-4-(4-methylphenyl)-1-oxobutan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pentanamide
Show/Hide
|
C37H52N4O5
|
1
|
1 |
IC50 = 305 nM
|
|
|
CP0213895
|
Kzr-616
Show/Hide
|
C30H42N4O8
|
1
|
1 |
IC50 = 522 nM
|
|
|
CP0062987
|
(2S)-3-(4-methoxyphenyl)-N-[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxo-3-phenylpropan-2-yl]-2-[[(2S)-2-[(2-morpholin-4-ylacetyl)amino]propanoyl]amino]propanamide
Show/Hide
|
C31H40N4O7
|
1
|
1 |
IC50 = 699 nM
|
|
|