Compound ID |
Compound Name |
Compound Formula |
CP0328884
|
(2R)-N'-(5-fluoro-2-methylpyridin-3-yl)-2-methyl-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide
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|
C23H26FN5O3
|
1
|
1 |
IC50 = 97 nM
|
|
|
CP0408802
|
(2R)-N'-(5-fluoro-2-methylpyridin-3-yl)-N-[(6S)-10-fluoro-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]-2-methylbutanediamide
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|
C23H25F2N5O3
|
1
|
1 |
IC50 = 121 nM
|
|
|
CP0460550
|
(2S)-2-cyclopropyl-N-[(6S)-5,11-dioxospiro[3,6-dihydro-1H-pyrazolo[1,2-b][2,3]benzodiazepine-2,1'-cyclopropane]-6-yl]-N'-(5-fluoro-2-methylpyridin-3-yl)butanediamide
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|
C27H28FN5O4
|
1
|
1 |
IC50 = 137 nM
|
|
|
CP0013376
|
N-[(2S,3S)-3-amino-2-hydroxy-3-[4-(trifluoromethoxy)phenyl]propyl]-4-tert-butyl-N-cyclobutylbenzenesulfonamide
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|
C24H31F3N2O4S
|
1
|
1 |
IC50 = 150 nM
|
|
|
CP0430084
|
(2R)-2-methyl-N'-(2-methylphenyl)-N-[(6S)-5-oxo-2,3,6,11-tetrahydro-1H-pyrazolo[1,2-b][2,3]benzodiazepin-6-yl]butanediamide
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|
C24H28N4O3
|
1
|
1 |
IC50 = 370 nM
|
|
|
CP0481546
|
(2S)-2-cyclopropyl-N-[(6S)-5,11-dioxo-1,2,3,6-tetrahydropyrazolo[1,2-b][2,3]benzodiazepin-6-yl]-N'-(5-fluoro-2-methylpyridin-3-yl)butanediamide
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|
C25H26FN5O4
|
1
|
1 |
IC50 = 496 nM
|
|
|