| Compound ID |
Compound Name |
Compound Formula |
|
CP0874591
|
2-(2-{bis[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C30H29FN8OS
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0887768
|
2-(2-{bis[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide tetrahydrochloride
Show/Hide
|
C30H33Cl4FN8O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0874581
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-chloropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C21H21ClN6O2
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0947240
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-chloropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H19ClN6OS
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0942114
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-5-chloro-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C21H23Cl4FN6OS
|
1
|
| 1 |
IC50 = 8.3 nM
|
|
|
|
CP0903120
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide trihydrochloride
Show/Hide
|
C21H24Cl3FN6O2
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0874586
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-(pyridin-2-ylmethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H22N6OS
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0880270
|
1-(2-((2-(1H-benzo[d]imidazol-2-yl)ethyl)amino)ethyl)-N-((3-fluoropyridin-2-yl)methyl)-1H-1,2,3-triazole-4-carboxamide
Show/Hide
|
C20H21FN8O
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0874584
|
1-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-chloropyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
Show/Hide
|
C21H22ClN7O
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0901637
|
2-{1-[2-(1H-1,3-benzodiazol-2-yl)ethyl]azetidin-3-yl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C22H21FN6O2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0901639
|
2-(2-{[2-(1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H21FN6OS
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0903140
|
2-(2-{[2-(1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-5-carboxamide
Show/Hide
|
C21H21FN6O2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0880267
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-methylpyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C21H25Cl3N6OS
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0946477
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-methylpyridin-4-yl)methyl]-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C21H25Cl3N6OS
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0903146
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide trihydrochloride
Show/Hide
|
C21H25Cl3N6O2
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0904080
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-(pyridazin-3-ylmethyl)-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C20H24Cl3N7OS
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0948408
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-(1,3-oxazol-2-ylmethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C18H18N6O2S
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0854890
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-(5,6,7,8-tetrahydroquinolin-8-yl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C23H24N6OS
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0903122
|
2-(2-{[2-(4-Fluoro-1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H20F2N6OS
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0904081
|
2-(2-{[2-(5-Fluoro-1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C21H23Cl3F2N6OS
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0874587
|
2-(2-{[2-(4,5-Difluoro-1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C21H19F3N6O2
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0887766
|
2-{1-[2-(1H-1,3-Benzodiazol-2-yl)ethyl]azetidin-3-yl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-5-carboxamide
Show/Hide
|
C22H21FN6O2
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0903130
|
1-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide tetrahydrochloride
Show/Hide
|
C21H26Cl4FN7O
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0903142
|
2-{1-[2-(4-Fluoro-1H-1,3-benzodiazol-2-yl)ethyl]azetidin-3-yl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C22H20F2N6O2
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0880284
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoro-6-methylpyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H21FN6OS
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0903753
|
2-(2-{[2-(4,6-Difluoro-1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C21H19F3N6O2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0874588
|
2-(2-{[2-(4-Fluoro-1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C21H20F2N6O2
|
1
|
| 1 |
IC50 = 46 nM
|
|
|
|
CP0958111
|
2-(2-(2-(1H-benzo[d]imidazol-2-yl)ethylamino)ethyl)-N-(6,7-dihydro-5H-cyclopenta[b]pyridin-7-yl)thiazole-4-carboxamide
Show/Hide
|
C23H24N6OS
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0874577
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C20H22Cl3FN6OS
|
1
|
| 1 |
IC50 = 49 nM
|
|
|
|
CP0903127
|
2-(2-{[2-(4-Chloro-1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C21H20ClFN6O2
|
1
|
| 1 |
IC50 = 49 nM
|
|
|
|
CP0954546
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-methoxypyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H22N6O2S
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0955513
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-chloro-5-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H18ClFN6OS
|
1
|
| 1 |
IC50 = 58 nM
|
|
|
|
CP0909892
|
5-chloro-N-(pyridin-2-ylmethyl)-2-(2-{1,8,12-triazatricyclo[7.4.0.02,7]trideca-2(7),3,5,8-tetraen-12-yl}ethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H21ClN6OS
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0957856
|
2-(2-{[2-(4,7-Difluoro-1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C21H19F3N6O2
|
1
|
| 1 |
IC50 = 62 nM
|
|
|
|
CP0871743
|
2-{1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]azetidin-3-yl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-5-carboxamide
Show/Hide
|
C22H20F2N6O2
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0947239
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-5-chloro-N-(pyridin-2-ylmethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H21ClN6OS
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0874579
|
2-(2-{[2-(5-cyano-1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C22H20FN7O2
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0903748
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-{5H,6H,7H-cyclopenta[b]pyridin-7-yl}-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C22H25Cl3N6OS
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0880280
|
1-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
Show/Hide
|
C21H23N7O
|
1
|
| 1 |
IC50 = 76 nM
|
|
|
|
CP0944109
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(4,6-dimethylpyridin-3-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H24N6OS
|
1
|
| 1 |
IC50 = 77 nM
|
|
|
|
CP0903750
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-(pyridin-2-ylmethyl)-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C20H23Cl3N6OS
|
1
|
| 1 |
IC50 = 80 nM
|
|
|
|
CP0903121
|
N-[(3-fluoropyridin-2-yl)methyl]-2-[2-({2-[4-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]ethyl}amino)ethyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C22H20F4N6O2
|
1
|
| 1 |
IC50 = 81 nM
|
|
|
|
CP0951408
|
2-(2-{[2-(7-Chloro-4-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C21H19ClF2N6O2
|
1
|
| 1 |
IC50 = 82 nM
|
|
|
|
CP0941165
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-4-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H19FN6OS
|
1
|
| 1 |
IC50 = 89 nM
|
|
|
|
CP0887764
|
1-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-{5H,6H,7H-cyclopenta[b]pyridin-7-yl}-1H-pyrazole-4-carboxamide trihydrochloride
Show/Hide
|
C23H28Cl3N7O
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0944213
|
2-{1-[2-(1H-1,3-benzodiazol-2-yl)ethyl]azetidin-3-yl}-N-(pyridazin-3-ylmethyl)-1,3-oxazole-4-carboxamide
Show/Hide
|
C21H21N7O2
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0905660
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-5-chloro-N-[(3-chloropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H18Cl2N6OS
|
1
|
| 1 |
IC50 = 91 nM
|
|
|
|
CP0941166
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(2-oxo-1,2-dihydropyridin-3-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H20N6O2S
|
1
|
| 1 |
IC50 = 96 nM
|
|
|
|
CP0946518
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide trihydrochloride
Show/Hide
|
C20H22Cl3FN6O2
|
1
|
| 1 |
IC50 = 96 nM
|
|
|
|
CP0850093
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3,5-dimethylpyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H24N6OS
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0944108
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-5-methyl-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H23FN6OS
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0874594
|
2-({[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}methyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C20H22Cl3FN6OS
|
1
|
| 1 |
IC50 = 103 nM
|
|
|
|
CP0942115
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-5-chloro-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H18ClFN6OS
|
1
|
| 1 |
IC50 = 111 nM
|
|
|
|
CP0905657
|
2-(2-{[(6-Fluoro-1H-1,3-benzodiazol-2-yl)methyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C20H21Cl3F2N6OS
|
1
|
| 1 |
IC50 = 118 nM
|
|
|
|
CP0951409
|
N-[(3-fluoropyridin-2-yl)methyl]-2-(2-{[2-(4-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-1,3-oxazole-4-carboxamide
Show/Hide
|
C22H23FN6O3
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0951422
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C19H21N7OS
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0957785
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3,5-difluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H18F2N6OS
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0903128
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-5-chloro-N-(pyridazin-3-ylmethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H20ClN7OS
|
1
|
| 1 |
IC50 = 131 nM
|
|
|
|
CP0903755
|
1-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1H-1,2,4-triazole-3-carboxamide
Show/Hide
|
C20H21FN8O
|
1
|
| 1 |
IC50 = 135 nM
|
|
|
|
CP0880273
|
2-(2-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C21H20F2N6O2
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0909890
|
2-(2-(2-(1H-benzo[d]imidazol-2-yl)ethylamino)ethyl)-N-((3-fluoropyridin-2-yl)methyl)-5-methyloxazole-4-carboxamide
Show/Hide
|
C22H23FN6O2
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0909886
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(6-methylpyridazin-3-yl)methyl]-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C21H26Cl3N7OS
|
1
|
| 1 |
IC50 = 141 nM
|
|
|
|
CP0874590
|
1-{1-[2-(1H-1,3-Benzodiazol-2-yl)ethyl]azetidin-3-yl}-N-[(3-fluoropyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
Show/Hide
|
C22H22FN7O
|
1
|
| 1 |
IC50 = 145 nM
|
|
|
|
CP0957855
|
2-(2-{[(4-fluoro-1H-1,3-benzodiazol-2-yl)methyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H18F2N6OS
|
1
|
| 1 |
IC50 = 145 nM
|
|
|
|
CP0874580
|
2-(2-{[2-(4-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
Show/Hide
|
C21H21FN6O2
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0880272
|
2-{1-[2-(4-Fluoro-1H-1,3-benzodiazol-2-yl)ethyl]azetidin-3-yl}-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
Show/Hide
|
C22H21FN6O2
|
1
|
| 1 |
IC50 = 152 nM
|
|
|
|
CP0900251
|
2-{2-[(1H-1,3-benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-5-carboxamide
Show/Hide
|
C20H19FN6O2
|
1
|
| 1 |
IC50 = 155 nM
|
|
|
|
CP0960692
|
2-({[3-(1H-1,3-Benzodiazol-2-yl)propyl]amino}methyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C21H24Cl3FN6OS
|
1
|
| 1 |
IC50 = 164 nM
|
|
|
|
CP0951377
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-chloropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C20H19ClN6O2
|
1
|
| 1 |
IC50 = 167 nM
|
|
|
|
CP0900252
|
2-{1-[2-(4-Fluoro-1H-1,3-benzodiazol-2-yl)ethyl]azetidin-3-yl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-5-carboxamide
Show/Hide
|
C22H20F2N6O2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0909889
|
N-[(3,5-Difluoropyridin-2-yl)methyl]-2-(2-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C21H22Cl3F3N6OS
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0951417
|
1-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-chloropyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
Show/Hide
|
C20H20ClN7O
|
1
|
| 1 |
IC50 = 179 nM
|
|
|
|
CP0874589
|
2-({[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}methyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C20H19FN6O2
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0905659
|
2-{1-[2-(1H-1,3-benzodiazol-2-yl)ethyl]azetidin-3-yl}-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
Show/Hide
|
C22H22N6O2
|
1
|
| 1 |
IC50 = 183 nM
|
|
|
|
CP0903683
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-(pyridin-3-ylmethyl)-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C20H23Cl3N6OS
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0944236
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-(pyridazin-3-ylmethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C19H19N7OS
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0946468
|
2-{1-[2-(1H-1,3-Benzodiazol-2-yl)ethyl]azetidin-3-yl}-N-[(3-chloropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H21ClN6OS
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0959707
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-{[2-(difluoromethoxy)phenyl]methyl}-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H21F2N5O2S
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0903124
|
Benzyl N-(3-{[2-(1H-1,3-benzodiazol-2-yl)ethyl][2-(4-{[(3-fluoropyridin-2-yl)methyl]carbamoyl}-1,3-thiazol-2-yl)ethyl]amino}propyl)carbamate
Show/Hide
|
C32H34FN7O3S
|
1
|
| 1 |
IC50 = 216 nM
|
|
|
|
CP0901638
|
2-(2-{[(4-fluoro-1H-1,3-benzodiazol-2-yl)methyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C20H18F2N6O2
|
1
|
| 1 |
IC50 = 226 nM
|
|
|
|
CP0880271
|
N-[(3-Fluoropyridin-2-yl)methyl]-2-(1-{2-[7-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]ethyl}azetidin-3-yl)-1,3-oxazole-4-carboxamide
Show/Hide
|
C23H20F4N6O2
|
1
|
| 1 |
IC50 = 228 nM
|
|
|
|
CP0903762
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-5-carboxamide
Show/Hide
|
C21H21FN6OS
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0941149
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(2-cyanophenyl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H20N6OS
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0941150
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-(pyridin-4-ylmethyl)-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C20H23Cl3N6OS
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0959235
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(5-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H19FN6OS
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0903109
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-5-chloro-N-(pyridin-2-ylmethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H19ClN6OS
|
1
|
| 1 |
IC50 = 256 nM
|
|
|
|
CP0959710
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(2,6-difluorophenyl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H19F2N5OS
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0941164
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(5-methylpyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H22N6OS
|
1
|
| 1 |
IC50 = 270 nM
|
|
|
|
CP0903132
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-{[3-chloro-5-(trifluoromethyl)pyridin-2-yl]methyl}-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H18ClF3N6OS
|
1
|
| 1 |
IC50 = 280 nM
|
|
|
|
CP0880276
|
2-{1-[2-(1H-1,3-Benzodiazol-2-yl)ethyl]azetidin-3-yl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H21FN6OS
|
1
|
| 1 |
IC50 = 287 nM
|
|
|
|
CP0905658
|
3-({[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}methyl)-N-[(3-fluoropyridin-2-yl)methyl]-1-methyl-1H-pyrazole-5-carboxamide
Show/Hide
|
C21H22FN7O
|
1
|
| 1 |
IC50 = 290 nM
|
|
|
|
CP0874583
|
1-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide
Show/Hide
|
C22H21F4N7O
|
1
|
| 1 |
IC50 = 297 nM
|
|
|
|
CP0942112
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-5-(trifluoromethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H20F4N6OS
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0903144
|
1-{1-[2-(1H-1,3-Benzodiazol-2-yl)ethyl]azetidin-3-yl}-N-{5H,6H,7H-cyclopenta[b]pyridin-7-yl}-1H-pyrazole-4-carboxamide
Show/Hide
|
C24H25N7O
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0903125
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-5-methyl-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H21FN6OS
|
1
|
| 1 |
IC50 = 343 nM
|
|
|
|
CP0960696
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[1-(pyridin-2-yl)ethyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H22N6OS
|
1
|
| 1 |
IC50 = 345 nM
|
|
|
|
CP0909893
|
2-(2-{[2-(1H-1,3-benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(5-methylpyrimidin-2-yl)methyl]-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C21H26Cl3N7OS
|
1
|
| 1 |
IC50 = 347 nM
|
|
|
|
CP0880286
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-(3-fluoropyridin-2-yl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C19H17FN6OS
|
1
|
| 1 |
IC50 = 350 nM
|
|
|
|
CP0874593
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-(pyrimidin-2-ylmethyl)-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C20H24Cl3N7OS
|
1
|
| 1 |
IC50 = 353 nM
|
|
|
|
CP0850092
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[2-(pyridin-2-yl)ethyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H22N6OS
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0960686
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-5-chloro-N-(pyridazin-3-ylmethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C19H18ClN7OS
|
1
|
| 1 |
IC50 = 361 nM
|
|
|
|
CP0887767
|
4-({[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}methyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-2-carboxamide
Show/Hide
|
C20H19FN6OS
|
1
|
| 1 |
IC50 = 370 nM
|
|
|
|
CP0874592
|
2-{3-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]propyl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C21H24Cl3FN6OS
|
1
|
| 1 |
IC50 = 377 nM
|
|
|
|
CP0903110
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl](methyl)amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C22H26Cl3FN6OS
|
1
|
| 1 |
IC50 = 378 nM
|
|
|
|
CP0944105
|
2-{1-[2-(1H-1,3-benzodiazol-2-yl)ethyl]azetidin-3-yl}-5-chloro-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H20ClFN6OS
|
1
|
| 1 |
IC50 = 379 nM
|
|
|
|
CP0909887
|
1-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
Show/Hide
|
C20H20FN7O
|
1
|
| 1 |
IC50 = 385 nM
|
|
|
|
CP0887769
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(1-methyl-1H-imidazol-5-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C19H21N7OS
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0903751
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-4-methyl-1,3-thiazole-5-carboxamide
Show/Hide
|
C22H23FN6OS
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0877275
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(6-cyanopyridin-3-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H19N7OS
|
1
|
| 1 |
IC50 = 410 nM
|
|
|
|
CP0957786
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H19F3N6OS
|
1
|
| 1 |
IC50 = 420 nM
|
|
|
|
CP0944217
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(5-methoxypyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H22N6O2S
|
1
|
| 1 |
IC50 = 440 nM
|
|
|
|
CP0880269
|
5-{[(2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-1,3-thiazol-4-yl)formamido]methyl}pyridine-2-carboxamide
Show/Hide
|
C21H21N7O2S
|
1
|
| 1 |
IC50 = 460 nM
|
|
|
|
CP0903147
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H23N7OS
|
1
|
| 1 |
IC50 = 460 nM
|
|
|
|
CP0907044
|
2-{2-[(1H-1,3-Benzodiazol-2-yl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide dihydrochloride
Show/Hide
|
C19H19Cl2FN6OS
|
1
|
| 1 |
IC50 = 473 nM
|
|
|
|
CP0871793
|
5-(2-((2-(1H-benzo[d]imidazol-2-yl)ethyl)amino)ethyl)-N-(pyridin-2-ylmethyl)-1,2,4-oxadiazole-3-carboxamide
Show/Hide
|
C20H21N7O2
|
1
|
| 1 |
IC50 = 476 nM
|
|
|
|
CP0874595
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(1-methyl-1H-pyrazol-3-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C19H21N7OS
|
1
|
| 1 |
IC50 = 480 nM
|
|
|
|
CP0957783
|
1-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-chloropyridin-2-yl)methyl]-1H-1,2,4-triazole-3-carboxamide
Show/Hide
|
C19H19ClN8O
|
1
|
| 1 |
IC50 = 482 nM
|
|
|
|
CP0887763
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-(pyridine-2-ylmethyl)-1,3-oxazole-4-carboxamid
Show/Hide
|
C20H20N6O2
|
1
|
| 1 |
IC50 = 514 nM
|
|
|
|
CP0871769
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-{[2-(morpholine-4-sulfonyl)phenyl]methyl}-1,3-thiazole-4-carboxamide
Show/Hide
|
C25H28N6O4S2
|
1
|
| 1 |
IC50 = 530 nM
|
|
|
|
CP0903133
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(6-methylpyridazin-3-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H21N7OS
|
1
|
| 1 |
IC50 = 530 nM
|
|
|
|
CP0903760
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-{[2-(dimethylamino)phenyl]methyl}-1,3-thiazole-4-carboxamide
Show/Hide
|
C23H26N6OS
|
1
|
| 1 |
IC50 = 530 nM
|
|
|
|
CP0947256
|
2-{1-[2-(4-Fluoro-1H-1,3-benzodiazol-2-yl)ethyl]azetidin-3-yl}-N-(pyridazin-3-ylmethyl)-1,3-oxazole-4-carboxamide
Show/Hide
|
C21H20FN7O2
|
1
|
| 1 |
IC50 = 554 nM
|
|
|
|
CP0904108
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-(pyrimidin-2-ylmethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C19H19N7OS
|
1
|
| 1 |
IC50 = 560 nM
|
|
|
|
CP0944214
|
1-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-{5H,6H,7H-cyclopenta[b]pyridin-7-yl}-1H-pyrazole-4-carboxamide
Show/Hide
|
C22H23N7O
|
1
|
| 1 |
IC50 = 580 nM
|
|
|
|
CP0874576
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-(pyrazin-2-ylmethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C19H19N7OS
|
1
|
| 1 |
IC50 = 590 nM
|
|
|
|
CP0903141
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(6-methylpyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H22N6OS
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0961170
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-{[2-(morpholin-4-yl)phenyl]methyl}-1,3-thiazole-4-carboxamide
Show/Hide
|
C25H28N6O2S
|
1
|
| 1 |
IC50 = 610 nM
|
|
|
|
CP0938647
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl](butyl)amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C25H29FN6OS
|
1
|
| 1 |
IC50 = 717 nM
|
|
|
|
CP0909891
|
2-{1-[2-(1H-1,3-Benzodiazol-2-yl)ethyl]azetidin-3-yl}-N-{5H,6H,7H-cyclopenta[b]pyridin-7-yl}-1,3-thiazole-4-carboxamide
Show/Hide
|
C24H24N6OS
|
1
|
| 1 |
IC50 = 720 nM
|
|
|
|
CP0959712
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(6-oxo-1,6-dihydropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H20N6O2S
|
1
|
| 1 |
IC50 = 720 nM
|
|
|
|
CP0909885
|
2-{1-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-3-hydroxyazetidin-3-yl}-5-chloro-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H20ClFN6O2S
|
1
|
| 1 |
IC50 = 747 nM
|
|
|
|
CP0903129
|
1-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-1H-1,2,4-triazole-3-carboxamide
Show/Hide
|
C19H19FN8O
|
1
|
| 1 |
IC50 = 750 nM
|
|
|
|
CP0880283
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(1-methyl-1H-pyrazol-5-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C19H21N7OS
|
1
|
| 1 |
IC50 = 780 nM
|
|
|
|
CP0903123
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)-2-methylpropyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C23H25FN6OS
|
1
|
| 1 |
IC50 = 780 nM
|
|
|
|
CP0854891
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-{[3-(trifluoromethyl)pyridin-2-yl]methyl}-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H19F3N6OS
|
1
|
| 1 |
IC50 = 810 nM
|
|
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CP0954513
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2-{2-[(3-Aminopropyl)[2-(1H-1,3-benzodiazol-2-yl)ethyl]amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
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C24H28FN7OS
|
1
|
| 1 |
IC50 = 828 nM
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CP0903134
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1-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
Show/Hide
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C20H21N7O
|
1
|
| 1 |
IC50 = 830 nM
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CP0903681
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2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(2-fluorophenyl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
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C21H20FN5OS
|
1
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| 1 |
IC50 = 850 nM
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CP0947257
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2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(2-methoxypyridin-4-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
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C21H22N6O2S
|
1
|
| 1 |
IC50 = 900 nM
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CP0969572
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2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-(thiophen-2-ylmethyl)-1,3-thiazole-4-carboxamide
Show/Hide
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C19H19N5OS2
|
1
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| 1 |
IC50 = 900 nM
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CP0903145
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2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-5-(trifluoromethyl)-1,3-thiazole-4-carboxamide
Show/Hide
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C21H18F4N6OS
|
1
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| 1 |
IC50 = 957 nM
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CP0942113
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2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-5-chloro-N-[(5-methylpyrimidin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
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C21H22ClN7OS
|
1
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| 1 |
IC50 = 989 nM
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CP0905656
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2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3,5-difluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
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C21H23Cl3F2N6OS
|
1
|
| 1 |
IC50 = 1000 nM
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CP0903756
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2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-5-chloro-N-(pyrimidin-2-ylmethyl)-1,3-thiazole-4-carboxamide
Show/Hide
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C19H18ClN7OS
|
1
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| 1 |
IC50 = 1025 nM
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CP0874582
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2-{2-[bis(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
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C28H25FN8OS
|
1
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| 1 |
IC50 = 1118 nM
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CP0903108
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4-(2-{[2-(1H-1,3-Benzodiazol-2-yl)-2,2-difluoroethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-2-carboxamide
Show/Hide
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C21H19F3N6OS
|
1
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| 1 |
IC50 = 1130 nM
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CP0880277
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2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-5-methyl-N-(pyrimidin-2-ylmethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H23N7OS
|
1
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| 1 |
IC50 = 1160 nM
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CP0874540
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2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-(pyrimidin-4-ylmethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C19H19N7OS
|
1
|
| 1 |
IC50 = 1330 nM
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|
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CP0959708
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-{[2-(trifluoromethoxy)phenyl]methyl}-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H20F3N5O2S
|
1
|
| 1 |
IC50 = 1360 nM
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|
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CP0941163
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(4-methylpyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H22N6OS
|
1
|
| 1 |
IC50 = 1520 nM
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CP0951544
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2-(2-{[3-(1H-1,3-Benzodiazol-2-yl)propyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C22H26Cl3FN6OS
|
1
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| 1 |
IC50 = 1660 nM
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|
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CP0951545
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2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-{[3-(hydroxymethyl)pyridin-2-yl]methyl}-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H22N6O2S
|
1
|
| 1 |
IC50 = 1699 nM
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CP0880282
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-{[6-(dimethylamino)pyridin-3-yl]methyl}-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H25N7OS
|
1
|
| 1 |
IC50 = 1850 nM
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|
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CP0904079
|
2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl](methyl)amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C22H23FN6O2
|
1
|
| 1 |
IC50 = 1900 nM
|
|
|
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CP0854892
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5-(2-((2-(1H-benzo[d]imidazol-2-yl)ethyl)amino)ethyl)-N-((3-fluoropyridin-2-yl)methyl)-1,2,4-oxadiazole-3-carboxamide
Show/Hide
|
C20H20FN7O2
|
1
|
| 1 |
IC50 = 2009 nM
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|
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CP0948455
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C19H21N7OS
|
1
|
| 1 |
IC50 = 2070 nM
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|
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CP0960687
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2-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl](cyclopropylmethyl)amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C25H27FN6OS
|
1
|
| 1 |
IC50 = 2085 nM
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|
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CP0955512
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(2-fluoropyridin-3-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H19FN6OS
|
1
|
| 1 |
IC50 = 2370 nM
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|
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CP0944216
|
N-(1H-1,3-Benzodiazol-2-ylmethyl)-2-{2-[(1H-1,3-benzodiazol-2-ylmethyl)amino]ethyl}-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H21N7OS
|
1
|
| 1 |
IC50 = 2390 nM
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|
|
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CP0960688
|
1-(2-{[2-(1H-1,3-Benzodiazol-2-yl)ethyl]amino}ethyl)-N-[(3-fluoropyridin-2-yl)methyl]-5-methyl-1H-imidazole-4-carboxamide
Show/Hide
|
C22H24FN7O
|
1
|
| 1 |
IC50 = 2430 nM
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|
|
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CP0880279
|
1-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide
Show/Hide
|
C21H19F4N7O
|
1
|
| 1 |
IC50 = 2462 nM
|
|
|
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CP0953916
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-{[2-(4-methylpiperazin-1-yl)phenyl]methyl}-1,3-thiazole-4-carboxamide
Show/Hide
|
C26H31N7OS
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
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CP0947244
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-{[2-(morpholin-4-yl)pyridin-4-yl]methyl}-1,3-thiazole-4-carboxamide
Show/Hide
|
C24H27N7O2S
|
1
|
| 1 |
IC50 = 2970 nM
|
|
|
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CP0880281
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(2-methylpyridin-4-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H22N6OS
|
1
|
| 1 |
IC50 = 2990 nM
|
|
|
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CP0941162
|
2-{3-[(1H-1,3-Benzodiazol-2-yl)amino]propyl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H19FN6OS
|
1
|
| 1 |
IC50 = 3407 nM
|
|
|
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CP0944107
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-5-chloro-N-[(5-methylpyrimidin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H20ClN7OS
|
1
|
| 1 |
IC50 = 3637 nM
|
|
|
|
CP0909888
|
2-{2-[(1H-1,3-Benzodiazol-5-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide 2-{2-[(1H-1,3-Benzodiazol-4-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H19FN6OS
|
1
|
| 1 |
IC50 = 3727 nM
|
|
|
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CP0957782
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-5-(prop-1-en-2-yl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C23H23FN6OS
|
1
|
| 1 |
IC50 = 4203 nM
|
|
|
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CP0942110
|
2-[(1R,5S,6S)-3-[2-(1H-1,3-Benzodiazol-2-yl)ethyl]-3-azabicyclo[3.1.0]hexan-6-yl]-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C24H23FN6OS
|
1
|
| 1 |
IC50 = 4500 nM
|
|
|
|
CP0874585
|
2-{2-[(1H-1,3-Benzodiazol-5-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H19FN6OS
|
1
|
| 1 |
IC50 = 4794 nM
|
|
|
|
CP0942111
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-1-methyl-1H-imidazole-4-carboxamide
Show/Hide
|
C21H22FN7O
|
1
|
| 1 |
IC50 = 4913 nM
|
|
|
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CP0957776
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]-2-methylpropyl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H23FN6OS
|
1
|
| 1 |
IC50 = 5200 nM
|
|
|
|
CP0942117
|
2-({[3-(1H-1,3-Benzodiazol-2-yl)propyl]amino}methyl)-N-[(3,5-difluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide dihydrochloride
Show/Hide
|
C21H22Cl2F2N6OS
|
1
|
| 1 |
IC50 = 6332 nM
|
|
|
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CP0953918
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-{[2-(pyrrolidin-1-yl)phenyl]methyl}-1,3-thiazole-4-carboxamide
Show/Hide
|
C25H28N6OS
|
1
|
| 1 |
IC50 = 6700 nM
|
|
|
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CP0960693
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-(1H-imidazol-2-ylmethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C18H19N7OS
|
1
|
| 1 |
IC50 = 7230 nM
|
|
|
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CP0880274
|
2-{1-[2-(1H-1,3-Benzodiazol-2-yl)ethyl]-3-methylazetidin-3-yl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C23H23FN6OS
|
1
|
| 1 |
IC50 = 8514 nM
|
|
|
|
CP0944293
|
2-(1-{[2-(1H-1,3-benzodiazol-2-yl)ethyl]amino}-2-methylpropan-2-yl)-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C23H25FN6OS
|
1
|
| 1 |
IC50 = 8920 nM
|
|
|
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CP0887765
|
1-({[2-(1H-1,3-Benzodiazol-2-yl)ethyl]carbamoyl}methyl)-N-[(3-fluoropyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide dihydrochloride
Show/Hide
|
C21H22Cl2FN7O2
|
1
|
| 1 |
IC50 = 9695 nM
|
|
|
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CP0941151
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-methyl-N-phenyl-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H21N5OS
|
1
|
| 1 |
IC50 = 10000 nM
|
|
|
|
CP0942116
|
1-[1-(1H-1,3-Benzodiazol-2-ylmethyl)azetidin-3-yl]-N-[(3-fluoropyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
Show/Hide
|
C21H20FN7O
|
1
|
| 1 |
IC50 = 10490 nM
|
|
|
|
CP0944106
|
1-({1-[2-(1H-1,3-Benzodiazol-2-yl)ethyl]azetidin-3-yl}methyl)-N-[(3-fluoropyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
Show/Hide
|
C23H24FN7O
|
1
|
| 1 |
IC50 = 13560 nM
|
|
|
|
CP0944294
|
2-(1-(2-(1H-benzo[d]imidazol-2-yl)ethyl)pyrrolidin-3-yl)-N-((3-fluoropyridin-2-yl)methyl)thiazole-4-carboxamide
Show/Hide
|
C23H23FN6OS
|
1
|
| 1 |
IC50 = 14100 nM
|
|
|
|
CP0903754
|
2-{1-[3-(1H-1,3-Benzodiazol-2-yl)propyl]azetidin-3-yl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C23H23FN6O2
|
1
|
| 1 |
IC50 = 16000 nM
|
|
|
|
CP0903126
|
1-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-3,5-dimethyl-1H-pyrazole-4-carboxamide
Show/Hide
|
C22H24FN7O
|
1
|
| 1 |
IC50 = 21606 nM
|
|
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CP0912267
|
2-{2-[(1,3-Benzoxazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide trihydrochloride
Show/Hide
|
C20H21Cl3FN5O2S
|
1
|
| 1 |
IC50 = 25000 nM
|
|
|
|
CP0954514
|
2-{2-[2-(1H-1,3-Benzodiazol-2-yl)acetamido]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-1,3-thiazole-4-carboxamide dihydrochloride
Show/Hide
|
C21H21Cl2FN6O2S
|
1
|
| 1 |
IC50 = 25000 nM
|
|
|
|
CP0957328
|
N-[(3-fluoropyridin-2-yl)methyl]-2-(2-{12-oxo-1,8,11-triazatricyclo[7.4.0.02,7]trideca-2(7),3,5,8-tetraen-11-yl}ethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H19FN6O2S
|
1
|
| 1 |
IC50 = 26035 nM
|
|
|
|
CP0880275
|
1-{1-[2-(1H-1,3-Benzodiazol-2-yl)ethyl]piperidin-4-yl}-N-[(3-fluoropyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
Show/Hide
|
C24H26FN7O
|
1
|
| 1 |
IC50 = 27050 nM
|
|
|
|
CP0944104
|
N-[(3-fluoropyridin-2-yl)methyl]-2-(2-{1,8,11-triazatricyclo[7.4.0.02,7]trideca-2(7),3,5,8-tetraen-11-yl}ethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H21FN6OS
|
1
|
| 1 |
IC50 = 27160 nM
|
|
|
|
CP0903143
|
2-{1-[2-(1H-1,3-Benzodiazol-2-yl)ethyl]pyrrolidin-3-yl}-N-(pyridin-2-ylmethyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C23H24N6OS
|
1
|
| 1 |
IC50 = 27700 nM
|
|
|
|
CP0953917
|
6-[2-(1H-1,3-Benzodiazol-2-yl)ethyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxamide
Show/Hide
|
C23H23N5OS
|
1
|
| 1 |
IC50 = 30580 nM
|
|
|
|
CP0880278
|
2-{2-[(1H-1,3-Benzodiazol-2-ylmethyl)amino]ethyl}-N-[(3-fluoropyridin-2-yl)methyl]-5-(propan-2-yl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C23H25FN6OS
|
1
|
| 1 |
IC50 = 30855 nM
|
|
|
|
CP0871792
|
2-(1-((1H-benzo[d]imidazol-2-yl)methyl)azetidin-3-yl)-N-((3-fluoropyridin-2-yl)methyl)oxazole-5-carboxamide
Show/Hide
|
C21H19FN6O2
|
1
|
| 1 |
IC50 = 50000 nM
|
|
|
|
CP0960691
|
1-{[1-(1H-1,3-Benzodiazol-2-ylmethyl)azetidin-3-yl]methyl}-N-[(3-fluoropyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
Show/Hide
|
C22H22FN7O
|
1
|
| 1 |
IC50 = 87000 nM
|
|
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