Brief Information of the Cell Line and Protein
Cell Line ID: CL000148 , Huh-7
Synonyms
HuH-7
HUH-7
HuH7
Huh7
HUH7
HUH7.0
JTC-39
Japanese Tissue Culture-39
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0336
Protein ID: PT01343 , Fibroblast growth factor receptor 4
Gene Name FGFR4
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID P22455
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000148  Protein ID: PT01343
 
Compound ID Compound Name Compound Formula
CP0176348
US10618902, Compound I-279
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C23H23ClFN5O5
 1
1
IC50 = 7.2 nM
   TI
   LI
   LO
   TS
CP0565334
US10189794, Compound I-241
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C23H23Cl2N5O5
 1
1
IC50 = 8.8 nM
   TI
   LI
   LO
   TS
CP0218526
US10618902, Compound I-281
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C23H23F2N5O5
 1
1
IC50 = 11.4 nM
   TI
   LI
   LO
   TS
CP0563793
US10618902, Compound I-250
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C22H23Cl2N5O6S
 1
1
IC50 = 20 nM
   TI
   LI
   LO
   TS
CP0558520
US10618902, Compound I-294
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C25H29N5O5
 1
1
IC50 = 25 nM
   TI
   LI
   LO
   TS
CP0322326
US10618902, Compound I-254
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C23H24ClN5O5
 1
1
IC50 = 29 nM
   TI
   LI
   LO
   TS
CP0322325
N-[(1S,2R)-2-[[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]cyclopentyl]prop-2-enamide
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C24H25Cl2N5O4
 1
1
IC50 = 35 nM
   TI
   LI
   LO
   TS
CP0486123
US10618902, Compound I-255
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C23H25N5O5
 1
1
IC50 = 685 nM
   TI
   LI
   LO
   TS
CP0229508
US10189794, Compound I-240
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C23H23Cl2N5O5
 1
1
IC50 = 2212 nM
   TI
   LI
   LO
   TS
CP0558518
N-[(3R,4S)-4-[[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl]amino]oxolan-3-yl]propanamide
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C23H25Cl2N5O5
 1
1
IC50 = 2926 nM
   TI
   LI
   LO
   TS