| Compound ID |
Compound Name |
Compound Formula |
|
CP0385612
|
6-chloro-2,4-dimethyl-N-[3-[4-[(5R)-2-oxo-5-phenyl-3-(pyridin-4-ylmethyl)imidazolidin-1-yl]piperidin-1-yl]butyl]pyridine-3-carboxamide
Show/Hide
|
C32H39ClN6O2
|
2
|
| 1 |
IC50 = 0.8 nM
|
|
|
| 2 |
IC50 = 5.7 nM
|
|
|
|
CP0391736
|
6-chloro-2,4-dimethyl-N-[3-[4-[(5R)-3-(oxan-4-ylmethyl)-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]butyl]pyridine-3-carboxamide
Show/Hide
|
C32H44ClN5O3
|
2
|
| 1 |
IC50 = 0.8 nM
|
|
|
| 2 |
IC50 = 14.6 nM
|
|
|
|
CP0379631
|
6-chloro-N-[3-[4-[(5R)-3-cyclopentyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]butyl]-2,4-dimethylpyridine-3-carboxamide
Show/Hide
|
C31H42ClN5O2
|
1
|
| 1 |
IC50 = 0.9 nM
|
|
|
|
CP0407515
|
6-chloro-2,4-dimethyl-N-[3-[4-[(5R)-3-[(4-methylpyridin-3-yl)methyl]-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]butyl]pyridine-3-carboxamide
Show/Hide
|
C33H41ClN6O2
|
2
|
| 1 |
IC50 = 1.2 nM
|
|
|
| 2 |
IC50 = 8 nM
|
|
|
|
CP0413861
|
N-[3-[4-[(5R)-3-benzyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]butyl]-6-chloro-2,4-dimethylpyridine-3-carboxamide
Show/Hide
|
C33H40ClN5O2
|
2
|
| 1 |
IC50 = 1.3 nM
|
|
|
| 2 |
IC50 = 9 nM
|
|
|
|
CP0375373
|
6-chloro-N-[(3S)-3-[4-[(5R)-3-cyclohexyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]butyl]-2,4-dimethylpyridine-3-carboxamide
Show/Hide
|
C32H44ClN5O2
|
2
|
| 1 |
IC50 = 1.5 nM
|
|
|
| 2 |
IC50 = 9.6 nM
|
|
|
|
CP0540420
|
6-chloro-N-[(3R)-3-[4-[(5R)-3-cyclohexyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]butyl]-2,4-dimethylpyridine-3-carboxamide
Show/Hide
|
C32H44ClN5O2
|
2
|
| 1 |
IC50 = 1.5 nM
|
|
|
| 2 |
IC50 = 13.6 nM
|
|
|
|
CP0379587
|
6-chloro-N-[3-[4-[(5R)-3-(cyclohexylmethyl)-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]butyl]-2,4-dimethylpyridine-3-carboxamide
Show/Hide
|
C33H46ClN5O2
|
2
|
| 1 |
IC50 = 1.8 nM
|
|
|
| 2 |
IC50 = 7.7 nM
|
|
|
|
CP0413840
|
6-chloro-N-[3-[4-[(5R)-3-cyclobutyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]butyl]-2,4-dimethylpyridine-3-carboxamide
Show/Hide
|
C30H40ClN5O2
|
2
|
| 1 |
IC50 = 2.3 nM
|
|
|
| 2 |
IC50 = 19.5 nM
|
|
|
|
CP0379630
|
6-chloro-N-[3-[4-(3-cyclohexyl-2-oxo-5-thiophen-3-ylimidazolidin-1-yl)piperidin-1-yl]butyl]-2,4-dimethylpyridine-3-carboxamide
Show/Hide
|
C30H42ClN5O2S
|
1
|
| 1 |
IC50 = 2.4 nM
|
|
|
|
CP0531452
|
6-chloro-2,4-dimethyl-N-[3-[4-[(5R)-2-oxo-5-phenyl-3-(pyridin-2-ylmethyl)imidazolidin-1-yl]piperidin-1-yl]butyl]pyridine-3-carboxamide
Show/Hide
|
C32H39ClN6O2
|
1
|
| 1 |
IC50 = 2.9 nM
|
|
|
|
CP0409023
|
6-chloro-2,4-dimethyl-N-[3-[4-[(5R)-2-oxo-5-phenyl-3-(pyridin-3-ylmethyl)imidazolidin-1-yl]piperidin-1-yl]butyl]pyridine-3-carboxamide
Show/Hide
|
C32H39ClN6O2
|
2
|
| 1 |
IC50 = 3.4 nM
|
|
|
| 2 |
IC50 = 52.4 nM
|
|
|
|
CP0391724
|
N-[3-[4-[(5R)-3-tert-butyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]butyl]-6-chloro-2,4-dimethylpyridine-3-carboxamide
Show/Hide
|
C30H42ClN5O2
|
1
|
| 1 |
IC50 = 3.6 nM
|
|
|
|
CP0408996
|
4-[[(4R)-3-[1-[4-[(6-chloro-2,4-dimethylpyridine-3-carbonyl)amino]butan-2-yl]piperidin-4-yl]-2-oxo-4-phenylimidazolidin-1-yl]methyl]benzoic acid
Show/Hide
|
C34H40ClN5O4
|
2
|
| 1 |
IC50 = 3.6 nM
|
|
|
| 2 |
IC50 = 42.2 nM
|
|
|
|
CP0467621
|
(4R)-3-[1-[1-(6-chloro-2,4-dimethylpyridine-3-carbonyl)-4-methylpiperidin-4-yl]piperidin-4-yl]-1-cyclohexyl-4-phenylimidazolidin-2-one
Show/Hide
|
C34H46ClN5O2
|
1
|
| 1 |
IC50 = 4.2 nM
|
|
|
|
CP0379629
|
N-[(3S)-3-[4-[(5R)-3-cyclohexyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
Show/Hide
|
C31H44N6O2
|
2
|
| 1 |
IC50 = 4.4 nM
|
|
|
| 2 |
IC50 = 16.6 nM
|
|
|
|
CP0379624
|
N-[3-[4-[3-cyclohexyl-5-(3,5-dimethylphenyl)-2-oxoimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
Show/Hide
|
C33H48N6O2
|
2
|
| 1 |
IC50 = 4.7 nM
|
|
|
| 2 |
IC50 = 36.5 nM
|
|
|
|
CP0390755
|
N-[3-[4-[5-(3-bromophenyl)-3-cyclohexyl-2-oxoimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
Show/Hide
|
C31H43BrN6O2
|
2
|
| 1 |
IC50 = 5.1 nM
|
|
|
| 2 |
IC50 = 22 nM
|
|
|
|
CP0395775
|
6-chloro-2,4-dimethyl-N-[3-[4-[(5R)-2-oxo-5-phenyl-3-propan-2-ylimidazolidin-1-yl]piperidin-1-yl]butyl]pyridine-3-carboxamide
Show/Hide
|
C29H40ClN5O2
|
1
|
| 1 |
IC50 = 5.3 nM
|
|
|
|
CP0409022
|
(4R)-1-cyclohexyl-3-[1-[1-(4,6-dimethylpyrimidine-5-carbonyl)-4-methylpiperidin-4-yl]piperidin-4-yl]-4-phenylimidazolidin-2-one
Show/Hide
|
C33H46N6O2
|
1
|
| 1 |
IC50 = 5.8 nM
|
|
|
|
CP0467620
|
N-[3-[4-[5-(3-chlorophenyl)-3-cyclohexyl-2-oxoimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
Show/Hide
|
C31H43ClN6O2
|
2
|
| 1 |
IC50 = 5.8 nM
|
|
|
| 2 |
IC50 = 19.5 nM
|
|
|
|
CP0390753
|
N-[3-[4-[3-cyclohexyl-5-(3-methylphenyl)-2-oxoimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
Show/Hide
|
C32H46N6O2
|
2
|
| 1 |
IC50 = 6 nM
|
|
|
| 2 |
IC50 = 31 nM
|
|
|
|
CP0413843
|
6-chloro-2,4-dimethyl-N-[3-[4-[(5R)-3-(oxan-4-yl)-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]butyl]pyridine-3-carboxamide
Show/Hide
|
C31H42ClN5O3
|
1
|
| 1 |
IC50 = 6.3 nM
|
|
|
|
CP0390757
|
4-[4-[[4-[(5R)-3-cyclohexyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]methyl]phenoxy]benzoic acid
Show/Hide
|
C34H39N3O4
|
2
|
| 1 |
IC50 = 6.4 nM
|
|
|
| 2 |
IC50 = 38.9 nM
|
|
|
|
CP0413857
|
4-[4-[[4-[(5R)-3-cyclohexyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]methyl]phenoxy]benzamide
Show/Hide
|
C34H40N4O3
|
2
|
| 1 |
IC50 = 6.9 nM
|
|
|
| 2 |
IC50 = 18 nM
|
|
|
|
CP0379626
|
N-[3-[4-[3-cyclohexyl-5-(3-fluoro-5-methylphenyl)-2-oxoimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
Show/Hide
|
C32H45FN6O2
|
2
|
| 1 |
IC50 = 7.1 nM
|
|
|
| 2 |
IC50 = 32 nM
|
|
|
|
CP0379585
|
4-[4-[[4-[(5R)-3-cyclohexyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]methyl]phenoxy]-N,N-dimethylbenzamide
Show/Hide
|
C36H44N4O3
|
2
|
| 1 |
IC50 = 7.5 nM
|
|
|
| 2 |
IC50 = 15.5 nM
|
|
|
|
CP0403867
|
6-chloro-2,4-dimethyl-N-[3-[4-[(5R)-2-oxo-5-phenyl-3-propylimidazolidin-1-yl]piperidin-1-yl]butyl]pyridine-3-carboxamide
Show/Hide
|
C29H40ClN5O2
|
2
|
| 1 |
IC50 = 7.5 nM
|
|
|
| 2 |
IC50 = 19.4 nM
|
|
|
|
CP0407513
|
4-[4-[[4-[(5R)-3-cyclohexyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]methyl]phenoxy]-N-methylbenzamide
Show/Hide
|
C35H42N4O3
|
2
|
| 1 |
IC50 = 9.6 nM
|
|
|
| 2 |
IC50 = 11.6 nM
|
|
|
|
CP0494102
|
3,5-dichloro-N-(3-(4-((6-chloropyridin-2-yloxy)(4-(methylsulfonyl)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
Show/Hide
|
C28H31Cl3N4O4S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0413842
|
(4R)-1-cyclohexyl-4-phenyl-3-[1-[(4-phenylphenyl)methyl]piperidin-4-yl]imidazolidin-2-one
Show/Hide
|
C33H39N3O
|
2
|
| 1 |
IC50 = 12.4 nM
|
|
|
| 2 |
IC50 = 41.8 nM
|
|
|
|
CP0413838
|
3-[4-[[4-[(5R)-3-cyclohexyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]methyl]phenoxy]benzoic acid
Show/Hide
|
C34H39N3O4
|
1
|
| 1 |
IC50 = 12.7 nM
|
|
|
|
CP0379622
|
(4R)-1-cyclohexyl-3-[1-[(4-phenoxyphenyl)methyl]piperidin-4-yl]-4-phenylimidazolidin-2-one
Show/Hide
|
C33H39N3O2
|
2
|
| 1 |
IC50 = 13.3 nM
|
|
|
| 2 |
IC50 = 22.5 nM
|
|
|
|
CP0390754
|
N-[(3R)-3-[4-[(5R)-3-cyclohexyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
Show/Hide
|
C31H44N6O2
|
2
|
| 1 |
IC50 = 13.6 nM
|
|
|
| 2 |
IC50 = 19.8 nM
|
|
|
|
CP0379625
|
N-[3-[4-[3-cyclohexyl-5-(3-fluorophenyl)-2-oxoimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
Show/Hide
|
C31H43FN6O2
|
2
|
| 1 |
IC50 = 15 nM
|
|
|
| 2 |
IC50 = 25.9 nM
|
|
|
|
CP0413841
|
(4R)-1-cyclohexyl-3-[1-[(4-morpholin-4-ylphenyl)methyl]piperidin-4-yl]-4-phenylimidazolidin-2-one
Show/Hide
|
C31H42N4O2
|
1
|
| 1 |
IC50 = 15.2 nM
|
|
|
|
CP0403869
|
4-[[4-[(5R)-3-cyclohexyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]methyl]-N-methylbenzamide
Show/Hide
|
C29H38N4O2
|
2
|
| 1 |
IC50 = 15.8 nM
|
|
|
| 2 |
IC50 = 85.1 nM
|
|
|
|
CP0390756
|
(4R)-1-cyclohexyl-4-phenyl-3-[1-[(4-pyrimidin-5-ylphenyl)methyl]piperidin-4-yl]imidazolidin-2-one
Show/Hide
|
C31H37N5O
|
2
|
| 1 |
IC50 = 17.3 nM
|
|
|
| 2 |
IC50 = 18.9 nM
|
|
|
|
CP0375304
|
(4R)-1-cyclohexyl-4-phenyl-3-[1-[(4-pyridin-3-ylphenyl)methyl]piperidin-4-yl]imidazolidin-2-one
Show/Hide
|
C32H38N4O
|
2
|
| 1 |
IC50 = 17.9 nM
|
|
|
| 2 |
IC50 = 43.7 nM
|
|
|
|
CP0511363
|
3,5-dichloro-N-(3-(4-((6-chloropyridin-2-yloxy)(4-(trifluoromethyl)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
Show/Hide
|
C28H28Cl3F3N4O2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0860204
|
rac-N-(3-(4-(3-cyclohexyl-2-oxo-5-phenylimidazolidin-1-yl)piperidin-1-yl)butyl)-4,6-dimethylpyrimidine-5-carboxamide
Show/Hide
|
C31H44N6O2
|
2
|
| 1 |
IC50 = 20.7 nM
|
|
|
| 2 |
IC50 = 77 nM
|
|
|
|
CP0403866
|
6-chloro-N-[3-[4-[(5R)-3-ethyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]butyl]-2,4-dimethylpyridine-3-carboxamide
Show/Hide
|
C28H38ClN5O2
|
1
|
| 1 |
IC50 = 24.7 nM
|
|
|
|
CP0463516
|
N-[3-[4-(N-benzyl-4-bromoanilino)piperidin-1-yl]butyl]-3,5-dichloropyridine-4-carboxamide
Show/Hide
|
C28H31BrCl2N4O
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0466185
|
3,5-dichloro-N-(3-(4-(2-(4-(trifluoromethyl)phenyl)benzo[d][1,3]dioxol-2-yl)piperidin-1-yl)butyl)isonicotinamide
Show/Hide
|
C29H28Cl2F3N3O3
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0484962
|
3,5-dichloro-N-(3-(4-((6-chloropyridin-2-yloxy)(4-(trifluoromethoxy)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
Show/Hide
|
C28H28Cl3F3N4O3
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0503385
|
3,5-dichloro-N-(3-(4-((pyridin-2-yloxy)(4-(trifluoromethyl)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
Show/Hide
|
C28H29Cl2F3N4O2
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0390752
|
N-[3-[4-[5-(3-cyanophenyl)-3-cyclohexyl-2-oxoimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
Show/Hide
|
C32H43N7O2
|
2
|
| 1 |
IC50 = 32.2 nM
|
|
|
| 2 |
IC50 = 34.8 nM
|
|
|
|
CP0379586
|
(4R)-1-cyclohexyl-4-phenyl-3-[1-[(4-pyridin-4-ylphenyl)methyl]piperidin-4-yl]imidazolidin-2-one
Show/Hide
|
C32H38N4O
|
2
|
| 1 |
IC50 = 39.3 nM
|
|
|
| 2 |
IC50 = 43.5 nM
|
|
|
|
CP0460765
|
3,5-dichloro-N-(3-(4-((6-methylpyridin-2-yloxy)(4-(trifluoromethyl)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
Show/Hide
|
C29H31Cl2F3N4O2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0484960
|
3,5-dichloro-N-(3-(4-((3-fluorophenoxy)(4-(trifluoromethyl)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
Show/Hide
|
C29H29Cl2F4N3O2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0554738
|
3,5-dichloro-N-(3-(4-(2-(4-(trifluoromethyl)phenyl)-2,3-dihydrobenzofuran-2-yl)piperidin-1-yl)butyl)isonicotinamide
Show/Hide
|
C30H30Cl2F3N3O2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0554743
|
3,5-dichloro-N-(3-(4-((6-cyanopyridin-2-yloxy)(4-(trifluoromethyl)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
Show/Hide
|
C29H28Cl2F3N5O2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0957158
|
Schering C
Show/Hide
|
C28H37BrN4O3
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0467624
|
(4R)-1-cyclohexyl-3-[1-[[4-(2-methyltetrazol-5-yl)phenyl]methyl]piperidin-4-yl]-4-phenylimidazolidin-2-one
Show/Hide
|
C29H37N7O
|
1
|
| 1 |
IC50 = 43.7 nM
|
|
|
|
CP0409018
|
N-[3-[4-(3-cyclohexyl-2-oxo-5-thiophen-3-ylimidazolidin-1-yl)piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
Show/Hide
|
C29H42N6O2S
|
2
|
| 1 |
IC50 = 44.4 nM
|
|
|
| 2 |
IC50 = 85 nM
|
|
|
|
CP0479105
|
3,5-dichloro-N-(3-(4-((4-methylpyridin-2-yloxy)(4-(trifluoromethyl)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
Show/Hide
|
C29H31Cl2F3N4O2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0486563
|
3,5-dichloro-N-(3-(4-((3-cyanophenoxy)(4-(trifluoromethyl)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
Show/Hide
|
C30H29Cl2F3N4O2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0511055
|
3,5-dichloro-N-(3-(4-(phenoxy(4-(trifluoromethyl)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
Show/Hide
|
C29H30Cl2F3N3O2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0379623
|
(4R)-3-[1-(3H-benzimidazol-5-ylmethyl)piperidin-4-yl]-1-cyclohexyl-4-phenylimidazolidin-2-one
Show/Hide
|
C28H35N5O
|
2
|
| 1 |
IC50 = 50.7 nM
|
|
|
| 2 |
IC50 = 91 nM
|
|
|
|
CP0484618
|
3,5-dichloro-N-(3-(4-((3-methylpyridin-2-yloxy)(4-(trifluoromethyl)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
Show/Hide
|
C29H31Cl2F3N4O2
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0511355
|
3,5-dichloro-N-(3-(4-((3-chlorophenoxy)(4-(trifluoromethyl)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
Show/Hide
|
C29H29Cl3F3N3O2
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0513676
|
3,5-dichloro-N-(3-(4-((4-chloropyridin-2-yloxy)(4-(trifluoromethyl)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
Show/Hide
|
C28H28Cl3F3N4O2
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0411656
|
N-[3-[4-[3-cyclohexyl-5-(2-fluorophenyl)-2-oxoimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
Show/Hide
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C31H43FN6O2
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2
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| 1 |
IC50 = 91 nM
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| 2 |
IC50 = 155 nM
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CP0486561
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3,5-dichloro-N-(3-(4-((2-cyanophenoxy)(4-(trifluoromethyl)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
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C30H29Cl2F3N4O2
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1
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| 1 |
IC50 = 100 nM
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CP0511056
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3,5-dichloro-N-(3-(4-((2-chlorophenoxy)(4-(trifluoromethyl)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
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C29H29Cl3F3N3O2
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1
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| 1 |
IC50 = 120 nM
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CP0511354
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N-[3-[4-[(4-bromophenyl)-phenoxymethyl]piperidin-1-yl]butyl]-3,5-dichloropyridine-4-carboxamide
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C28H30BrCl2N3O2
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1
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| 1 |
IC50 = 130 nM
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CP0524507
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(E)-N-(3-(4-((4-bromophenyl)(ethoxyimino)methyl)piperidin-1-yl)butyl)-3,5-dichloroisonicotinamide
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C24H29BrCl2N4O2
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1
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| 1 |
IC50 = 130 nM
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CP0554741
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3,5-dichloro-N-(3-(4-((4-(trifluoromethyl)phenyl)(6-(trifluoromethyl)pyridin-2-yloxy)methyl)piperidin-1-yl)butyl)isonicotinamide
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C29H28Cl2F6N4O2
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1
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| 1 |
IC50 = 130 nM
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CP0486566
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3,5-dichloro-N-(3-(4-((3-chloropyridin-2-yloxy)(4-(trifluoromethyl)phenyl)methyl)piperidin-1-yl)butyl)isonicotinamide
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C28H28Cl3F3N4O2
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1
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| 1 |
IC50 = 140 nM
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CP0505365
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N-[3-[4-[(4-bromophenyl)-pyridin-2-yloxymethyl]piperidin-1-yl]butyl]-3,5-dichloropyridine-4-carboxamide
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C27H29BrCl2N4O2
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1
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| 1 |
IC50 = 140 nM
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CP0554740
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N-[3-[4-[(4-bromophenyl)-(4-methylpyridin-2-yl)oxymethyl]piperidin-1-yl]butyl]-3,5-dichloropyridine-4-carboxamide
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C28H31BrCl2N4O2
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1
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| 1 |
IC50 = 140 nM
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CP0413837
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N-[3-[4-[3-cyclohexyl-5-(6-methylpyridin-2-yl)-2-oxoimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
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C31H45N7O2
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1
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| 1 |
IC50 = 149.8 nM
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CP0379620
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methyl 3-[1-cyclohexyl-3-[1-[4-[(4,6-dimethylpyrimidine-5-carbonyl)amino]butan-2-yl]piperidin-4-yl]-2-oxoimidazolidin-4-yl]benzoate
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C33H46N6O4
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2
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| 1 |
IC50 = 157.6 nM
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| 2 |
IC50 = 175.8 nM
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CP0379621
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(4R)-1-cyclohexyl-4-phenyl-3-[1-[(4-pyrimidin-2-ylphenyl)methyl]piperidin-4-yl]imidazolidin-2-one
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C31H37N5O
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2
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| 1 |
IC50 = 169 nM
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| 2 |
IC50 = 334 nM
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CP0911520
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(E)-3-(3-(4-((4-bromophenyl)(ethoxyimino)methyl)piperidin-1-yl)propylcarbamoyl)-2,4-dimethylpyridine 1-oxide
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C25H33BrN4O3
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1
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| 1 |
IC50 = 180 nM
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CP0486565
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N-[3-[4-[(4-bromophenyl)-(3-methylpyridin-2-yl)oxymethyl]piperidin-1-yl]butyl]-3,5-dichloropyridine-4-carboxamide
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C28H31BrCl2N4O2
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1
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| 1 |
IC50 = 190 nM
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CP0395765
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N-[3-[4-[5-(2-chlorophenyl)-3-cyclohexyl-2-oxoimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
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C31H43ClN6O2
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2
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| 1 |
IC50 = 195 nM
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| 2 |
IC50 = 1526 nM
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CP0513675
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N-[3-[4-[(4-bromophenyl)-(6-methylpyridin-2-yl)oxymethyl]piperidin-1-yl]butyl]-3,5-dichloropyridine-4-carboxamide
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C28H31BrCl2N4O2
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1
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| 1 |
IC50 = 220 nM
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CP0910882
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(E)-3-(3-(4-((4-bromophenyl)(ethoxyimino)methyl)piperidin-1-yl)butylcarbamoyl)-2,4-dimethylpyridine 1-oxide
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C26H35BrN4O3
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1
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| 1 |
IC50 = 290 nM
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CP0411652
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N-[3-[4-(3-cyclohexyl-2-oxo-5-pyridin-2-ylimidazolidin-1-yl)piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
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C30H43N7O2
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1
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| 1 |
IC50 = 300.7 nM
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CP0449632
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N-[3-[4-[3-cyclohexyl-5-(2-methylphenyl)-2-oxoimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
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C32H46N6O2
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1
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| 1 |
IC50 = 322 nM
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CP0426747
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N-[3-[4-[5-(4-bromophenyl)-3-cyclohexyl-2-oxoimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
Show/Hide
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C31H43BrN6O2
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1
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| 1 |
IC50 = 700.8 nM
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CP0531886
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4-[(4R)-3-[1-[4-[(6-chloro-2,4-dimethylpyridine-3-carbonyl)amino]butan-2-yl]piperidin-4-yl]-2-oxo-4-phenylimidazolidin-1-yl]cyclohexane-1-carboxylic acid
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C33H44ClN5O4
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1
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| 1 |
IC50 = 807.2 nM
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CP0409008
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N-[3-[4-(3-cyclohexyl-2-oxo-5-pyridin-3-ylimidazolidin-1-yl)piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
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C30H43N7O2
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1
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| 1 |
IC50 = 832 nM
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CP0554739
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N-[3-[4-[(4-bromophenyl)-pyridin-3-yloxymethyl]piperidin-1-yl]butyl]-3,5-dichloropyridine-4-carboxamide
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C27H29BrCl2N4O2
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1
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| 1 |
IC50 = 970 nM
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CP0460766
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methyl 6-[[1-[4-[(3,5-dichloropyridine-4-carbonyl)amino]butan-2-yl]piperidin-4-yl]-[4-(trifluoromethyl)phenyl]methoxy]pyridine-2-carboxylate
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C30H31Cl2F3N4O4
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1
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| 1 |
IC50 = 1050 nM
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CP0411626
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N-[(3S)-3-[4-[(5S)-3-cyclohexyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
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C31H44N6O2
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1
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| 1 |
IC50 = 1465 nM
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CP0395771
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(4R)-1-cyclohexyl-3-[1-[[1-(2-methylphenyl)piperidin-4-yl]methyl]piperidin-4-yl]-4-phenylimidazolidin-2-one
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C33H46N4O
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1
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| 1 |
IC50 = 1595 nM
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CP0541205
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(E)-N-(3-(4-((4-bromophenyl)(ethoxyimino)methyl)piperidin-1-yl)-3-methylbutyl)-3,5-dichloroisonicotinamide
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C25H31BrCl2N4O2
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1
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| 1 |
IC50 = 1760 nM
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CP0530022
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N-[3-[4-[(4-bromophenyl)-hydroxymethyl]piperidin-1-yl]butyl]-3,5-dichloropyridine-4-carboxamide
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C22H26BrCl2N3O2
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1
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| 1 |
IC50 = 3390 nM
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CP0484961
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N-[3-[4-[(4-bromophenyl)-(5-methylpyridin-2-yl)oxymethyl]piperidin-1-yl]butyl]-3,5-dichloropyridine-4-carboxamide
Show/Hide
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C28H31BrCl2N4O2
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1
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| 1 |
IC50 = 3800 nM
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CP0935650
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(E)-3-((3-(4-((4-bromophenyl)(ethoxyimino)methyl)piperidin-1-yl)butyl)(methyl)carbamoyl)-2,4-dimethylpyridine 1-oxide
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C27H37BrN4O3
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1
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| 1 |
IC50 = 5620 nM
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CP0464755
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N-[3-[4-(7-bromo-1H-2,3-benzoxazin-4-yl)piperidin-1-yl]butyl]-3,5-dichloropyridine-4-carboxamide
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C23H25BrCl2N4O2
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1
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| 1 |
IC50 = 12250 nM
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CP0411627
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N-[(3R)-3-[4-[(5S)-3-cyclohexyl-2-oxo-5-phenylimidazolidin-1-yl]piperidin-1-yl]butyl]-4,6-dimethylpyrimidine-5-carboxamide
Show/Hide
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C31H44N6O2
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1
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| 1 |
IC50 > 16000 nM
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CP0900117
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(E)-3-(2-(4-((4-bromophenyl)(ethoxyimino)methyl)piperidin-1-yl)propylcarbamoyl)-2,4-dimethylpyridine 1-oxide
Show/Hide
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C25H33BrN4O3
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1
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| 1 |
IC50 = 17010 nM
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CP0501376
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(E)-N-(2-(1-(4-((4-bromophenyl)(ethoxyimino)methyl)piperidin-1-yl)cyclopropyl)ethyl)-3,5-dichloroisonicotinamide
Show/Hide
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C25H29BrCl2N4O2
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1
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| 1 |
IC50 = 21370 nM
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