| Compound ID |
Compound Name |
Compound Formula |
|
CP0519695
|
1-[[6-chloro-2-(3,6-dihydro-2H-pyridin-1-yl)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C18H17ClN4O2S
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0557515
|
6-[(6-methoxy-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
Show/Hide
|
C21H17N3O3
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0510384
|
1-[[6-chloro-2-(diethylamino)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C17H19ClN4O2S
|
1
|
| 1 |
IC50 = 6.2 nM
|
|
|
|
CP0533843
|
5-[[6-chloro-2-(3,6-dihydro-2H-pyridin-1-yl)-1,3-benzothiazol-4-yl]sulfanyl]furan-2-carboxylic acid
Show/Hide
|
C17H13ClN2O3S2
|
1
|
| 1 |
IC50 = 6.4 nM
|
|
|
|
CP0392335
|
6-[(6-chloro-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
Show/Hide
|
C20H14ClN3O2
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0411727
|
1-[(5-chloro-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C19H15ClN4O2
|
1
|
| 1 |
IC50 = 9.4 nM
|
|
|
|
CP0481525
|
1-[[2-(3,6-dihydro-2H-pyridin-1-yl)-6-ethenyl-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C20H20N4O2S
|
1
|
| 1 |
IC50 = 9.9 nM
|
|
|
|
CP0489170
|
6-[(6-bromo-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
Show/Hide
|
C20H14BrN3O2
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0481527
|
1-[[6-chloro-2-[ethyl(methyl)amino]-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C16H17ClN4O2S
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0523257
|
6-[[2-phenyl-6-(trifluoromethyl)pyrazolo[1,5-a]pyridin-3-yl]methyl]pyridine-2-carboxylic acid
Show/Hide
|
C21H14F3N3O2
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0566082
|
1-[[2-(3,6-dihydro-2H-pyridin-1-yl)-6-fluoro-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C18H17FN4O2S
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0489171
|
6-[(6-methyl-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
Show/Hide
|
C21H17N3O2
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0560506
|
6-[(6-ethenyl-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
Show/Hide
|
C22H17N3O2
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0484547
|
1-[(5-chloro-2-phenyl-1-benzofuran-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C20H15ClN2O3
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0559181
|
1-[[6-bromo-2-(3,6-dihydro-2H-pyridin-1-yl)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C18H17BrN4O2S
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0475870
|
3-[(6-chloro-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]benzoic acid
Show/Hide
|
C21H15ClN2O2
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0472686
|
1-[(6-chloro-2-pyrrolidin-1-yl-1,3-benzothiazol-4-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C17H17ClN4O2S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0510383
|
1-[[6-chloro-2-(5-methyl-3,6-dihydro-2H-pyridin-1-yl)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C19H19ClN4O2S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0517957
|
1-[(6-chloro-2-phenyl-1,3-benzothiazol-4-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C19H14ClN3O2S
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0460415
|
1-[[2-(3,6-dihydro-2H-pyridin-1-yl)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C18H18N4O2S
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0475118
|
1-[(6-chloro-2-prop-1-en-2-yl-1,3-benzothiazol-4-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C16H14ClN3O2S
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
|
CP0571939
|
1-[[2-(3,6-dihydro-2H-pyridin-1-yl)-6-methoxy-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C19H20N4O3S
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0460416
|
1-[(6-chloro-2-piperidin-1-yl-1,3-benzothiazol-4-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C18H19ClN4O2S
|
1
|
| 1 |
IC50 = 43 nM
|
|
|
|
CP0538602
|
6-[(2-tert-butyl-6-chloropyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
Show/Hide
|
C18H18ClN3O2
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0566081
|
1-[[6-chloro-2-(3,6-dihydro-2H-pyridin-1-yl)-1,3-benzothiazol-4-yl]methyl]pyrazole-3-carboxylic acid
Show/Hide
|
C17H15ClN4O2S
|
1
|
| 1 |
IC50 = 51 nM
|
|
|
|
CP0534665
|
5-[[6-chloro-2-(3,6-dihydro-2H-pyridin-1-yl)-1,3-benzothiazol-4-yl]methyl]furan-2-carboxylic acid
Show/Hide
|
C18H15ClN2O3S
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0494019
|
5-[(6-methoxy-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]furan-2-carboxylic acid
Show/Hide
|
C20H16N2O4
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0571941
|
1-[(6-chloro-2-morpholin-4-yl-1,3-benzothiazol-4-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C17H17ClN4O3S
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0481526
|
1-[[6-chloro-2-(4-methyl-3,6-dihydro-2H-pyridin-1-yl)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C19H19ClN4O2S
|
1
|
| 1 |
IC50 = 64 nM
|
|
|
|
CP0519271
|
1-[(6-chloro-2-thiomorpholin-4-yl-1,3-benzothiazol-4-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C17H17ClN4O2S2
|
1
|
| 1 |
IC50 = 66 nM
|
|
|
|
CP0458617
|
1-[(5-chloro-2-cyclohexylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C19H21ClN4O2
|
1
|
| 1 |
IC50 = 71 nM
|
|
|
|
CP0570333
|
6-[(6-chloro-2-piperidin-1-ylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
Show/Hide
|
C19H19ClN4O2
|
1
|
| 1 |
IC50 = 79 nM
|
|
|
|
CP0557516
|
6-[(6-methylsulfanyl-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
Show/Hide
|
C21H17N3O2S
|
1
|
| 1 |
IC50 = 87 nM
|
|
|
|
CP0479672
|
1-[(5-chloro-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]pyrazole-3-carboxylic acid
Show/Hide
|
C18H13ClN4O2
|
1
|
| 1 |
IC50 = 89 nM
|
|
|
|
CP0523133
|
1-[(5-chloro-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-propylpyrazole-3-carboxylic acid
Show/Hide
|
C21H19ClN4O2
|
1
|
| 1 |
IC50 = 97 nM
|
|
|
|
CP0458381
|
1-[[2-(3,6-dihydro-2H-pyridin-1-yl)-6-(trifluoromethoxy)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C19H17F3N4O3S
|
1
|
| 1 |
IC50 = 97 nM
|
|
|
|
CP0475117
|
1-[[6-chloro-2-(dimethylamino)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C15H15ClN4O2S
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0446923
|
1-[[5-chloro-2-(3-methoxyphenyl)pyrazolo[1,5-a]pyridin-7-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C20H17ClN4O3
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0559183
|
1-[[6-chloro-2-(cyclohexen-1-yl)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C19H18ClN3O2S
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0566083
|
1-[[6-chloro-2-(2,5-dihydropyrrol-1-yl)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C17H15ClN4O2S
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0569200
|
6-[(6-chloro-2-thiophen-3-ylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
Show/Hide
|
C18H12ClN3O2S
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0575551
|
2-[(6-chloro-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C18H12ClN3O2S
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0479676
|
5-methyl-1-[(2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]pyrazole-3-carboxylic acid
Show/Hide
|
C19H16N4O2
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0523259
|
6-[[6-chloro-2-(furan-3-yl)pyrazolo[1,5-a]pyridin-3-yl]methyl]pyridine-2-carboxylic acid
Show/Hide
|
C18H12ClN3O3
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0479674
|
1-[[5-chloro-2-(3-chlorophenyl)pyrazolo[1,5-a]pyridin-7-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C19H14Cl2N4O2
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0481523
|
5-[[6-chloro-2-(3,6-dihydro-2H-pyridin-1-yl)-1,3-benzothiazol-4-yl]oxy]furan-2-carboxylic acid
Show/Hide
|
C17H13ClN2O4S
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0475913
|
1-[[2-(3,6-dihydro-2H-pyridin-1-yl)-6-prop-1-en-2-yl-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C21H22N4O2S
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0472709
|
1-[(5-chloro-2-cyclopropylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C16H15ClN4O2
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0549006
|
1-[(5-chloro-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]pyrrole-3-carboxylic acid
Show/Hide
|
C19H14ClN3O2
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0569309
|
6-[(6-cyclopropyl-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
Show/Hide
|
C23H19N3O2
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0519374
|
1-[[6-acetyl-2-(3,6-dihydro-2H-pyridin-1-yl)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C20H20N4O3S
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0560508
|
6-[[6-chloro-2-(2-methylpropyl)pyrazolo[1,5-a]pyridin-3-yl]methyl]pyridine-2-carboxylic acid
Show/Hide
|
C18H18ClN3O2
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0519381
|
1-[[2-(3,6-dihydro-2H-pyridin-1-yl)-6-(dimethylamino)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C20H23N5O2S
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0454782
|
1-[[5-chloro-2-(2-chlorophenyl)pyrazolo[1,5-a]pyridin-7-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C19H14Cl2N4O2
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0520187
|
1-[[6-cyano-2-(3,6-dihydro-2H-pyridin-1-yl)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C19H17N5O2S
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0475912
|
1-[[6-chloro-2-(3,6-dihydro-2H-pyridin-1-yl)-1,3-benzothiazol-4-yl]methyl]pyrrole-3-carboxylic acid
Show/Hide
|
C18H16ClN3O2S
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0560510
|
6-[(6-chloro-2-thiomorpholin-4-ylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
Show/Hide
|
C18H17ClN4O2S
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0411726
|
1-[[6-chloro-2-[ethyl(propyl)amino]-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C18H21ClN4O2S
|
1
|
| 1 |
IC50 = 270 nM
|
|
|
|
CP0519382
|
1-[[2-(azepan-1-yl)-6-chloro-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C19H21ClN4O2S
|
1
|
| 1 |
IC50 = 270 nM
|
|
|
|
CP0454781
|
1-[[5-chloro-2-(4-chlorophenyl)pyrazolo[1,5-a]pyridin-7-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C19H14Cl2N4O2
|
1
|
| 1 |
IC50 = 290 nM
|
|
|
|
CP0408380
|
6-[(2-phenyl-6-prop-1-en-2-ylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
Show/Hide
|
C23H19N3O2
|
1
|
| 1 |
IC50 = 290 nM
|
|
|
|
CP0472708
|
1-[(5-chloro-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-ethylpyrazole-3-carboxylic acid
Show/Hide
|
C20H17ClN4O2
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0549007
|
5-methyl-1-[[2-phenyl-5-(trifluoromethyl)pyrazolo[1,5-a]pyridin-7-yl]methyl]pyrazole-3-carboxylic acid
Show/Hide
|
C20H15F3N4O2
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0475116
|
1-[[2-(azetidin-1-yl)-6-chloro-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C16H15ClN4O2S
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
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CP0472711
|
1-[(5-ethenyl-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C21H18N4O2
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0411669
|
6-[(6-fluoro-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
Show/Hide
|
C20H14FN3O2
|
1
|
| 1 |
IC50 = 380 nM
|
|
|
|
CP0454779
|
1-[[5-chloro-2-(4-methoxyphenyl)pyrazolo[1,5-a]pyridin-7-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C20H17ClN4O3
|
1
|
| 1 |
IC50 = 410 nM
|
|
|
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CP0507074
|
1-[(5-chloro-2-cyclopentylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C18H19ClN4O2
|
1
|
| 1 |
IC50 = 410 nM
|
|
|
|
CP0447004
|
1-[(6-chloro-2-cyclohexyl-1,3-benzothiazol-4-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C19H20ClN3O2S
|
1
|
| 1 |
IC50 = 430 nM
|
|
|
|
CP0557517
|
6-[(6-cyano-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
Show/Hide
|
C21H14N4O2
|
1
|
| 1 |
IC50 = 440 nM
|
|
|
|
CP0472712
|
5-methyl-1-[(5-methyl-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]pyrazole-3-carboxylic acid
Show/Hide
|
C20H18N4O2
|
1
|
| 1 |
IC50 = 450 nM
|
|
|
|
CP0511748
|
1-[[6-chloro-2-(methylamino)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C14H13ClN4O2S
|
1
|
| 1 |
IC50 = 470 nM
|
|
|
|
CP0396231
|
6-[[6-chloro-2-(3-chlorophenyl)pyrazolo[1,5-a]pyridin-3-yl]methyl]pyridine-2-carboxylic acid
Show/Hide
|
C20H13Cl2N3O2
|
1
|
| 1 |
IC50 = 480 nM
|
|
|
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CP0566063
|
1-[(6-chloro-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C19H15ClN4O2
|
1
|
| 1 |
IC50 = 540 nM
|
|
|
|
CP0523134
|
1-[(5-acetyl-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C21H18N4O3
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0396387
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6-[[6-chloro-2-(2-chlorophenyl)pyrazolo[1,5-a]pyridin-3-yl]methyl]pyridine-2-carboxylic acid
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C20H13Cl2N3O2
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1
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| 1 |
IC50 = 640 nM
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CP0570334
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6-[(6-chloro-2-morpholin-4-ylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
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C18H17ClN4O3
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1
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| 1 |
IC50 = 740 nM
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CP0475914
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1-[(5-chloro-2-phenyl-1,3-benzoxazol-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
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C19H14ClN3O3
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1
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| 1 |
IC50 = 750 nM
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CP0570332
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6-[[6-chloro-2-(3-methoxyphenyl)pyrazolo[1,5-a]pyridin-3-yl]methyl]pyridine-2-carboxylic acid
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C21H16ClN3O3
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1
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| 1 |
IC50 = 800 nM
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CP0472710
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1-[[5-chloro-2-(2-methoxyphenyl)pyrazolo[1,5-a]pyridin-7-yl]methyl]-5-methylpyrazole-3-carboxylic acid
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C20H17ClN4O3
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1
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| 1 |
IC50 = 840 nM
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CP0432679
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1-[(5-cyano-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
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C20H15N5O2
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1
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| 1 |
IC50 = 1000 nM
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CP0510395
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1-[(4-methoxy-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
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C20H18N4O3
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1
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| 1 |
IC50 = 1100 nM
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CP0489172
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6-[[6-chloro-2-(4-chlorophenyl)pyrazolo[1,5-a]pyridin-3-yl]methyl]pyridine-2-carboxylic acid
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C20H13Cl2N3O2
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1
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| 1 |
IC50 = 1100 nM
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CP0494027
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6-[(6-acetyl-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
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C22H17N3O3
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1
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| 1 |
IC50 = 1100 nM
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CP0560507
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6-[(6-chloro-2-thiophen-2-ylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
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C18H12ClN3O2S
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1
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| 1 |
IC50 = 1100 nM
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CP0417767
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1-[(5-chloro-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-propan-2-ylpyrazole-3-carboxylic acid
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C21H19ClN4O2
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1
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| 1 |
IC50 = 1200 nM
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CP0481464
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6-[[6-chloro-2-(furan-2-yl)pyrazolo[1,5-a]pyridin-3-yl]methyl]pyridine-2-carboxylic acid
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C18H12ClN3O3
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1
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| 1 |
IC50 = 1200 nM
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CP0481465
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6-[(6-chloro-2-cyclohexylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
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C20H20ClN3O2
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1
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| 1 |
IC50 = 1200 nM
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CP0458614
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1-[[5-chloro-2-(2-methylpropyl)pyrazolo[1,5-a]pyridin-7-yl]methyl]-5-methylpyrazole-3-carboxylic acid
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C17H19ClN4O2
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1
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| 1 |
IC50 = 1400 nM
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CP0520483
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6-[[2-(azepan-1-yl)-6-chloropyrazolo[1,5-a]pyridin-3-yl]methyl]pyridine-2-carboxylic acid
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C20H21ClN4O2
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1
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| 1 |
IC50 = 1400 nM
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CP0461855
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1-[(6-methoxy-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
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C20H18N4O3
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1
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| 1 |
IC50 = 1500 nM
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CP0479675
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1-[[5-[(E)-hex-1-enyl]-2-phenylpyrazolo[1,5-a]pyridin-7-yl]methyl]-5-methylpyrazole-3-carboxylic acid
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C25H26N4O2
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1
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| 1 |
IC50 = 1500 nM
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CP0521213
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6-[(6-chloro-2-cyclopropylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
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C17H14ClN3O2
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1
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| 1 |
IC50 = 1500 nM
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CP0560509
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6-[(6-chloro-2-pyrrolidin-1-ylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
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C18H17ClN4O2
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1
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| 1 |
IC50 = 1800 nM
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CP0479673
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1-[(2-butyl-5-chloropyrazolo[1,5-a]pyridin-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
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C17H19ClN4O2
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1
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| 1 |
IC50 = 1900 nM
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CP0446921
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1-[(5-chloro-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-(2-methylpropyl)pyrazole-3-carboxylic acid
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C22H21ClN4O2
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1
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| 1 |
IC50 = 2000 nM
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CP0417768
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1-[(2-tert-butyl-5-chloropyrazolo[1,5-a]pyridin-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
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C17H19ClN4O2
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1
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| 1 |
IC50 = 2100 nM
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CP0523256
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6-[(2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
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C20H15N3O2
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1
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| 1 |
IC50 = 2300 nM
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CP0559180
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1-[[2-(3,6-dihydro-2H-pyridin-1-yl)-6-methyl-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
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C19H20N4O2S
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1
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| 1 |
IC50 = 2500 nM
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CP0432691
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1-[(4-chloro-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
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C19H15ClN4O2
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1
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| 1 |
IC50 = 2600 nM
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CP0571940
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1-[[6-chloro-2-(1,1-dioxo-1,4-thiazinan-4-yl)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
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C17H17ClN4O4S2
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1
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| 1 |
IC50 = 4200 nM
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CP0523260
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6-[(6-methoxy-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyrazine-2-carboxylic acid
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C20H16N4O3
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1
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| 1 |
IC50 = 4500 nM
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CP0566084
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1-[[6-chloro-2-(4-methylpiperazin-1-yl)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
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C18H20ClN5O2S
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1
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| 1 |
IC50 = 4900 nM
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CP0559182
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1-[[6-chloro-2-(4,5-dimethyl-3,6-dihydro-2H-pyridin-1-yl)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
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C20H21ClN4O2S
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1
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| 1 |
IC50 = 5200 nM
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CP0392336
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6-[(6-methylsulfonyl-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
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C21H17N3O4S
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1
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| 1 |
IC50 = 5400 nM
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CP0569198
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6-[[6-chloro-2-(4-methoxyphenyl)pyrazolo[1,5-a]pyridin-3-yl]methyl]pyridine-2-carboxylic acid
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C21H16ClN3O3
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1
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| 1 |
IC50 = 5400 nM
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CP0447003
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1-[[6-amino-2-(3,6-dihydro-2H-pyridin-1-yl)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
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C18H19N5O2S
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1
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| 1 |
IC50 = 7800 nM
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CP0534818
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4-[(3-carboxy-5-methylpyrazol-1-yl)methyl]-2-(3,6-dihydro-2H-pyridin-1-yl)-1,3-benzothiazole-6-carboxylic acid
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C19H18N4O4S
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1
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| 1 |
IC50 = 7900 nM
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CP0534666
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1-[(5-chloro-2-phenyl-1,3-benzothiazol-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
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C19H14ClN3O2S
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1
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| 1 |
IC50 = 7953 nM
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CP0389262
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1-[(6-chloro-2-phenyl-1,3-benzoxazol-4-yl)methyl]-5-methylpyrazole-3-carboxylic acid
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C19H14ClN3O3
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1
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| 1 |
IC50 = 8698 nM
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CP0519685
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1-[[2-(3,6-dihydro-2H-pyridin-1-yl)-6-(methylamino)-1,3-benzothiazol-4-yl]methyl]-5-methylpyrazole-3-carboxylic acid
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C19H21N5O2S
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1
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| 1 |
IC50 = 8800 nM
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CP0408381
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6-[(5-methoxy-2-phenylpyrazolo[1,5-a]pyridin-3-yl)methyl]pyridine-2-carboxylic acid
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C21H17N3O3
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1
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| 1 |
IC50 = 9100 nM
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CP0454783
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1-[(5-methoxy-2-phenylpyrazolo[1,5-a]pyridin-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
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C20H18N4O3
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1
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| 1 |
IC50 = 9600 nM
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