Brief Information of the Cell Line and Protein
Cell Line ID: CL000109 , COS-1
Synonyms
Cos-1
COS 1
Cos 1
COS1
Cos1
CV-1 in Origin Simian-1
Category Transformed cell line
Organism
Chlorocebus aethiops (Green monkey)
Cellosaurus ID
CVCL_0223
Protein ID: PT00915 , Peroxisome proliferator-activated receptor gamma
Gene Name PPARG
Organism Homo sapiens, Human
Protein Classification Transcription factor
Uniprot ID P37231
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000109  Protein ID: PT00915
 
Compound ID Compound Name Compound Formula
CP0407555
(S)-2-(3-((3-(4-methoxybenzoyl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl)methyl)phenoxy)propanoic acid
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C28H24F3NO6
 1
1
EC50 = 1 nM
   TI
   LI
   LO
   TS
CP0259373
(2S)-2-[3-[[3-(4-Chlorobenzoyl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl]methyl]phenoxy]propanoicAcid
   Show/Hide
C27H21ClF3NO5
 1
1
EC50 = 1 nM
   TI
   LI
   LO
   TS
CP0282604
(2S)-2-{3-[[3-(4-Chlorobenzoyl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl]methyl]phenoxy}pentanoic Acid
   Show/Hide
C29H25ClF3NO5
 1
1
EC50 = 1 nM
   TI
   LI
   LO
   TS
CP0208054
2-Methyl-2-{4-[4-(3-phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-butoxy]-phenoxy}-propionic acid
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C30H33NO6
 1
1
EC50 = 2 nM
   TI
   LI
   LO
   TS
CP0048507
(2S)-2-(3-{[1-(4-METHOXYBENZOYL)-2-METHYL-5-(TRIFLUOROMETHOXY)-1H-INDOL-3-YL]METHYL}PHENOXY)PROPANOIC ACID
   Show/Hide
C28H24F3NO6
 1
1
EC50 = 2 nM
   TI
   LI
   LO
   TS
CP0422144
(R)-2-(3-(3-(4-methoxybenzoyl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl)phenoxy)butanoic acid
   Show/Hide
C28H24F3NO6
 1
1
EC50 = 2 nM
   TI
   LI
   LO
   TS
CP0045050
(R)-2-{3-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluoromethoxy-1H-indol-3-ylmethyl]-phenoxy}-propionic acid
   Show/Hide
C28H24F3NO6
 1
1
EC50 = 2 nM
   TI
   LI
   LO
   TS
CP0045059
2-{3-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluoromethoxy-1H-indol-3-ylmethyl]-phenoxy}-pentanoic acid
   Show/Hide
C30H28F3NO6
 1
1
EC50 = 2 nM
   TI
   LI
   LO
   TS
CP0083609
2-{3-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluoromethoxy-1H-indol-3-ylmethyl]-phenoxy}-propionic acid
   Show/Hide
C28H24F3NO6
 1
1
EC50 = 2 nM
   TI
   LI
   LO
   TS
CP0149811
(2S)-2-(2-{[1-(4-METHOXYBENZOYL)-2-METHYL-5-(TRIFLUOROMETHOXY)-1H-INDOL-3-YL]METHYL}PHENOXY)PROPANOIC ACID
   Show/Hide
C28H24F3NO6
 1
1
EC50 = 2 nM
   TI
   LI
   LO
   TS
CP0043911
(2R)-2-{3-[[3-(4-Chlorobenzoyl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl]methyl]phenoxy}butanoic Acid
   Show/Hide
C28H23ClF3NO5
 1
1
EC50 = 2 nM
   TI
   LI
   LO
   TS
CP0174902
(2R)-2-{3-[[3-(4-Chlorobenzoyl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl]methyl]phenoxy}isobutyric Acid
   Show/Hide
C29H25ClF3NO5
 1
1
EC50 = 2 nM
   TI
   LI
   LO
   TS
CP0293294
(+)-2-{3-[[3-(4-Chlorobenzoyl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl]methyl]phenoxy}-2-methylbutanoic Acid
   Show/Hide
C29H25ClF3NO5
 1
1
EC50 = 2 nM
   TI
   LI
   LO
   TS
CP0293295
2-[3-[[3-(4-Chlorobenzoyl)-2-methyl-6-(trifluoromethoxy)-1Hindol-1-yl]methyl]phenoxy]acetic Acid
   Show/Hide
C26H19ClF3NO5
 1
1
EC50 = 2 nM
   TI
   LI
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   TS
CP0077514
(2S)-2-(4-chloro-3-(1-(6-chlorobenzo[d]isoxazol-3-yl)-2-methyl-5-(trifluoromethoxy)-1H-indol-3-yloxy)phenoxy)propanoic acid
   Show/Hide
C26H17Cl2F3N2O6
 1
1
EC50 = 3 nM
   TI
   LI
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   TS
CP0374380
(2S)-2-(4-chloro-3-((3-(6-methoxybenzo[d]isoxazol-3-yl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl)methyl)phenoxy)propanoic acid
   Show/Hide
C28H22ClF3N2O6
 1
1
EC50 = 3 nM
   TI
   LI
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   TS
CP0505050
(S)-2-(2-chloro-5-((3-(4-chlorophenoxy)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl)methyl)phenoxy)propanoic acid
   Show/Hide
C26H20Cl2F3NO5
 1
1
EC50 = 3 nM
   TI
   LI
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   TS
CP0051869
2-{3-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluoromethoxy-1H-indol-3-ylmethyl]-phenoxy}-butyric acid
   Show/Hide
C29H26F3NO6
 1
1
EC50 = 3 nM
   TI
   LI
   LO
   TS
CP0083607
2-{2-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluoromethoxy-1H-indol-3-ylmethyl]-phenoxy}-propionic acid
   Show/Hide
C28H24F3NO6
 1
1
EC50 = 3 nM
   TI
   LI
   LO
   TS
CP0316148
2-(3-((1-(4-chlorobenzoyl)-2-methyl-5-(trifluoromethoxy)-1H-indol-3-yl)methyl)phenoxy)acetic acid
   Show/Hide
C26H19ClF3NO5
 1
1
EC50 = 3 nM
   TI
   LI
   LO
   TS
CP0130403
2-[3-chloro-4-[3-[(3-phenyl-7-propyl-1,2-benzoxazol-6-yl)oxy]propylsulfanyl]phenyl]acetic acid
   Show/Hide
C27H26ClNO4S
 1
1
EC50 = 4 nM
   TI
   LI
   LO
   TS
CP0070863
(2R)-2-[3-[[3-(4-Chlorobenzoyl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl]methyl]phenoxy]propanoicAcid
   Show/Hide
C27H21ClF3NO5
 1
1
EC50 = 4 nM
   TI
   LI
   LO
   TS
CP0274733
(2R)-2-[2-chloro-5-[[3-(7-methyl-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
   Show/Hide
C26H19ClF3N3O5
 1
1
EC50 = 4.1 nM
   TI
   LI
   LO
   TS
CP0155637
(3-{4-[(3-phenyl-7-propyl-1,2-benzisoxazol-6-yl)oxy]butoxy}phenyl)acetic acid
   Show/Hide
C28H29NO5
 1
1
EC50 = 6 nM
   TI
   LI
   LO
   TS
CP0045061
2-{3-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluoromethoxy-1H-indol-3-ylmethyl]-phenoxy}-2-methyl-propionic acid
   Show/Hide
C29H26F3NO6
 1
1
EC50 = 6 nM
   TI
   LI
   LO
   TS
CP0333136
2-{2-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluoromethoxy-1H-indol-3-ylmethyl]-phenoxy}-butyric acid
   Show/Hide
C29H26F3NO6
 1
1
EC50 = 6 nM
   TI
   LI
   LO
   TS
CP0048728
(2S)-2-{3-[[3-(4-Chlorobenzoyl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl]methyl]phenoxy}butanoic Acid
   Show/Hide
C28H23ClF3NO5
 1
1
EC50 = 6 nM
   TI
   LI
   LO
   TS
CP0077172
(5R)-5-[4-chloro-3-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxobenzimidazol-1-yl]methyl]phenyl]-5-methyl-1,3-oxazolidine-2,4-dione
   Show/Hide
C26H19ClN4O6
 1
1
EC50 = 9.1 nM
   TI
   LI
   LO
   TS
CP0207654
2-Methyl-2-{4-[4-(3-phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-butoxy]-phenyl}-propionic acid
   Show/Hide
C30H33NO5
 1
1
EC50 = 10 nM
   TI
   LI
   LO
   TS
CP0108857
(2R)-2-{3-[[3-(4-Chlorobenzoyl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl]methyl]phenoxy}pentanoic Acid
   Show/Hide
C29H25ClF3NO5
 1
1
EC50 = 10 nM
   TI
   LI
   LO
   TS
CP0130444
(2R)-2-[2-chloro-5-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethoxy)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
   Show/Hide
C26H19ClF3N3O7
 1
1
EC50 = 11.4 nM
   TI
   LI
   LO
   TS
CP0280959
2-{2-[1-(4-Chloro-benzoyl)-5-methoxy-2-methyl-1H-indol-3-ylmethyl]-phenoxy}-2-methyl-propionic acid
   Show/Hide
C28H26ClNO5
 1
1
EC50 = 12 nM
   TI
   LI
   LO
   TS
CP0174901
1-{3-[[3-(4-Chlorobenzoyl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl]methyl]phenoxy}-1-cyclobutanecarboxylic Acid
   Show/Hide
C29H23ClF3NO5
 1
1
EC50 = 12 nM
   TI
   LI
   LO
   TS
CP0130445
(2R)-2-[2-chloro-5-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxo-5-(trifluoromethoxy)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
   Show/Hide
C26H19ClF3N3O7
 1
1
EC50 = 13.2 nM
   TI
   LI
   LO
   TS
CP0651087
5-(3-(3-(4-phenoxy-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione
   Show/Hide
C27H27NO5S
 1
1
EC50 = 14 nM
   TI
   LI
   LO
   TS
CP0464471
2-{2-[1-(4-Chloro-benzoyl)-5-methoxy-2-methyl-1H-indol-3-ylmethyl]-phenoxy}-propionic acid
   Show/Hide
C27H24ClNO5
 1
1
EC50 = 14 nM
   TI
   LI
   LO
   TS
CP0101367
2-{4-[4-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-butoxy]-phenoxy}-propionic acid
   Show/Hide
C29H31NO6
 1
1
EC50 = 16 nM
   TI
   LI
   LO
   TS
CP0077171
(5R)-5-[4-chloro-3-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenyl]-5-methyl-1,3-oxazolidine-2,4-dione
   Show/Hide
C27H18ClF3N4O6
 1
1
EC50 = 17 nM
   TI
   LI
   LO
   TS
CP0080155
2-{3-[1-(4-Chloro-benzoyl)-5-methoxy-2-methyl-1H-indol-3-ylmethyl]-phenoxy}-2-methyl-propionic acid
   Show/Hide
C28H26ClNO5
 1
1
EC50 = 19 nM
   TI
   LI
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   TS
CP0334496
2-{3-[1-(4-Chloro-benzoyl)-5-methoxy-2-methyl-1H-indol-3-ylmethyl]-phenoxy}-propionic acid
   Show/Hide
C27H24ClNO5
 1
1
EC50 = 19 nM
   TI
   LI
   LO
   TS
CP0005387
Avandamet
   Show/Hide
C18H19N3O3S
 6
1
EC50 = 20 nM
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   LI
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   TS
2
EC50 = 21 nM
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3
EC50 = 23 nM
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4
EC50 = 48 nM
   TI
   LI
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5
EC50 = 120 nM
   TI
   LI
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   TS
6
EC50 = 200 nM
   TI
   LI
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   TS
CP0679717
5-(4-(3-(4-(biphenyl-4-yloxy)-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione
   Show/Hide
C33H31NO5S
 1
1
EC50 = 20 nM
   TI
   LI
   LO
   TS
CP0178891
2,2-Dimethyl-3-{4-[4-(3-phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-butoxy]-phenyl}-propionic acid
   Show/Hide
C31H35NO5
 1
1
EC50 = 20 nM
   TI
   LI
   LO
   TS
CP0677691
(S)-7-(2-{2-[(1E)-1,5-Dimethylhexen-1-yl]-5-methyloxazol-4-yl}ethoxy)-2-[(2E,4E)-hexadienoyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C34H49N3O5
 1
1
EC50 = 20 nM
   TI
   LI
   LO
   TS
CP0704227
(S)-2-Hexanoyl-7-(2-{5-methyl-2-[(1E)-5-methylhexen-1-yl]oxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C33H51N3O5
 1
1
EC50 = 20 nM
   TI
   LI
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   TS
CP0715179
(S)-2-[(2E)-3-Ethoxyacryloyl]-7-(2-{5-methyl-2-[(1E)-5-methylhexen-1-yl]oxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C32H47N3O6
 1
1
EC50 = 20 nM
   TI
   LI
   LO
   TS
CP0290029
(R)-2-{2-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluoromethoxy-1H-indol-3-ylmethyl]-phenoxy}-propionic acid
   Show/Hide
C28H24F3NO6
 1
1
EC50 = 21 nM
   TI
   LI
   LO
   TS
CP0108856
(2S)-2-{3-[[3-(4-Chlorobenzoyl)-2-methyl-6-(trifluoromethoxy)-1H-indol-1-yl]methyl]phenoxy}isobutyric Acid
   Show/Hide
C29H25ClF3NO5
 1
1
EC50 = 21 nM
   TI
   LI
   LO
   TS
CP0661032
5-(3-{3-[4-(4-Hydroxy-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione
   Show/Hide
C27H27NO6S
 1
1
EC50 = 23 nM
   TI
   LI
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   TS
CP0654731
5-(3-{3-[4-(4-Chloro-3-methyl-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione
   Show/Hide
C28H28ClNO5S
 1
1
EC50 = 27 nM
   TI
   LI
   LO
   TS
CP0078110
2-{4-[3-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-propoxy]-phenoxy}-propionic acid
   Show/Hide
C28H29NO6
 1
1
EC50 = 27 nM
   TI
   LI
   LO
   TS
CP0191197
(2R)-2-[2-chloro-5-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxobenzimidazol-1-yl]methyl]phenoxy]propanoic acid
   Show/Hide
C25H20ClN3O6
 1
1
EC50 = 28.1 nM
   TI
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CP0100328
(E)-3-{4-[4-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-butoxy]-phenyl}-acrylic acid
   Show/Hide
C29H29NO5
 1
1
EC50 = 29 nM
   TI
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   TS
CP0658355
5-(4-(3-(4-(4-methoxyphenoxy)-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione
   Show/Hide
C28H29NO6S
 1
1
EC50 = 30 nM
   TI
   LI
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   TS
CP0705705
5-(4-(3-(4-(4-isobutylphenoxy)-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione
   Show/Hide
C31H35NO5S
 1
1
EC50 = 30 nM
   TI
   LI
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   TS
CP0715178
(S)-2-[(2E,4E)-Hexadienoyl]-7-[2-{5-methyl-2-[(1E)-5-methylhexen-1-yl]oxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C33H47N3O5
 1
1
EC50 = 30 nM
   TI
   LI
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   TS
CP0778408
(S)-2-[(2E)-Hexenoyl]-7-(2-{5-methyl-2-[(1E)-5-methylhexen-1-yl]oxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C33H49N3O5
 1
1
EC50 = 30 nM
   TI
   LI
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   TS
CP0786452
(S)-2-[(2E,4E)-5-Methylhexadienoyl]-7-(2-{5-methyl-2-[(1E)-5-methylhexen-1-yl]oxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C34H49N3O5
 1
1
EC50 = 30 nM
   TI
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   TS
CP0088604
3-Methyl-3-{4-[4-(3-phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-butoxy]-phenyl}-butyric acid
   Show/Hide
C31H35NO5
 1
1
EC50 = 37 nM
   TI
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   TS
CP0726657
(S)-7-(2-{5-Methyl-2-[(1E)-5-methylhexen-1-yl]oxazol-4-yl}ethoxy)-2-[(2E)-3-(thiophen-2-yl)acryloyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C34H45N3O5S
 1
1
EC50 = 40 nM
   TI
   LI
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   TS
CP0738191
(S)-7-(2-{5-Methyl-2-[(1E)-5-methylhexen-1-yl]oxazol-4-yl}ethoxy)-2-(4-pentenoyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C32H47N3O5
 1
1
EC50 = 40 nM
   TI
   LI
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   TS
CP0708518
5-(3-(3-(4-(3,4-dichlorophenoxy)-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione
   Show/Hide
C27H25Cl2NO5S
 1
1
EC50 = 47 nM
   TI
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   TS
CP0152777
2-{2-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluoromethoxy-1H-indol-3-ylmethyl]-phenoxy}-2-methyl-propionic acid
   Show/Hide
C29H26F3NO6
 1
1
EC50 = 50 nM
   TI
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   TS
CP0704226
(S)-2-(5-Hexenoyl)-7-(2-{5-methyl-2-[(1E)-5-methylhexen-1-yl]oxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C33H49N3O5
 1
1
EC50 = 50 nM
   TI
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   TS
CP0778409
(S)-2-[(2E,4E)-2-Methylhexadienoyl]-7-(2-{5-methyl-2-[(1E)-5-methylhexen-1-yl]oxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C34H49N3O5
 1
1
EC50 = 50 nM
   TI
   LI
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   TS
CP0163263
(2R)-2-[4-chloro-3-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxobenzimidazol-1-yl]methyl]phenoxy]propanoic acid
   Show/Hide
C25H20ClN3O6
 1
1
EC50 = 51.1 nM
   TI
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CP0257979
2-Methyl-2-{3-[4-(3-phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-butoxy]-phenyl}-propionic acid
   Show/Hide
C30H33NO5
 1
1
EC50 = 52 nM
   TI
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   TS
CP0645378
5-(4-(3-(4-(4-fluorophenoxy)-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione
   Show/Hide
C27H26FNO5S
 2
1
EC50 = 60 nM
   TI
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2
EC50 = 80 nM
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CP0208053
2-[4-[4-[(3-phenyl-7-propyl-1,2-benzoxazol-6-yl)oxy]butoxy]phenyl]acetic acid
   Show/Hide
C28H29NO5
 1
1
EC50 = 60 nM
   TI
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   TS
CP0654439
5-(3-{3-[4-(4-Methoxy-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione
   Show/Hide
C28H29NO6S
 1
1
EC50 = 69 nM
   TI
   LI
   LO
   TS
CP0738901
(S)-2-(3-Cyclopropylacryloyl)-7-(2-{5-methyl-2-[(1E)-5-methylhexen-1-yl]oxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C33H47N3O5
 1
1
EC50 = 70 nM
   TI
   LI
   LO
   TS
CP0792212
(S)-2-(3-Ethoxypropionyl)-7-(2-{5-methyl-2-[(1E)-5-methylhexen-1-yl]oxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C32H49N3O6
 1
1
EC50 = 70 nM
   TI
   LI
   LO
   TS
CP0834401
(S)-2-[(2E)-3-(Furan-2-yl)acryloyl]-7-(2-{5-methyl-2-[(1E)-5-methylhexen-1-yl]oxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C34H45N3O6
 1
1
EC50 = 70 nM
   TI
   LI
   LO
   TS
CP0220490
2-[4-[3-[(3-phenyl-7-propyl-1,2-benzoxazol-6-yl)oxy]propoxy]phenoxy]acetic acid
   Show/Hide
C27H27NO6
 1
1
EC50 = 75 nM
   TI
   LI
   LO
   TS
CP0334535
2-[3-[[1-(4-chlorobenzoyl)-5-methoxy-2-methylindol-3-yl]methyl]phenoxy]acetic acid
   Show/Hide
C26H22ClNO5
 1
1
EC50 = 77 nM
   TI
   LI
   LO
   TS
CP0166787
(2R)-2-[2-chloro-5-[[3-(6-methyl-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
   Show/Hide
C26H19ClF3N3O5
 1
1
EC50 = 77.5 nM
   TI
   LI
   LO
   TS
CP0672440
5-(4-(3-(4-(4-chlorophenoxy)-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione
   Show/Hide
C27H26ClNO5S
 1
1
EC50 = 80 nM
   TI
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   LO
   TS
CP0166789
(2R)-2-[2-chloro-5-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxo-5-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
   Show/Hide
C26H19ClF3N3O6
 1
1
EC50 = 83 nM
   TI
   LI
   LO
   TS
CP0646515
5-(3-{3-[4-(4-Fluoro-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione
   Show/Hide
C27H26FNO5S
 1
1
EC50 = 85 nM
   TI
   LI
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   TS
CP0036283
2-[3-[4-[(3-phenyl-7-propyl-1,2-benzoxazol-6-yl)oxy]butoxy]phenoxy]acetic acid
   Show/Hide
C28H29NO6
 1
1
EC50 = 87 nM
   TI
   LI
   LO
   TS
CP0715180
(S)-2-[(2E)-4-Ethoxybutenoyl]-7-(2-{5-methyl-2-[(1E)-5-methylhexen-1-yl]oxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C33H49N3O6
 1
1
EC50 = 90 nM
   TI
   LI
   LO
   TS
CP0680900
5-(3-methyl-4-(3-(4-phenoxy-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione
   Show/Hide
C28H29NO5S
 1
1
EC50 = 100 nM
   TI
   LI
   LO
   TS
CP0220876
2-Methyl-2-{3-[4-(3-phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-butoxy]-phenoxy}-propionic acid
   Show/Hide
C30H33NO6
 1
1
EC50 = 100 nM
   TI
   LI
   LO
   TS
CP0191195
(2R)-2-[4-chloro-3-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
   Show/Hide
C26H19ClF3N3O6
 1
1
EC50 = 102 nM
   TI
   LI
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   TS
CP0308909
(5R)-5-[3-[[3-(6-chloro-1,2-benzoxazol-3-yl)-2-oxobenzimidazol-1-yl]methyl]phenyl]-5-methyl-1,3-oxazolidine-2,4-dione
   Show/Hide
C25H17ClN4O5
 1
1
EC50 = 102 nM
   TI
   LI
   LO
   TS
CP0152328
(2R)-2-[2-chloro-5-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
   Show/Hide
C26H19ClF3N3O6
 1
1
EC50 = 103 nM
   TI
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   TS
CP0672411
5-(3-{3-[4-(4-Fluoro-3-methyl-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione
   Show/Hide
C28H28FNO5S
 1
1
EC50 = 106 nM
   TI
   LI
   LO
   TS
CP0756803
(S)-2-[(2E,4E)-Hexadienoyl]-7-{2-[5-methyl-2-(5-methylhexyl)oxazol-4-yl]ethoxy}-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C33H49N3O5
 1
1
EC50 = 110 nM
   TI
   LI
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   TS
CP0761841
5-(4-(3-(4-(4-(methylsulfonyl)phenoxy)-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione
   Show/Hide
C28H29NO7S2
 1
1
EC50 = 120 nM
   TI
   LI
   LO
   TS
CP0667009
(S)-2-[(2E,4E)-Hexadienoyl]-7-(2-{5-methyl-2-[(1E)-1-methylbuten-1-yl]oxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C31H43N3O5
 1
1
EC50 = 120 nM
   TI
   LI
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   TS
CP0130443
(2R)-2-[2-chloro-5-[[3-(5-chloro-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
   Show/Hide
C25H16Cl2F3N3O5
 1
1
EC50 = 120 nM
   TI
   LI
   LO
   TS
CP0672145
5-(3-{3-[4-(4-Cyclopentyl-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione
   Show/Hide
C32H35NO5S
 1
1
EC50 = 123 nM
   TI
   LI
   LO
   TS
CP0131874
(2R)-2-[5-[[3-(4-tert-butylphenyl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]-2-chlorophenoxy]propanoic acid
   Show/Hide
C28H26ClF3N2O4
 1
1
EC50 = 135 nM
   TI
   LI
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   TS
CP0324132
4-{4-[3-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-propoxy]-phenyl}-butyric acid
   Show/Hide
C29H31NO5
 1
1
EC50 = 156 nM
   TI
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   TS
CP0787014
(S)-2-[(2E,4E)-Hexadienoyl]-7-(2-{5-methyl-2-{[(1E)-4-methylpenten-1-yl]oxazol-4-yl}ethoxy-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C32H45N3O5
 1
1
EC50 = 160 nM
   TI
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   TS
CP0808196
(S)-7-(2-{2-[(1E)-4,4-Dimethylpenten-1-yl]-5-methyloxazol-4-yl}ethoxy)-2-[(2E,4E)-hexadienoyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C33H47N3O5
 1
1
EC50 = 160 nM
   TI
   LI
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   TS
CP0686397
5-(3-{3-[4-(4-Chloro-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione
   Show/Hide
C27H26ClNO5S
 1
1
EC50 = 165 nM
   TI
   LI
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   TS
CP0782507
5-(3-{3-[4-(4-Isopropyl-phenoxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione
   Show/Hide
C30H33NO5S
 1
1
EC50 = 167 nM
   TI
   LI
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   TS
CP0038450
(R)-7-{3-[2-Chloro-4-(4-fluoro-phenoxy)-phenoxy]-propoxy}-2-ethyl-chroman-2-carboxylic acid
   Show/Hide
C27H26ClFO6
 1
1
EC50 = 170 nM
   TI
   LI
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   TS
CP0430218
2-[2-[[1-(4-chlorobenzoyl)-5-methoxy-2-methylindol-3-yl]methyl]phenoxy]acetic acid
   Show/Hide
C26H22ClNO5
 1
1
EC50 = 191 nM
   TI
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   TS
CP0208071
3-[4-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-butoxy]-benzoic acid
   Show/Hide
C27H27NO5
 1
1
EC50 = 193 nM
   TI
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   TS
CP0213824
2-(4-(3-(3-phenyl-7-propylbenzo[d]isoxazol-6-yloxy)propoxy)phenyl)acetic acid
   Show/Hide
C27H27NO5
 1
1
EC50 = 194 nM
   TI
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   TS
CP0734398
5-(4-(3-(4-phenoxy-2-propylphenoxy)propoxy)-3-propylphenyl)thiazolidine-2,4-dione
   Show/Hide
C30H33NO5S
 1
1
EC50 = 200 nM
   TI
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   TS
CP0308908
(2R)-2-[2-chloro-5-[[3-(6-chloro-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
   Show/Hide
C25H16Cl2F3N3O5
 1
1
EC50 = 200 nM
   TI
   LI
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   TS
CP0282728
(5R)-5-[3-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenyl]-5-methyl-1,3-oxazolidine-2,4-dione
   Show/Hide
C27H19F3N4O6
 1
1
EC50 = 237 nM
   TI
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   TS
CP0180190
(R)-7-{3-[2-Chloro-4-(4-fluoro-phenoxy)-phenoxy]-propoxy}-2-methyl-chroman-2-carboxylic acid
   Show/Hide
C26H24ClFO6
 1
1
EC50 = 240 nM
   TI
   LI
   LO
   TS
CP0761576
(S)-2-[(2E)-4-Hydroxyhexenoyl]-7-(2-{5-methyl-2-[(1E)-5-methylhexen-1-yl]oxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C33H49N3O6
 1
1
EC50 = 240 nM
   TI
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   TS
CP0036288
(E)-3-{4-[3-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-propoxy]-phenyl}-acrylic acid
   Show/Hide
C28H27NO5
 1
1
EC50 = 254 nM
   TI
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   TS
CP0051952
3-[1-(4-Chloro-benzoyl)-5-methoxy-2-methyl-1H-indol-3-ylmethyl]-benzoic acid
   Show/Hide
C25H20ClNO4
 1
1
EC50 = 280 nM
   TI
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   TS
CP0654730
5-(4-(3-(4-phenoxy-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione
   Show/Hide
C27H27NO5S
 1
1
EC50 = 300 nM
   TI
   LI
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   TS
CP0761598
5-(4-(4-(4-phenoxy-2-propylphenoxy)butoxy)phenyl)thiazolidine-2,4-dione
   Show/Hide
C28H29NO5S
 1
1
EC50 = 300 nM
   TI
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   TS
CP0783387
5-(3-fluoro-4-(3-(4-phenoxy-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione
   Show/Hide
C27H26FNO5S
 1
1
EC50 = 300 nM
   TI
   LI
   LO
   TS
CP0761577
(S)-2-[(2E,4E)-Hexadienoyl]-7-(2-{5-methyl-2-[(1E)-3-methylhexen-1-yl]oxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C33H47N3O5
 1
1
EC50 = 310 nM
   TI
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   TS
CP0677693
(S)-7-(2-{2-[(1E)-1-Ethylpropen-1-yl]-5-methyloxazol-4-yl}ethoxy)-2-[(2E,4E)-hexadienoyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C31H43N3O5
 1
1
EC50 = 350 nM
   TI
   LI
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   TS
CP0727828
5-(3-{3-[4-(Biphenyl-4-yloxy)-2-propyl-phenoxy]-propoxy}-phenyl)-thiazolidine-2,4-dione
   Show/Hide
C33H31NO5S
 1
1
EC50 = 353 nM
   TI
   LI
   LO
   TS
CP0126336
(5R)-5-[3-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxobenzimidazol-1-yl]methyl]phenyl]-5-methyl-1,3-oxazolidine-2,4-dione
   Show/Hide
C26H20N4O6
 1
1
EC50 = 360 nM
   TI
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CP0041219
Actos
   Show/Hide
C19H20N2O3S
 1
1
EC50 = 390 nM
   TI
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   TS
CP0677669
5-(3-methoxy-4-(3-(4-phenoxy-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione
   Show/Hide
C28H29NO6S
 1
1
EC50 = 400 nM
   TI
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   TS
CP0111376
(R)-7-[3-(2-Chloro-4-cyclohexyl-phenoxy)-propoxy]-2-ethyl-chroman-2-carboxylic acid
   Show/Hide
C27H33ClO5
 1
1
EC50 = 400 nM
   TI
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   TS
CP0160927
(R)-7-{3-[2-Chloro-4-(2,2,2-trifluoro-ethoxy)-phenoxy]-propoxy}-2-ethyl-chroman-2-carboxylic acid
   Show/Hide
C23H24ClF3O6
 1
1
EC50 = 400 nM
   TI
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   TS
CP0186194
3-{4-[4-(3-Phenyl-7-propyl-benzo[d]isoxazol-6-yloxy)-butoxy]-phenyl}-propionic acid
   Show/Hide
C29H31NO5
 1
1
EC50 = 485 nM
   TI
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   TS
CP0166785
(2R)-2-[2-chloro-5-[[3-(4-chlorobenzoyl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
   Show/Hide
C25H17Cl2F3N2O5
 1
1
EC50 = 489 nM
   TI
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   TS
CP0716559
N-(4-(4-(3-(4-(2,4-dioxothiazolidin-5-yl)phenoxy)propoxy)-3-propylphenoxy)phenyl)-4-methylbenzenesulfonamide
   Show/Hide
C34H34N2O7S2
 1
1
EC50 = 500 nM
   TI
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CP0046923
(R)-7-[3-(2-Chloro-4-trifluoromethoxy-phenoxy)-propoxy]-2-ethyl-chroman-2-carboxylic acid
   Show/Hide
C22H22ClF3O6
 1
1
EC50 = 500 nM
   TI
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   TS
CP0051867
(R)-7-[3-(2-Chloro-4-isobutyl-phenoxy)-propoxy]-2-methyl-chroman-2-carboxylic acid
   Show/Hide
C24H29ClO5
 1
1
EC50 = 500 nM
   TI
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   TS
CP0083171
(R)-7-[3-(2-Chloro-4-spiro[2.5]oct-6-yl-phenoxy)-propoxy]-2-ethyl-chroman-2-carboxylic acid
   Show/Hide
C29H35ClO5
 1
1
EC50 = 500 nM
   TI
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   TS
CP0677692
(S)-2-[(2E,4E)]-Hexadienoyl]-7-(2-{2-[(1E)-3,3-dimethylbuten-1-yl]-5-methyloxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C32H45N3O5
 1
1
EC50 = 540 nM
   TI
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   TS
CP0080418
(R)-7-[3-(2-Chloro-4-isobutyl-phenoxy)-propoxy]-2-ethyl-chroman-2-carboxylic acid
   Show/Hide
C25H31ClO5
 1
1
EC50 = 600 nM
   TI
   LI
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   TS
CP0778411
(S)-2-[(2E,4E)-Hexadienoyl]-7-(5-methyl-2-{2-[(1E)-3-methylbuten-1-yl]oxazol-4-yl}ethoxy)-1,2,3,4-tetrahydroisoqunoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C31H43N3O5
 1
1
EC50 = 670 nM
   TI
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   TS
CP0684997
5-(3-chloro-4-(3-(4-phenoxy-2-propylphenoxy)propoxy)phenyl)thiazolidine-2,4-dione
   Show/Hide
C27H26ClNO5S
 1
1
EC50 = 700 nM
   TI
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   TS
CP0045073
(R)-7-[3-(2-Chloro-4-cyclohexyl-phenoxy)-propoxy]-2-methyl-chroman-2-carboxylic acid
   Show/Hide
C26H31ClO5
 1
1
EC50 = 700 nM
   TI
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   TS
CP0184722
(R)-7-[3-(2-Chloro-4-cyclobutylmethoxy-phenoxy)-propoxy]-2-methyl-chroman-2-carboxylic acid
   Show/Hide
C25H29ClO6
 1
1
EC50 = 700 nM
   TI
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   TS
CP0334515
(R)-7-[3-(2-Chloro-4-cyclopentyl-phenoxy)-propoxy]-2-methyl-chroman-2-carboxylic acid
   Show/Hide
C25H29ClO5
 1
1
EC50 = 700 nM
   TI
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   TS
CP0761578
(S)-7-(2-{2-[(1E)-3,3-Dimethylpenten-1-yl]-5-methyloxazol-4-yl}ethoxy)-2-[(2E,4E)-hexadienoyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C33H47N3O5
 1
1
EC50 = 760 nM
   TI
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   TS
CP0778410
(S)-7-(2-{2-[(1E)-3-Ethylpenten-1-yl]-5-methyloxazol-4-yl}ethoxy)-2-[(2E,4E)-hexadienoyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid tert-butylamine salt
   Show/Hide
C33H47N3O5
 1
1
EC50 = 760 nM
   TI
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   TS
CP0039118
2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)sulfanyl]phenoxy}acetic acid
   Show/Hide
C21H18F3NO3S2
 1
1
EC50 = 912 nM
   TI
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   TS
CP0040986
(R)-7-[3-(2,4-Dichloro-phenoxy)-propoxy]-2-ethyl-chroman-2-carboxylic acid
   Show/Hide
C21H22Cl2O5
 1
1
EC50 = 1000 nM
   TI
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   TS
CP0048558
(R)-7-[3-(2-Chloro-4-trifluoromethyl-phenoxy)-propoxy]-2-ethyl-chroman-2-carboxylic acid
   Show/Hide
C22H22ClF3O5
 1
1
EC50 = 1000 nM
   TI
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   TS
CP0082083
(R)-7-[3-(2-Chloro-4-spiro[2.5]oct-6-yl-phenoxy)-propoxy]-2-methyl-chroman-2-carboxylic acid
   Show/Hide
C28H33ClO5
 1
1
EC50 = 1000 nM
   TI
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   TS
CP0149897
(R)-7-{3-[2-Chloro-4-(4,4-dimethyl-cyclohexyl)-phenoxy]-propoxy}-2-methyl-chroman-2-carboxylic acid
   Show/Hide
C28H35ClO5
 1
1
EC50 = 1000 nM
   TI
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   TS
CP0152968
(R)-7-[3-(4-tert-Butyl-2-chloro-phenoxy)-propoxy]-2-ethyl-chroman-2-carboxylic acid
   Show/Hide
C25H31ClO5
 1
1
EC50 = 1000 nM
   TI
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   TS
CP0152971
(R)-7-[3-(2-Chloro-4-isopropyl-phenoxy)-propoxy]-2-ethyl-chroman-2-carboxylic acid
   Show/Hide
C24H29ClO5
 1
1
EC50 = 1200 nM
   TI
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   TS
CP0380855
2-(3-(3-(2-(4-methylbenzoyl)-1H-pyrrol-1-yl)prop-1-enyl)phenoxy)acetic acid
   Show/Hide
C23H21NO4
 1
1
EC50 = 1200 nM
   TI
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CP0080583
(R)-7-{3-[2-Chloro-4-(4,4-dimethyl-cyclohexyl)-phenoxy]-propoxy}-2-ethyl-chroman-2-carboxylic acid
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C29H37ClO5
 1
1
EC50 = 1400 nM
   TI
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   TS
CP0412240
2-(3-(3-(2-(4-methoxybenzoyl)-1H-pyrrol-1-yl)prop-1-enyl)phenoxy)acetic acid
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C23H21NO5
 1
1
EC50 = 1900 nM
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CP0412238
2-(3-(3-(2-(4-methoxybenzoyl)-1H-pyrrol-1-yl)prop-1-enyl)phenyl)acetic acid
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C23H21NO4
 1
1
EC50 = 2000 nM
   TI
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CP0080381
(R)-7-{3-[2-Chloro-4-(2,2,2-trifluoro-ethoxy)-phenoxy]-propoxy}-2-methyl-chroman-2-carboxylic acid
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C22H22ClF3O6
 1
1
EC50 = 3000 nM
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CP0080420
(R)-7-[3-(2-Chloro-4-fluoro-phenoxy)-propoxy]-2-ethyl-chroman-2-carboxylic acid
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C21H22ClFO5
 1
1
EC50 = 3000 nM
   TI
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   TS
CP0277228
7-{3-[2-Chloro-4-(2,2,2-trifluoro-ethoxy)-phenoxy]-propoxy}-chroman-2-carboxylic acid
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C21H20ClF3O6
 1
1
EC50 = 3000 nM
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CP0281023
(R)-7-[3-(2-Chloro-4-isopropyl-phenoxy)-propoxy]-2-methyl-chroman-2-carboxylic acid
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C23H27ClO5
 1
1
EC50 = 3000 nM
   TI
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CP0071331
(2S)-2-[2-chloro-5-[[3-(6-methoxy-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
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C26H19ClF3N3O6
 1
1
EC50 = 3000 nM
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CP0285884
(2R)-2-[2-chloro-5-[[3-[(4-chlorophenyl)methyl]-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
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C25H19Cl2F3N2O4
 1
1
EC50 = 3000 nM
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CP0298456
(2R)-2-[2-chloro-5-[[3-(5-methyl-1,2-benzoxazol-3-yl)-2-oxo-6-(trifluoromethyl)benzimidazol-1-yl]methyl]phenoxy]propanoic acid
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C26H19ClF3N3O5
 1
1
EC50 = 3000 nM
   TI
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CP0412944
(E)-9-oxohexadec-10-enoic acid
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C16H28O3
 1
1
EC50 = 8500 nM
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CP0444887
(E)-9-oxohexadec-7-enoic acid
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C16H28O3
 1
1
EC50 = 10000 nM
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CP0427644
5-chloro-2-(3-(2-(4-methoxybenzoyl)-4-methyl-1H-pyrrol-1-yl)prop-1-enyl)-N-(methylsulfonyl)benzamide
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C24H23ClN2O5S
 1
1
EC50 = 12000 nM
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CP0467414
(2E,4E,8Z,11Z,14Z,17Z)-icosa-2,4,8,11,14,17-hexaenoic acid
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C20H28O2
 1
1
EC50 > 1000 nM
   TI
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CP0467415
2-[2-ethyl-4-[[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]methylsulfanyl]phenoxy]-2-fluoroacetic acid
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C22H19F4NO3S2
 1
1
EC50 > 1000 nM
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CP0499556
2-fluoro-2-[2-methyl-4-[[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]methylsulfanyl]phenoxy]acetic acid
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C21H17F4NO3S2
 1
1
EC50 > 1000 nM
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CP0524690
2-fluoro-2-[4-[[4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]methylsulfanyl]-2-propan-2-ylphenoxy]acetic acid
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C23H21F4NO3S2
 1
1
EC50 > 1000 nM
   TI
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CP0034717
(S)-2-(4-(3-(2-chloro-4-cyclohexylphenoxy)propoxy)benzyl)-2-methylbutanoic acid
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C27H35ClO4
 1
1
EC50 > 3000 nM
   TI
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   TS
CP0104587
(S)-2-(4-(3-(2-chloro-4-(4,4-dimethylcyclohexyl)phenoxy)propoxy)benzyl)-2-methylbutanoic acid
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C29H39ClO4
 1
1
EC50 > 3000 nM
   TI
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CP0159827
(S)-2-((4-(3-(6-chloro-2-oxo-4-(trifluoromethyl)-2H-chromen-7-yloxy)propoxy)phenyl)methyl)-2-methylbutanoic acid
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C25H24ClF3O6
 1
1
EC50 > 3000 nM
   TI
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   TS
CP0170629
(S)-2-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propoxy)benzyl)-2-methylbutanoic acid
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C27H28ClFO5
 1
1
EC50 > 3000 nM
   TI
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CP0076778
2-(4-(4-Chlorobenzoyl)phenoxy)-2-methylpropanoic acid 1-methylethyl ester
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C20H21ClO4
 1
1
EC50 > 5000 nM
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CP0290865
(R)-7-{3-[2-Chloro-4-(tetrahydro-pyran-4-yl)-phenoxy]-propoxy}-2-ethyl-chroman-2-carboxylic acid
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C26H31ClO6
 1
1
EC50 ~ 15600 nM
   TI
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   TS