| Compound ID |
Compound Name |
Compound Formula |
|
CP0295856
|
9-methyl-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
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|
C16H12N2O2S
|
2
|
| 1 |
EC50 = 500 nM
|
|
|
| 2 |
EC50 = 800 nM
|
|
|
|
CP0295855
|
9-(trifluoromethyl)-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
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|
C16H9F3N2O2S
|
2
|
| 1 |
EC50 = 700 nM
|
|
|
| 2 |
EC50 = 1000 nM
|
|
|
|
CP0001758
|
(S)-4-methyl-2-(3-phenyl-propionylamino)-pentanoic acid [(S)-1-((S)-1-formyl-3-methyl-butylcarbamoyl)-3-methyl-butyl]-amide
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|
C26H41N3O5
|
2
|
| 1 |
EC50 = 1000 nM
|
|
|
| 2 |
EC50 = 5200 nM
|
|
|
|
CP0222585
|
2-methyl-5-nitro-N-quinolin-8-ylbenzenesulfonamide
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|
C16H13N3O4S
|
2
|
| 1 |
EC50 = 1000 nM
|
|
|
| 2 |
EC50 > 10000 nM
|
|
|
|
CP0192225
|
9-chloro-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
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|
C15H9ClN2O2S
|
2
|
| 1 |
EC50 = 1100 nM
|
|
|
| 2 |
EC50 = 11000 nM
|
|
|
|
CP0311125
|
9-methoxy-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
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|
C16H12N2O3S
|
2
|
| 1 |
EC50 = 1300 nM
|
|
|
| 2 |
EC50 = 1400 nM
|
|
|
|
CP0344211
|
11-methoxy-9-methyl-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
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|
C17H14N2O3S
|
2
|
| 1 |
EC50 = 1300 nM
|
|
|
| 2 |
EC50 = 1600 nM
|
|
|
|
CP0287020
|
11-methoxy-3,9-dimethyl-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
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|
C18H16N2O3S
|
2
|
| 1 |
EC50 = 1400 nM
|
|
|
| 2 |
EC50 = 2300 nM
|
|
|
|
CP0287021
|
5-chloro-N-(2-methylquinolin-8-yl)thiophene-2-sulfonamide
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|
C14H11ClN2O2S2
|
2
|
| 1 |
EC50 = 1400 nM
|
|
|
| 2 |
EC50 = 2100 nM
|
|
|
|
CP0211410
|
5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
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|
C15H10N2O2S
|
2
|
| 1 |
EC50 = 2200 nM
|
|
|
| 2 |
EC50 = 2600 nM
|
|
|
|
CP0344212
|
5-chloro-N-quinolin-8-ylthiophene-2-sulfonamide
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|
C13H9ClN2O2S2
|
1
|
| 1 |
EC50 = 2700 nM
|
|
|
|
CP0457822
|
2-amino-N-(6-methoxy-2-methylquinolin-8-yl)-4-methylbenzenesulfonamide
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|
C18H19N3O3S
|
2
|
| 1 |
EC50 = 3000 nM
|
|
|
| 2 |
EC50 = 9400 nM
|
|
|
|
CP0349445
|
9-methoxy-3-methyl-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
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|
C17H14N2O3S
|
2
|
| 1 |
EC50 = 3400 nM
|
|
|
| 2 |
EC50 = 3700 nM
|
|
|
|
CP0336677
|
2-nitro-N-quinolin-8-yl-4-(trifluoromethyl)benzenesulfonamide
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|
C16H10F3N3O4S
|
2
|
| 1 |
EC50 = 3600 nM
|
|
|
| 2 |
EC50 = 20000 nM
|
|
|
|
CP0336676
|
N-(2-methylquinolin-8-yl)-2-nitro-4-(trifluoromethyl)benzenesulfonamide
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|
C17H12F3N3O4S
|
2
|
| 1 |
EC50 = 3600 nM
|
|
|
| 2 |
EC50 = 10000 nM
|
|
|
|
CP0349446
|
2-amino-N-(6-methoxyquinolin-8-yl)-4-methylbenzenesulfonamide
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|
C17H17N3O3S
|
1
|
| 1 |
EC50 = 4000 nM
|
|
|
|
CP0294411
|
9-fluoro-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
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|
C15H9FN2O2S
|
2
|
| 1 |
EC50 = 4100 nM
|
|
|
| 2 |
EC50 = 12000 nM
|
|
|
|
CP0311126
|
N-quinolin-8-ylthiophene-2-sulfonamide
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|
C13H10N2O2S2
|
2
|
| 1 |
EC50 = 5300 nM
|
|
|
| 2 |
EC50 = 9000 nM
|
|
|
|
CP0102947
|
5-bromo-N-quinolin-8-ylthiophene-2-sulfonamide
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|
C13H9BrN2O2S2
|
2
|
| 1 |
EC50 = 5900 nM
|
|
|
| 2 |
EC50 = 6800 nM
|
|
|
|
CP0229637
|
N-(2-methylquinolin-8-yl)-3-nitrobenzenesulfonamide
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|
C16H13N3O4S
|
2
|
| 1 |
EC50 = 6000 nM
|
|
|
| 2 |
EC50 = 13000 nM
|
|
|
|
CP0222583
|
5-bromo-N-(2-methylquinolin-8-yl)thiophene-2-sulfonamide
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|
C14H11BrN2O2S2
|
2
|
| 1 |
EC50 = 6100 nM
|
|
|
| 2 |
EC50 = 6400 nM
|
|
|
|
CP0195678
|
4-nitro-N-quinolin-8-ylbenzenesulfonamide
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|
C15H11N3O4S
|
2
|
| 1 |
EC50 = 6500 nM
|
|
|
| 2 |
EC50 = 17000 nM
|
|
|
|
CP0168365
|
4-methyl-2-nitro-N-(8-quinolinyl)benzenesulfonamide
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|
C16H13N3O4S
|
2
|
| 1 |
EC50 = 6800 nM
|
|
|
| 2 |
EC50 = 10000 nM
|
|
|
|
CP0311127
|
N-(6-methoxyquinolin-8-yl)-4-methyl-2-nitrobenzenesulfonamide
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|
C17H15N3O5S
|
2
|
| 1 |
EC50 = 6800 nM
|
|
|
| 2 |
EC50 = 7600 nM
|
|
|
|
CP0349450
|
N-(2-methylquinolin-8-yl)-2-nitrobenzenesulfonamide
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|
C16H13N3O4S
|
2
|
| 1 |
EC50 = 6800 nM
|
|
|
| 2 |
EC50 = 8000 nM
|
|
|
|
CP0192224
|
2-methyl-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
Show/Hide
|
C16H12N2O2S
|
2
|
| 1 |
EC50 = 7000 nM
|
|
|
| 2 |
EC50 = 10000 nM
|
|
|
|
CP0339464
|
3-methyl-9-(trifluoromethyl)-5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide
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|
C17H11F3N2O2S
|
2
|
| 1 |
EC50 = 7200 nM
|
|
|
| 2 |
EC50 = 8900 nM
|
|
|
|
CP0052115
|
2-amino-N-(2-methylquinolin-8-yl)benzenesulfonamide
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|
C16H15N3O2S
|
1
|
| 1 |
EC50 = 8000 nM
|
|
|
|
CP0222582
|
3-methyl-6,6-dioxo-5H-quinolino[8,7-c][1,2]benzothiazin-9-ol
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|
C16H12N2O3S
|
2
|
| 1 |
EC50 = 8000 nM
|
|
|
| 2 |
EC50 = 11000 nM
|
|
|
|
CP0232467
|
2-amino-N-quinolin-8-ylbenzenesulfonamide
Show/Hide
|
C15H13N3O2S
|
2
|
| 1 |
EC50 = 8500 nM
|
|
|
| 2 |
EC50 = 11000 nM
|
|
|
|
CP0222584
|
N-(6-methoxy-2-methylquinolin-8-yl)-4-methyl-2-nitrobenzenesulfonamide
Show/Hide
|
C18H17N3O5S
|
2
|
| 1 |
EC50 > 10000 nM
|
|
|
| 2 |
EC50 > 57000 nM
|
|
|
|
CP0041688
|
2-nitro-N-(8-quinolinyl)benzenesulfonamide
Show/Hide
|
C15H11N3O4S
|
2
|
| 1 |
EC50 = 11000 nM
|
|
|
| 2 |
EC50 = 12000 nM
|
|
|
|
CP0031043
|
N-quinolin-8-ylbenzenesulfonamide
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|
C15H12N2O2S
|
2
|
| 1 |
EC50 = 17000 nM
|
|
|
| 2 |
EC50 = 20000 nM
|
|
|
|
CP0339465
|
2-methyl-N-(2-methylquinolin-8-yl)-5-nitrobenzenesulfonamide
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|
C17H15N3O4S
|
2
|
| 1 |
EC50 > 20000 nM
|
|
|
| 2 |
EC50 > 57000 nM
|
|
|
|
CP0349448
|
N-(6-methoxy-2-methylquinolin-8-yl)-4-methylbenzenesulfonamide
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|
C18H18N2O3S
|
1
|
| 1 |
EC50 = 20000 nM
|
|
|
