Compound ID |
Compound Name |
Compound Formula |
CP0067951
|
N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-4-sulfonamide
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|
C23H27N5O3S
|
1
|
1 |
IC50 = 1 nM
|
|
|
CP0447538
|
N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-5-sulfonamide
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|
C23H27N5O3S
|
1
|
1 |
IC50 = 12.59 nM
|
|
|
CP0065780
|
4-amino-3,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
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|
C21H25Cl2N5O3S
|
1
|
1 |
IC50 = 15.85 nM
|
|
|
CP0445928
|
N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-6-sulfonamide
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|
C23H27N5O3S
|
1
|
1 |
IC50 = 15.85 nM
|
|
|
CP0419712
|
3-amino-N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-2,4-dimethylbenzenesulfonamide
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|
C23H31N5O3S
|
1
|
1 |
IC50 = 79.43 nM
|
|
|
CP0534634
|
4-amino-3,5-dichloro-N-[4-(2-chloroimidazol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamide
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|
C19H24Cl3N5O3S
|
1
|
1 |
IC50 = 251.19 nM
|
|
|
CP0427286
|
4-amino-3,5-dichloro-N-[(2R)-1-(4-methylpiperidin-1-yl)-1-oxo-4-phenylbutan-2-yl]benzenesulfonamide
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|
C22H27Cl2N3O3S
|
1
|
1 |
IC50 = 501.19 nM
|
|
|
CP0419711
|
4-amino-3,5-dichloro-N-[1-(4-methylpiperidin-1-yl)-1-oxo-4-pyrazol-1-ylbutan-2-yl]benzenesulfonamide
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|
C19H25Cl2N5O3S
|
1
|
1 |
IC50 = 1258.93 nM
|
|
|
CP0427285
|
4-amino-3,5-dichloro-N-[1-(4-methylpiperidin-1-yl)-1-oxo-4-(triazol-2-yl)butan-2-yl]benzenesulfonamide
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|
C18H24Cl2N6O3S
|
1
|
1 |
IC50 = 1258.93 nM
|
|
|
CP0519192
|
4-amino-3,5-dichloro-N-[(2S)-1-(4-methylpiperidin-1-yl)-1-oxo-4-phenylbutan-2-yl]benzenesulfonamide
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|
C22H27Cl2N3O3S
|
1
|
1 |
IC50 > 10000 nM
|
|
|