| Compound ID |
Compound Name |
Compound Formula |
|
CP0190068
|
N-[4-methyl-3-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]oxyphenyl]-4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)benzamide
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|
C33H38F3N5O3
|
1
|
| 1 |
GI50 = 658 nM
|
|
|
|
CP0065873
|
1-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-2-(dimethylamino)ethanone
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|
C26H29N7O2
|
1
|
| 1 |
GI50 = 940 nM
|
|
|
|
CP0389976
|
4-(methylamino)-2-[4-methyl-3-(prop-2-enoylamino)anilino]-N-[2-methyl-5-[[3-(trifluoromethyl)benzoyl]amino]phenyl]pyrimidine-5-carboxamide
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|
C31H28F3N7O3
|
2
|
| 1 |
GI50 = 5900 nM
|
|
|
| 2 |
GI50 > 10000 nM
|
|
|
|
CP0387299
|
4-(methylamino)-2-[4-methyl-3-(propanoylamino)anilino]-N-[2-methyl-5-[[3-(trifluoromethyl)benzoyl]amino]phenyl]pyrimidine-5-carboxamide
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|
C31H30F3N7O3
|
2
|
| 1 |
GI50 = 6500 nM
|
|
|
| 2 |
GI50 > 10000 nM
|
|
|
|
CP0002778
|
4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamide
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|
C29H31N7O
|
1
|
| 1 |
GI50 > 10000 nM
|
|
|
|
CP0224766
|
4-(methylamino)-2-[4-methyl-3-(prop-2-enoylamino)anilino]-N-[2-methyl-5-[(3,4,5-trimethoxybenzoyl)amino]phenyl]pyrimidine-5-carboxamide
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|
C33H35N7O6
|
1
|
| 1 |
GI50 > 10000 nM
|
|
|
|
CP0387298
|
4-(methylamino)-2-[4-methyl-3-(propanoylamino)anilino]-N-[2-methyl-5-[(3,4,5-trimethoxybenzoyl)amino]phenyl]pyrimidine-5-carboxamide
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|
C33H37N7O6
|
1
|
| 1 |
GI50 > 10000 nM
|
|
|
|
CP0061016
|
3-(4-Amino-7-cyclopentyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)-phenol
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|
C17H18N4O
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0388620
|
methyl N-[4-[7-amino-3-(3,4-dimethoxyphenyl)-5-(1-methylpiperidin-4-yl)oxypyrazolo[1,5-a]pyrimidin-6-yl]phenyl]carbamate
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|
C28H32N6O5
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0388616
|
3-(3,4-dimethoxyphenyl)-5-(1-methylpiperidin-4-yl)oxy-6-phenylpyrazolo[1,5-a]pyrimidin-7-amine
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|
C26H29N5O3
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0418567
|
3-[4-amino-7-[3-(hydroxymethyl)cyclobutyl]pyrrolo[2,3-d]pyrimidin-5-yl]phenol
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|
C17H18N4O2
|
1
|
| 1 |
IC50 = 570 nM
|
|
|
|
CP0138866
|
1-[4-[3-[4-amino-5-(2-fluoro-5-hydroxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclobutyl]piperazin-1-yl]ethanone
Show/Hide
|
C22H25FN6O2
|
1
|
| 1 |
IC50 = 3600 nM
|
|
|
|
CP0388615
|
3-(3,4-dimethoxyphenyl)-5-(1-methylpiperidin-4-yl)oxy-6-(1,3-thiazol-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
Show/Hide
|
C23H26N6O3S
|
1
|
| 1 |
IC50 = 8200 nM
|
|
|
