| Compound ID |
Compound Name |
Compound Formula |
|
CP0561634
|
US9434725, 122
Show/Hide
|
C23H25N7O
|
1
|
| 1 |
IC50 = 71.5 nM
|
|
|
|
CP0393246
|
US9434725, 168
Show/Hide
|
C20H20N8
|
1
|
| 1 |
IC50 = 75.5 nM
|
|
|
|
CP0564892
|
US9434725, 172
Show/Hide
|
C22H24N8O
|
1
|
| 1 |
IC50 = 111 nM
|
|
|
|
CP0567653
|
US9434725, 285
Show/Hide
|
C21H23N9
|
1
|
| 1 |
IC50 = 112 nM
|
|
|
|
CP0478323
|
US9434725, 306
Show/Hide
|
C21H19F4N7
|
1
|
| 1 |
IC50 = 129 nM
|
|
|
|
CP0479633
|
US9434725, 165
Show/Hide
|
C22H22N8
|
1
|
| 1 |
IC50 = 139 nM
|
|
|
|
CP0513361
|
US9434725, 282
Show/Hide
|
C21H23N9O
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0578206
|
US9434725, 208
Show/Hide
|
C21H23N9
|
1
|
| 1 |
IC50 = 173 nM
|
|
|
|
CP0419275
|
US9434725, 162
Show/Hide
|
C21H22F2N8
|
1
|
| 1 |
IC50 = 175 nM
|
|
|
|
CP0516120
|
US9434725, 189
Show/Hide
|
C21H21F3N8O
|
1
|
| 1 |
IC50 = 181 nM
|
|
|
|
CP0532564
|
US9434725, 150
Show/Hide
|
C22H24N8
|
1
|
| 1 |
IC50 = 196 nM
|
|
|
|
CP0516406
|
US9434725, 218
Show/Hide
|
C22H24N8O
|
1
|
| 1 |
IC50 = 212 nM
|
|
|
|
CP0578203
|
US9434725, 181
Show/Hide
|
C24H26N8
|
1
|
| 1 |
IC50 = 214 nM
|
|
|
|
CP0085927
|
US9434725, 186
Show/Hide
|
C22H24N8O
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0483229
|
US9434725, 190
Show/Hide
|
C21H22N8
|
1
|
| 1 |
IC50 = 235 nM
|
|
|
|
CP0512362
|
US9434725, 313
Show/Hide
|
C19H19N9
|
1
|
| 1 |
IC50 = 236 nM
|
|
|
|
CP0518526
|
US9434725, 149
Show/Hide
|
C21H22N8
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0478322
|
US9434725, 304
Show/Hide
|
C20H19N7O
|
1
|
| 1 |
IC50 = 255 nM
|
|
|
|
CP0471270
|
US9434725, 278
Show/Hide
|
C21H22N8O2
|
1
|
| 1 |
IC50 = 261 nM
|
|
|
|
CP0479634
|
US9434725, 166
Show/Hide
|
C21H21N7
|
1
|
| 1 |
IC50 = 270 nM
|
|
|
|
CP0451558
|
US9434725, 174
Show/Hide
|
C22H24N8
|
1
|
| 1 |
IC50 = 271 nM
|
|
|
|
CP0567651
|
US9434725, 205
Show/Hide
|
C22H24N8
|
1
|
| 1 |
IC50 = 278 nM
|
|
|
|
CP0406605
|
US9434725, 123
Show/Hide
|
C20H20N8
|
1
|
| 1 |
IC50 = 284 nM
|
|
|
|
CP0465859
|
US9434725, 153
Show/Hide
|
C21H23FN8
|
1
|
| 1 |
IC50 = 291 nM
|
|
|
|
CP0539934
|
US9434725, 154
Show/Hide
|
C21H21F3N8
|
1
|
| 1 |
IC50 = 344 nM
|
|
|
|
CP0479635
|
US9434725, 179
Show/Hide
|
C20H20F3N9
|
1
|
| 1 |
IC50 = 376 nM
|
|
|
|
CP0488613
|
US9434725, 260
Show/Hide
|
C22H23F3N8O
|
1
|
| 1 |
IC50 = 380 nM
|
|
|
|
CP0515240
|
US9434725, 284
Show/Hide
|
C22H23N9
|
1
|
| 1 |
IC50 = 385 nM
|
|
|
|
CP0529004
|
US9434725, 144
Show/Hide
|
C19H18N8
|
1
|
| 1 |
IC50 = 385 nM
|
|
|
|
CP0578204
|
US9434725, 188
Show/Hide
|
C21H21F3N8O
|
1
|
| 1 |
IC50 = 418 nM
|
|
|
|
CP0565323
|
US9434725, 295
Show/Hide
|
C22H23N7O
|
1
|
| 1 |
IC50 = 425 nM
|
|
|
|
CP0445039
|
US9434725, 112
Show/Hide
|
C24H25N7
|
1
|
| 1 |
IC50 = 490 nM
|
|
|
|
CP0575914
|
US9434725, 201
Show/Hide
|
C22H21N9
|
1
|
| 1 |
IC50 = 490 nM
|
|
|
|
CP0497624
|
US9434725, 155
Show/Hide
|
C21H21N9
|
1
|
| 1 |
IC50 = 518 nM
|
|
|
|
CP0393247
|
US9434725, 176
Show/Hide
|
C21H21ClN8
|
1
|
| 1 |
IC50 = 533 nM
|
|
|
|
CP0419273
|
US9434725, 151
Show/Hide
|
C21H22N8O
|
1
|
| 1 |
IC50 = 544 nM
|
|
|
|
CP0549620
|
US9434725, 167
Show/Hide
|
C20H20N8
|
1
|
| 1 |
IC50 = 546 nM
|
|
|
|
CP0515238
|
US9434725, 178
Show/Hide
|
C20H20F3N9
|
1
|
| 1 |
IC50 = 549 nM
|
|
|
|
CP0483230
|
US9434725, 196
Show/Hide
|
C21H22N8
|
1
|
| 1 |
IC50 = 572 nM
|
|
|
|
CP0110430
|
US9434725, 138
Show/Hide
|
C21H22N8
|
1
|
| 1 |
IC50 = 574 nM
|
|
|
|
CP0563781
|
US9434725, 279
Show/Hide
|
C20H18F2N8
|
1
|
| 1 |
IC50 = 622 nM
|
|
|
|
CP0483233
|
US9434725, 273
Show/Hide
|
C20H20N8O
|
1
|
| 1 |
IC50 = 629 nM
|
|
|
|
CP0564894
|
US9434725, 307
Show/Hide
|
C20H20N8
|
1
|
| 1 |
IC50 = 640 nM
|
|
|
|
CP0483232
|
US9434725, 209
Show/Hide
|
C21H23N9
|
1
|
| 1 |
IC50 = 682 nM
|
|
|
|
CP0483234
|
US9434725, 281
Show/Hide
|
C22H23N9O
|
1
|
| 1 |
IC50 = 695 nM
|
|
|
|
CP0554650
|
US9434725, 216
Show/Hide
|
C24H26N8
|
1
|
| 1 |
IC50 = 715 nM
|
|
|
|
CP0393248
|
US9434725, 180
Show/Hide
|
C19H20N8
|
1
|
| 1 |
IC50 = 745 nM
|
|
|
|
CP0566379
|
US9434725, 274
Show/Hide
|
C21H20N8
|
1
|
| 1 |
IC50 = 749 nM
|
|
|
|
CP0564882
|
US9434725, 294
Show/Hide
|
C21H20FN7
|
1
|
| 1 |
IC50 = 772 nM
|
|
|
|
CP0567652
|
US9434725, 228
Show/Hide
|
C21H23N9
|
1
|
| 1 |
IC50 = 778 nM
|
|
|
|
CP0563393
|
US9434725, 301
Show/Hide
|
C22H24N8O
|
1
|
| 1 |
IC50 = 781 nM
|
|
|
|
CP0495376
|
US9434725, 146
Show/Hide
|
C22H26N8
|
1
|
| 1 |
IC50 = 797 nM
|
|
|
|
CP0564470
|
US9434725, 124
Show/Hide
|
C20H21N7S
|
1
|
| 1 |
IC50 = 804 nM
|
|
|
|
CP0514648
|
US9434725, 225
Show/Hide
|
C21H20N8O
|
1
|
| 1 |
IC50 = 840 nM
|
|
|
|
CP0515239
|
US9434725, 227
Show/Hide
|
C22H22F2N8
|
1
|
| 1 |
IC50 = 869 nM
|
|
|
|
CP0530438
|
US9434725, 147
Show/Hide
|
C23H26N8
|
1
|
| 1 |
IC50 = 869 nM
|
|
|
|
CP0393254
|
US9434725, 277
Show/Hide
|
C21H22N8O2
|
1
|
| 1 |
IC50 = 912 nM
|
|
|
|
CP0469600
|
US9434725, 191
Show/Hide
|
C21H22N8
|
1
|
| 1 |
IC50 = 919 nM
|
|
|
|
CP0564064
|
US9434725, 187
Show/Hide
|
C22H24N8
|
1
|
| 1 |
IC50 = 963 nM
|
|
|
|
CP0512361
|
US9434725, 293
Show/Hide
|
C23H24N8
|
1
|
| 1 |
IC50 = 976 nM
|
|
|
|
CP0393253
|
US9434725, 214
Show/Hide
|
C22H22N8
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0445042
|
US9434725, 141
Show/Hide
|
C22H23N7
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0513362
|
US9434725, 283
Show/Hide
|
C24H27N9O
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0563782
|
US9434725, 317
Show/Hide
|
C22H20N8
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0393250
|
US9434725, 198
Show/Hide
|
C21H21FN8
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0565321
|
US9434725, 184
Show/Hide
|
C22H24N8
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0471272
|
US9434725, 297
Show/Hide
|
C17H15N7
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0497619
|
US9434725, 106
Show/Hide
|
C23H25N7O
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0530436
|
US9434725, 103
Show/Hide
|
C24H27N7
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0564878
|
US9434725, 215
Show/Hide
|
C21H21FN8
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0564880
|
US9434725, 220
Show/Hide
|
C22H21F3N8
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0515254
|
US9434725, 308
Show/Hide
|
C18H16N8
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0576939
|
US9434725, 300
Show/Hide
|
C22H20N8O
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0497625
|
US9434725, 156
Show/Hide
|
C22H24N8
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0561635
|
US9434725, 125
Show/Hide
|
C21H24N8
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0564469
|
US9434725, 120
Show/Hide
|
C20H21N7S
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0393251
|
US9434725, 207
Show/Hide
|
C22H24N8O2
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0481144
|
US9434725, 194
Show/Hide
|
C21H22N8
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0481145
|
US9434725, 224
Show/Hide
|
C20H22N8
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0497620
|
US9434725, 130
Show/Hide
|
C20H20N8O
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0559292
|
US9434725, 152
Show/Hide
|
C21H24N8O
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0563439
|
US9434725, 109
Show/Hide
|
C18H17N7S
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0564468
|
US9434725, 104
Show/Hide
|
C22H23N7
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0499635
|
US9434725, 105
Show/Hide
|
C23H25N7
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0513363
|
US9434725, 299
Show/Hide
|
C21H21N7O
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0536004
|
US9434725, 298
Show/Hide
|
C21H21N7O
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0532642
|
US9434725, 101
Show/Hide
|
C20H22N8
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0565735
|
US9434725, 110
Show/Hide
|
C19H19N7S
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0575913
|
US9434725, 192
Show/Hide
|
C21H21FN8
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0576940
|
US9434725, 315
Show/Hide
|
C21H18N8
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0497621
|
US9434725, 137
Show/Hide
|
C21H22N8
|
1
|
| 1 |
IC50 = 2100 nM
|
|
|
|
CP0578205
|
US9434725, 197
Show/Hide
|
C24H26N8
|
1
|
| 1 |
IC50 = 2200 nM
|
|
|
|
CP0500959
|
US9434725, 139
Show/Hide
|
C26H29N7
|
1
|
| 1 |
IC50 = 2300 nM
|
|
|
|
CP0529051
|
US9434725, 107
Show/Hide
|
C24H27N7
|
1
|
| 1 |
IC50 = 2400 nM
|
|
|
|
CP0497623
|
US9434725, 145
Show/Hide
|
C23H28N8
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0563458
|
US9434725, 157
Show/Hide
|
C22H26N8O2S
|
1
|
| 1 |
IC50 = 2800 nM
|
|
|
|
CP0530437
|
US9434725, 117
Show/Hide
|
C23H24ClN7
|
1
|
| 1 |
IC50 = 2900 nM
|
|
|
|
CP0445040
|
US9434725, 133
Show/Hide
|
C21H24N8
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0488614
|
US9434725, 296
Show/Hide
|
C18H17N7
|
1
|
| 1 |
IC50 = 3800 nM
|
|
|
|
CP0563392
|
US9434725, 286
Show/Hide
|
C21H23N9O
|
1
|
| 1 |
IC50 = 4200 nM
|
|
|
|
CP0495375
|
US9434725, 108
Show/Hide
|
C24H27N7
|
1
|
| 1 |
IC50 = 4500 nM
|
|
|
|
CP0564893
|
US9434725, 302
Show/Hide
|
C22H22N8O
|
1
|
| 1 |
IC50 = 6100 nM
|
|
|
|
CP0483235
|
US9434725, 303
Show/Hide
|
C22H22N8O
|
1
|
| 1 |
IC50 = 6600 nM
|
|
|
|
CP0483236
|
US9434725, 316
Show/Hide
|
C21H22FN7
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
