| Compound ID |
Compound Name |
Compound Formula |
|
CP0190068
|
N-[4-methyl-3-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]oxyphenyl]-4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)benzamide
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|
C33H38F3N5O3
|
1
|
| 1 |
GI50 = 33 nM
|
|
|
|
CP0451979
|
4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[1-(pyridine-2-carbonyl)piperidin-4-yl]oxyphenyl]-3-(trifluoromethyl)benzamide
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|
C32H36F3N5O3
|
1
|
| 1 |
GI50 = 72 nM
|
|
|
|
CP0451447
|
N-[4-methyl-3-[1-(5-methylpyridine-3-carbonyl)piperidin-4-yl]oxyphenyl]-4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)benzamide
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|
C33H38F3N5O3
|
1
|
| 1 |
GI50 = 79 nM
|
|
|
|
CP0884002
|
N-(4-Methyl-3-((1-(quinoline-3-carbonyl)piperidin-4-yl)oxy)-phenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
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|
C36H38F3N5O3
|
1
|
| 1 |
GI50 = 86 nM
|
|
|
|
CP0401091
|
4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[1-(pyridine-4-carbonyl)piperidin-4-yl]oxyphenyl]-3-(trifluoromethyl)benzamide
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|
C32H36F3N5O3
|
1
|
| 1 |
GI50 = 88 nM
|
|
|
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CP0897977
|
N-(4-Methyl-3-((1-(thiophene-3-carbonyl)piperidin-4-yl)oxy)-phenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)-benzamide
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|
C31H35F3N4O3S
|
1
|
| 1 |
GI50 = 135 nM
|
|
|
|
CP0883945
|
N-(3-((1-(Furan-3-carbonyl)piperidin-4-yl)oxy)-4-methylphenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
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|
C31H35F3N4O4
|
1
|
| 1 |
GI50 = 153 nM
|
|
|
|
CP0890778
|
N-(4-Methyl-3-((1-nicotinoylpiperidin-4-yl)oxy)phenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
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|
C32H36F3N5O3
|
1
|
| 1 |
GI50 = 164 nM
|
|
|
|
CP0888364
|
N-(3-((1-(2-Aminopyrimidine-5-carbonyl)piperidin-4-yl)oxy)-4-methylphenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
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|
C31H36F3N7O3
|
1
|
| 1 |
GI50 = 168 nM
|
|
|
|
CP0446640
|
N-[4-methyl-3-[1-(4-methylpyridine-3-carbonyl)piperidin-4-yl]oxyphenyl]-4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)benzamide
Show/Hide
|
C33H38F3N5O3
|
1
|
| 1 |
GI50 = 203 nM
|
|
|
|
CP0895611
|
N-(3-((1-(5-Chloronicotinoyl)piperidin-4-yl)oxy)-4-methylphenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
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|
C32H35ClF3N5O3
|
1
|
| 1 |
GI50 = 219 nM
|
|
|
|
CP0903642
|
N-(4-Chloro-3-((1-nicotinoylpiperidin-4-yl)oxy)phenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
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|
C31H33ClF3N5O3
|
1
|
| 1 |
GI50 = 253 nM
|
|
|
|
CP0002778
|
4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamide
Show/Hide
|
C29H31N7O
|
1
|
| 1 |
GI50 = 270 nM
|
|
|
|
CP0897981
|
N-(3-((1-Acryloylpiperidin-4-yl)oxy)-4-methylphenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
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|
C29H35F3N4O3
|
1
|
| 1 |
GI50 = 427 nM
|
|
|
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CP0897978
|
N-(3-((1-Benzoylpiperidin-4-yl)oxy)-4-methylphenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C33H37F3N4O3
|
1
|
| 1 |
GI50 = 635 nM
|
|
|
|
CP0897980
|
N-(3-((1-(6,7-Dimethoxyquinazolin-4-yl)piperidin-4-yl)oxy)-4-methylphenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
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|
C36H41F3N6O4
|
1
|
| 1 |
GI50 = 773 nM
|
|
|
|
CP0942783
|
N-(4-Methyl-3-((1-propionylpiperidin-4-yl)oxy)phenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
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|
C29H37F3N4O3
|
1
|
| 1 |
GI50 = 998 nM
|
|
|
|
CP0942782
|
N-(2-(2-Methyl-5-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamido)phenoxy)ethyl)nicotinamide
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|
C29H32F3N5O3
|
1
|
| 1 |
GI50 = 1550 nM
|
|
|
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CP0890764
|
N-(4-Methyl-3-((1-(6-oxo-1,6-dihydropyridine-3-carbonyl)-piperidin-4-yl)oxy)phenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C32H36F3N5O4
|
1
|
| 1 |
GI50 = 1970 nM
|
|
|
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CP0893566
|
N-(3-((1-(2-Fluoronicotinoyl)piperidin-4-yl)oxy)-4-methylphenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C32H35F4N5O3
|
1
|
| 1 |
GI50 = 2000 nM
|
|
|
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CP0859245
|
N-(4-Methyl-3-((1-(2-methylnicotinoyl)piperidin-4-yl)oxy)-phenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)-benzamide
Show/Hide
|
C33H38F3N5O3
|
1
|
| 1 |
GI50 = 2210 nM
|
|
|
|
CP0859246
|
N-(3-((1-(2-Chloronicotinoyl)piperidin-4-yl)oxy)-4-methylphenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C32H35ClF3N5O3
|
1
|
| 1 |
GI50 = 2760 nM
|
|
|
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CP0883946
|
N-(3-((1-(2-(Dimethylamino)acetyl)piperidin-4-yl)oxy)-4-methylphenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C30H40F3N5O3
|
1
|
| 1 |
GI50 = 3070 nM
|
|
|
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CP0888365
|
N-(4-Methyl-3-((1-(pyrimidin-2-yl)piperidin-4-yl)oxy)phenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C30H35F3N6O2
|
1
|
| 1 |
GI50 = 3220 nM
|
|
|
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CP0942862
|
N-(4-Methyl-3-((1-(phenylsulfonyl)piperidin-4-yl)oxy)phenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C32H37F3N4O4S
|
1
|
| 1 |
GI50 = 4770 nM
|
|
|
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CP0897979
|
N-(4-Methyl-3-((1-nicotinoylpyrrolidin-3-yl)methoxy)phenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C32H36F3N5O3
|
1
|
| 1 |
GI50 = 4940 nM
|
|
|
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CP0859247
|
N-(4-Methyl-3-((1-nicotinoylazetidin-3-yl)methoxy)phenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C31H34F3N5O3
|
1
|
| 1 |
GI50 = 5400 nM
|
|
|
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CP0883947
|
N-(4-Methyl-3-((1-(2-(pyridin-3-yl)acetyl)piperidin-4-yl)oxy)-phenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)-benzamide
Show/Hide
|
C33H38F3N5O3
|
1
|
| 1 |
GI50 = 5520 nM
|
|
|
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CP0883937
|
N-(4-Methoxy-3-((1-nicotinoylpiperidin-4-yl)oxy)phenyl)-4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C32H36F3N5O4
|
1
|
| 1 |
GI50 = 8410 nM
|
|
|
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CP0922099
|
N-(4-Methyl-3-((1-nicotinoylpiperidin-4-yl)oxy)phenyl)-4-((4-methylpiperazin-1-yl)methyl)benzamide
Show/Hide
|
C31H37N5O3
|
1
|
| 1 |
GI50 = 8780 nM
|
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