| Compound ID |
Compound Name |
Compound Formula |
|
CP0966272
|
N-[(1R,3S)-3-[(3aS,6aS)-4-acetyl-2,3,3a,5,6,6a-hexahydropyrrolo[3,2-b]pyrrol-1-yl]cyclohexyl]-4-fluoro-7-methyl-1H-indole-2-carboxamide
Show/Hide
|
C24H31FN4O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0970274
|
N-[(1R,3S)-3-[(8aS)-6-oxo-1,3,4,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-2-yl]cyclohexyl]-4-fluoro-7-methyl-1H-indole-2-carboxamide
Show/Hide
|
C23H29FN4O2
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0953005
|
N-[(1R,3S)-3-[(3aS,6aS)-1-acetyl-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-5-yl]cyclohexyl]-4-fluoro-7-methyl-1H-indole-2-carboxamide
Show/Hide
|
C24H31FN4O2
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0964776
|
4-fluoro-7-methyl-N-((1R,3S)-3-((S)-3-(N-methylmethylsulfonamido)pyrrolidin-1-yl)cyclohexyl)-1H-indole-2-carboxamide
Show/Hide
|
C22H31FN4O3S
|
2
|
| 1 |
IC50 = 20 nM
|
|
|
| 2 |
IC50 = 23 nM
|
|
|
|
CP0967445
|
4-fluoro-N-(3-fluoro-5-(3-(N-methylacetamido)pyrrolidin-1-yl)phenyl)-7-methyl-1H-indole-2-carboxamide
Show/Hide
|
C23H24F2N4O2
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0578575
|
EZM-0414
Show/Hide
|
C22H29FN4O2
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0578225
|
N-[3-(4-acetylpiperazin-1-yl)-5-fluorophenyl]-4-fluoro-7-methyl-1H-indole-2-carboxamide
Show/Hide
|
C22H22F2N4O2
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0769272
|
4-fluoro-7-methyl-N-((1R,3S)-3-((R)-3-(N-methylmethylsulfonamido)pyrrolidin-1-yl)cyclohexyl)-1H-indole-2-carboxamide
Show/Hide
|
C24H37FN4O3S
|
1
|
| 1 |
IC50 = 64 nM
|
|
|
|
CP0969976
|
4-fluoro-7-methyl-N-((1R,3S)-3-((R)-3-(N-methylacetamido)pyrrolidin-1-yl)cyclohexyl)-1H-indole-2-carboxamide
Show/Hide
|
C23H31FN4O2
|
1
|
| 1 |
IC50 = 74 nM
|
|
|
|
CP0969135
|
4-fluoro-7-methyl-N-(3-(3-(N-methylacetamido)pyrrolidin-1-yl)phenyl)-1H-indole-2-carboxamide
Show/Hide
|
C23H25FN4O2
|
1
|
| 1 |
IC50 = 93 nM
|
|
|
|
CP0969975
|
4-fluoro-7-methyl-N-((1R,3S)-3-((S)-3-(N-methylacetamido)pyrrolidin-1-yl)cyclohexyl)-1H-indole-2-carboxamide
Show/Hide
|
C23H31FN4O2
|
1
|
| 1 |
IC50 = 127 nM
|
|
|
|
CP0579810
|
N-[3-(4-acetylpiperazin-1-yl)phenyl]-4-fluoro-7-methyl-1H-indole-2-carboxamide
Show/Hide
|
C22H23FN4O2
|
1
|
| 1 |
IC50 = 134 nM
|
|
|
|
CP0950353
|
4-fluoro-7-methyl-N-((1R,3S)-3-(4-(methylsulfonyl)piperazin-1-yl)cyclohexyl)-1H-indole-2-carboxamide
Show/Hide
|
C21H29FN4O3S
|
1
|
| 1 |
IC50 = 162 nM
|
|
|
|
CP0576300
|
N-[3-[4-(dimethylamino)piperidin-1-yl]-5-fluorophenyl]-4-fluoro-7-methyl-1H-indole-2-carboxamide
Show/Hide
|
C23H26F2N4O
|
1
|
| 1 |
IC50 = 175 nM
|
|
|
|
CP0578688
|
N-[3-[4-(dimethylamino)piperidin-1-yl]phenyl]-4-fluoro-7-methyl-1H-indole-2-carboxamide
Show/Hide
|
C23H27FN4O
|
1
|
| 1 |
IC50 = 235 nM
|
|
|
|
CP0969255
|
4-fluoro-7-methyl-N-((1R,3S)-3-(pyridin-4-yl)cyclohexyl)-1H-indole-2-carboxamide
Show/Hide
|
C21H22FN3O
|
1
|
| 1 |
IC50 = 257 nM
|
|
|
|
CP0826362
|
4-fluoro-7-methyl-N-((1R,3S)-3-(4-methyl-3-oxopiperazin-1-yl)cyclohexyl)-1H-indole-2-carboxamide
Show/Hide
|
C21H27FN4O2
|
1
|
| 1 |
IC50 = 340 nM
|
|
|
|
CP0552448
|
N-[3-[4-(dimethylamino)piperidin-1-yl]-5-methylphenyl]-4-fluoro-7-methyl-1H-indole-2-carboxamide
Show/Hide
|
C24H29FN4O
|
1
|
| 1 |
IC50 = 379 nM
|
|
|
|
CP0542623
|
N-[3-chloro-5-[4-(dimethylamino)piperidin-1-yl]phenyl]-4-fluoro-7-methyl-1H-indole-2-carboxamide
Show/Hide
|
C23H26ClFN4O
|
1
|
| 1 |
IC50 = 384 nM
|
|
|
|
CP0578689
|
4-fluoro-7-methyl-N-(3-morpholin-4-ylphenyl)-1H-indole-2-carboxamide
Show/Hide
|
C20H20FN3O2
|
1
|
| 1 |
IC50 = 397 nM
|
|
|
|
CP0968662
|
4-fluoro-7-methyl-N-((1R,3S)-3-morpholinocyclohexyl)-1H-indole-2-carboxamide
Show/Hide
|
C20H26FN3O2
|
1
|
| 1 |
IC50 = 449 nM
|
|
|
|
CP0578735
|
4-fluoro-7-methyl-N-[3-(4-methylpiperazin-1-yl)phenyl]-1H-indole-2-carboxamide
Show/Hide
|
C21H23FN4O
|
1
|
| 1 |
IC50 = 540 nM
|
|
|
|
CP0569468
|
7-methyl-N-(3-morpholin-4-ylphenyl)-1H-indole-2-carboxamide
Show/Hide
|
C20H21N3O2
|
1
|
| 1 |
IC50 = 2040 nM
|
|
|
|
CP0970222
|
N-[(1S,3R)-3-(4-acetylpiperazin-1-yl)cyclohexyl]-4-fluoro-7-methyl-1H-indole-2-carboxamide
Show/Hide
|
C22H29FN4O2
|
1
|
| 1 |
IC50 > 2000 nM
|
|
|
|
CP0970486
|
N-[(1S,3S)-3-(4-acetylpiperazin-1-yl)cyclohexyl]-4-fluoro-7-methyl-1H-indole-2-carboxamide
Show/Hide
|
C22H29FN4O2
|
1
|
| 1 |
IC50 > 2000 nM
|
|
|
|
CP0970646
|
N-[(1R,3R)-3-(4-acetylpiperazin-1-yl)cyclohexyl]-4-fluoro-7-methyl-1H-indole-2-carboxamide
Show/Hide
|
C22H29FN4O2
|
1
|
| 1 |
IC50 > 2000 nM
|
|
|
