Brief Information of the Cell Line and Protein
Cell Line ID: CL000065 , HEK293-EBNA
Synonyms
293 c18
293c18
HEK 293 c18
HEK-293 c18
HEK293-EBNA1
HEK-293-EBNA
HEK 293-EBNA
HEK 293 EBNA
HEK293EBNA
293 EBNA
293-EBNA1
293-EBNA
293/EBNA
293EBNA
EBNA-293
EBNA293
293E
HEK293E
HEK/EBNA
HEK-EBNA
HEK.EBNA
293/EBNA-1
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_6974
Protein ID: PT00941 , 5-hydroxytryptamine receptor 7
Gene Name HTR7
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P34969
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000065  Protein ID: PT00941
 
Compound ID Compound Name Compound Formula
CP0378319
4-methyl-8-propan-2-yloxy-1,4-dihydroquinazolin-2-amine
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C12H17N3O
 1
1
Ki = 1 nM
   TI
   LI
   LO
   TS
CP0378317
N,4-dimethyl-8-propan-2-yloxy-3,4-dihydro-1H-quinazolin-2-imine
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C13H19N3O
 1
1
Ki = 2.4 nM
   TI
   LI
   LO
   TS
CP0438872
5,8-dichloro-4-methyl-1,4-dihydroquinazolin-2-amine
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C9H9Cl2N3
 1
1
Ki = 2.4 nM
   TI
   LI
   LO
   TS
CP0378316
6-chloro-8-methoxy-4,5-dimethyl-1,4-dihydroquinazolin-2-amine
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C11H14ClN3O
 1
1
Ki = 2.5 nM
   TI
   LI
   LO
   TS
CP0496556
8-methoxy-4-methyl-1,4-dihydroquinazolin-2-amine
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C10H13N3O
 1
1
Ki = 8.2 nM
   TI
   LI
   LO
   TS
CP0288769
5,6-dichloro-4-methyl-1,4-dihydroquinazolin-2-amine
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C9H9Cl2N3
 1
1
Ki = 8.7 nM
   TI
   LI
   LO
   TS
CP0378318
6-chloro-5-methoxy-4-methyl-1,4-dihydroquinazolin-2-amine
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C10H12ClN3O
 1
1
Ki = 12.4 nM
   TI
   LI
   LO
   TS
CP0378320
5,6-dichloro-N,4-dimethyl-3,4-dihydro-1H-quinazolin-2-imine
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C10H11Cl2N3
 1
1
Ki = 13.2 nM
   TI
   LI
   LO
   TS
CP0490337
5-chloro-N,4-dimethyl-3,4-dihydro-1H-quinazolin-2-imine
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C10H12ClN3
 1
1
Ki = 15.3 nM
   TI
   LI
   LO
   TS
CP0079728
5-chloro-4-methyl-1,4-dihydroquinazolin-2-amine
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C9H10ClN3
 1
1
Ki = 15.9 nM
   TI
   LI
   LO
   TS
CP0441065
5,6-dichloro-4-ethyl-1,4-dihydroquinazolin-2-amine
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C10H11Cl2N3
 1
1
Ki = 73 nM
   TI
   LI
   LO
   TS
CP0387950
4-(fluoromethyl)-N-[2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl]-N-pyridin-2-ylbicyclo[2.2.2]octane-1-carboxamide
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C28H37FN4O2
 1
1
Ki = 77 nM
   TI
   LI
   LO
   TS
CP0382538
4-(fluoromethyl)-N-[2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl]-N-pyridin-2-ylbicyclo[2.2.1]heptane-1-carboxamide
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C27H35FN4O2
 1
1
Ki = 97 nM
   TI
   LI
   LO
   TS
CP0393077
5-chloro-4-ethyl-1,4-dihydroquinazolin-2-amine
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C10H12ClN3
 1
1
Ki = 97.4 nM
   TI
   LI
   LO
   TS
CP0387949
4-(fluoromethyl)-N-[2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl]-N-pyridin-2-ylcubane-1-carboxamide
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C28H31FN4O2
 1
1
Ki = 132 nM
   TI
   LI
   LO
   TS
CP0288744
5,6-dichloro-1,4-dihydroquinazolin-2-amine
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C8H7Cl2N3
 1
1
Ki = 294 nM
   TI
   LI
   LO
   TS
CP0371440
5-chloro-1,4-dihydroquinazolin-2-amine
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C8H8ClN3
 1
1
Ki = 793 nM
   TI
   LI
   LO
   TS
CP0699181
N-{2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl}-N-(2-pyridinyl)cyclohexane carboxamide trihydrochloride
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C25H37Cl3N4O2
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS