| Compound ID |
Compound Name |
Compound Formula |
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CP0416268
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3-[(1E)-1-[8-[(4-methyl-2-propylbenzimidazol-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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C30H28N4O3
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1
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| 1 |
EC50 = 2.4 nM
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CP0492620
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3-[(1E)-1-[8-[(2-propylbenzimidazol-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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C29H26N4O3
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1
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| 1 |
EC50 = 2.7 nM
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|
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CP0421190
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3-[(1E)-1-[8-[(7-chloro-2-cyclopropylimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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C29H22ClFN4O3
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1
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| 1 |
EC50 = 3.6 nM
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CP0472427
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3-[(1E)-1-[8-[(8-chloro-2-cyclopropylimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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C29H22ClFN4O3
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1
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| 1 |
EC50 = 4.2 nM
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CP0457474
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3-[(1E)-1-[4-fluoro-8-[(2-propylbenzimidazol-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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C29H25FN4O3
|
1
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| 1 |
EC50 = 4.4 nM
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CP0468897
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3-[(1E)-1-[8-[[7-chloro-2-(methoxymethyl)imidazo[1,2-a]pyridin-3-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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C28H22ClFN4O4
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1
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| 1 |
EC50 = 5.3 nM
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|
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CP0391626
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3-[(1E)-1-[8-[[8-chloro-2-(methoxymethyl)imidazo[1,2-a]pyridin-3-yl]methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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|
C28H22ClFN4O4
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1
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| 1 |
EC50 = 7.3 nM
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|
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CP0421187
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3-[(1E)-1-[3-fluoro-8-[(2-propylbenzimidazol-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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C29H25FN4O3
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1
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| 1 |
EC50 = 7.4 nM
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|
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CP0421189
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3-[(1E)-1-[8-[(6-chloro-2-cyclopropylimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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|
C29H22ClFN4O3
|
1
|
| 1 |
EC50 = 11 nM
|
|
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CP0421186
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3-[(1E)-1-[2-fluoro-8-[(2-propylbenzimidazol-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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|
C29H25FN4O3
|
1
|
| 1 |
EC50 = 12 nM
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|
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CP0471829
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3-[(1E)-1-[8-[[4-(2-hydroxypropan-2-yl)-2-propylbenzimidazol-1-yl]methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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|
C32H32N4O4
|
1
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| 1 |
EC50 = 13 nM
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|
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CP0391625
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3-[(1E)-1-[8-[(2-cyclopropyl-7-fluoroimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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C29H22F2N4O3
|
1
|
| 1 |
EC50 = 13 nM
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|
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CP0440167
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3-[(1E)-1-[8-[(2-ethylbenzimidazol-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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|
C28H24N4O3
|
1
|
| 1 |
EC50 = 17 nM
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|
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CP0468896
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3-[(1E)-1-[8-[(2-cyclopropylimidazo[1,2-a]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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|
C29H23FN4O3
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1
|
| 1 |
EC50 = 19 nM
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|
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CP0391624
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3-[(1E)-1-[8-[(2-cyclopropylthieno[3,4-d]imidazol-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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C27H21FN4O3S
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1
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| 1 |
EC50 = 21 nM
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CP0411178
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3-[(1E)-1-[8-[(4-cyclopropyl-10-oxa-3,6-diazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7-tetraen-5-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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C31H25FN4O4
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1
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| 1 |
EC50 = 23 nM
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|
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CP0457475
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3-[(1E)-1-[8-[(4-chloro-2-cyclopropylimidazo[4,5-c]pyridin-1-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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|
C28H21ClFN5O3
|
1
|
| 1 |
EC50 = 24 nM
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|
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CP0421188
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3-[(1E)-1-[8-[(7-chloro-2-cyclopropylimidazo[4,5-b]pyridin-3-yl)methyl]-3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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|
C28H21ClFN5O3
|
1
|
| 1 |
EC50 = 32 nM
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|
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CP0416270
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3-[(1E)-1-[8-[[4-(hydroxymethyl)-2-propylbenzimidazol-1-yl]methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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|
C30H28N4O4
|
1
|
| 1 |
EC50 = 33 nM
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CP0473774
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N-(2-hydroxyethyl)-1-[[(11E)-11-[1-(5-oxo-4H-1,2,4-oxadiazol-3-yl)ethylidene]-6H-benzo[c][1]benzoxepin-8-yl]methyl]-2-propylbenzimidazole-4-carboxamide
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|
C32H31N5O5
|
1
|
| 1 |
EC50 = 57 nM
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CP0158747
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2,4-dichloro-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)benzenesulfonamide
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|
C21H12Cl4N2O3S
|
1
|
| 1 |
EC50 = 59 nM
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CP0467726
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3-[(1E)-1-[8-[(2-ethyl-5,7-dimethylimidazo[4,5-b]pyridin-3-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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|
C29H27N5O3
|
1
|
| 1 |
EC50 = 84 nM
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CP0560150
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3-[(1E)-1-[3-[(4-methyl-2-propylbenzimidazol-1-yl)methyl]-5H-[1]benzoxepino[3,4-b]pyridin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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|
C29H27N5O3
|
1
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| 1 |
EC50 = 86 nM
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CP0416269
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3-[(1E)-1-[8-[(4-phenyl-2-propylimidazol-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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|
C31H28N4O3
|
1
|
| 1 |
EC50 = 151 nM
|
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CP0416271
|
ATx08-001
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C21H23Cl2N3O3S
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1
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| 1 |
EC50 = 163 nM
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CP0492619
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N-[1-[[(11E)-11-[1-(5-oxo-4H-1,2,4-oxadiazol-3-yl)ethylidene]-6H-benzo[c][1]benzoxepin-8-yl]methyl]-2-propylbenzimidazol-4-yl]methanesulfonamide
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C30H29N5O5S
|
1
|
| 1 |
EC50 = 166 nM
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CP0440166
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3-[(1Z)-1-[6-[(2-ethyl-5,7-dimethylimidazo[4,5-b]pyridin-3-yl)methyl]-2-tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaenylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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C30H29N5O2
|
1
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| 1 |
EC50 = 177 nM
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CP0572822
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2-ethyl-5,7-dimethyl-3-[[2-[1-(2H-tetrazol-5-yl)ethyl]-6-tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaenyl]methyl]imidazo[4,5-b]pyridine
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C29H31N7
|
1
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| 1 |
EC50 = 197 nM
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CP0572821
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2-ethyl-5,7-dimethyl-3-[[(2Z)-2-[1-(2H-tetrazol-5-yl)ethylidene]-6-tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaenyl]methyl]imidazo[4,5-b]pyridine
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C29H29N7
|
1
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| 1 |
EC50 = 251 nM
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CP0566187
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3-[(1E)-1-[8-[(2-propyl-4-pyridin-4-ylimidazol-1-yl)methyl]-6H-benzo[c][1]benzoxepin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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|
C30H27N5O3
|
1
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| 1 |
EC50 = 593 nM
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CP0041219
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Actos
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C19H20N2O3S
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1
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| 1 |
EC50 = 2053 nM
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CP0572798
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3-[(1Z)-1-[8-[(4-methyl-2-propylbenzimidazol-1-yl)methyl]-5H-[1]benzoxepino[3,4-b]pyridin-11-ylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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C29H27N5O3
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1
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| 1 |
EC50 = 2194 nM
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CP0876439
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ARHALOFENATE
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C19H17ClF3NO4
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1
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| 1 |
EC50 = 7365 nM
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