Brief Information of the Compound and Protein
Compound Name
3-[(1Z)-1-[6-[(2-ethyl-5,7-dimethylimidazo[4,5-b]pyridin-3-yl)methyl]-2-tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaenylidene]ethyl]-4H-1,2,4-oxadiazol-5-one
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PubChem ID
CID: 136364739
Canonical SMILES
CCc1nc2c(C)cc(C)nc2n1Cc1ccc2c(CCc3ccccc3\C2=C(/C)c2noc(=O)[nH]2)c1
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Compound Formula C30H29N5O2
Compound Structure
Protein Name
Peroxisome proliferator-activated receptor gamma
Protein Classification
Transcription factor
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Nuclear receptor
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Nuclear hormone receptor subfamily 1
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Nuclear hormone receptor subfamily 1 group C
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Nuclear hormone receptor subfamily 1 group C member 3
Uniprot ID
P37231
Gene Name
PPARG
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000065 HEK293-EBNA Homo sapiens (Human)  1
1
EC50 = 177 nM
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